KR101806786B1 - Dpp-iv 억제제의 용도 - Google Patents
Dpp-iv 억제제의 용도 Download PDFInfo
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- KR101806786B1 KR101806786B1 KR1020167024324A KR20167024324A KR101806786B1 KR 101806786 B1 KR101806786 B1 KR 101806786B1 KR 1020167024324 A KR1020167024324 A KR 1020167024324A KR 20167024324 A KR20167024324 A KR 20167024324A KR 101806786 B1 KR101806786 B1 KR 101806786B1
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- KR
- South Korea
- Prior art keywords
- inhibitor
- glucose
- treatment
- inhibitors
- combination
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Abstract
Description
Claims (24)
- 삭제
- 삭제
- 삭제
- 삭제
- 삭제
- 삭제
- 삭제
- 삭제
- 삭제
- 삭제
- 삭제
- 삭제
- 삭제
- 다른 활성 성분의 존재 또는 부재하에 1-[(4-메틸-퀴나졸린-2-일)메틸]-3-메틸-7-(2-부틴-1-일)-8-(3-(R)-아미노-피페리딘-1-일)-크산틴인 DPP-IV 억제제 또는 이의 치료학적으로 활성인 염을 포함하는, 심부전증 환자에서 2형 당뇨병 치료용 약제로서,
상기 DPP-IV 억제제가 2.5mg 또는 5mg의 용량으로 존재하거나 사용되고,
상기 다른 활성 성분이 다른 항당뇨병약 및 심부전증 치료용 활성 성분 중에서 선택되는, 약제. - 삭제
- 삭제
- 삭제
- 삭제
- 삭제
- 제14항에 있어서, 상기 DPP-IV 억제제의 1일 경구 용량이 5mg인, 약제.
- 1-[(4-메틸-퀴나졸린-2-일)메틸]-3-메틸-7-(2-부틴-1-일)-8-(3-(R)-아미노-피페리딘-1-일)-크산틴인 DPP-IV 억제제 또는 이의 치료학적으로 활성인 염을 포함하는, 심부전증 환자에서 2형 당뇨병 치료에 적합한 약제로서,
1-[(4-메틸-퀴나졸린-2-일)메틸]-3-메틸-7-(2-부틴-1-일)-8-(3-(R)-아미노-피페리딘-1-일)-크산틴 5mg이 1일 0.25mg 내지 0.6mg의 용량의 디곡신과 병용 투여되는, 약제. - 삭제
- 1일 1회 5mg의 경구 용량의 1-[(4-메틸-퀴나졸린-2-일)메틸]-3-메틸-7-(2-부틴-1-일)-8-(3-(R)-아미노-피페리딘-1-일)-크산틴의 2형 당뇨병 치료용 약제로서, 상기 약제가 정제 형태인, 약제.
- 제23항에 있어서, 상기 약제가 피복된 정제 형태인, 약제.
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EP06009203.8 | 2006-05-04 | ||
EP06009203 | 2006-05-04 | ||
PCT/EP2007/054270 WO2007128761A2 (de) | 2006-05-04 | 2007-05-03 | Verwendungen von dpp iv inhibitoren |
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KR1020087026975A KR20090021152A (ko) | 2006-05-04 | 2007-05-03 | Dpp-iv 억제제의 용도 |
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US7495005B2 (en) * | 2002-08-22 | 2009-02-24 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Xanthine derivatives, their preparation and their use in pharmaceutical compositions |
US7569574B2 (en) | 2002-08-22 | 2009-08-04 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Purine derivatives, the preparation thereof and their use as pharmaceutical compositions |
US7482337B2 (en) | 2002-11-08 | 2009-01-27 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Xanthine derivatives, the preparation thereof and their use as pharmaceutical compositions |
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