DE60230591D1 - Glykopyranosyloxypyrazolderivate und deren medizinische verwendung - Google Patents

Glykopyranosyloxypyrazolderivate und deren medizinische verwendung

Info

Publication number
DE60230591D1
DE60230591D1 DE60230591T DE60230591T DE60230591D1 DE 60230591 D1 DE60230591 D1 DE 60230591D1 DE 60230591 T DE60230591 T DE 60230591T DE 60230591 T DE60230591 T DE 60230591T DE 60230591 D1 DE60230591 D1 DE 60230591D1
Authority
DE
Germany
Prior art keywords
glycopyranosyloxypyrazole
derivatives
medical use
medical
glycopyranosyloxypyrazole derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE60230591T
Other languages
English (en)
Inventor
Toshihiro Nishimura
Nobuhiko Fushimi
Hideki Fujikura
Kenji Katsuno
Yoshimitsu Komatsu
Masayuki Isaji
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Kissei Pharmaceutical Co Ltd
Original Assignee
Kissei Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kissei Pharmaceutical Co Ltd filed Critical Kissei Pharmaceutical Co Ltd
Application granted granted Critical
Publication of DE60230591D1 publication Critical patent/DE60230591D1/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/203—Monocyclic carbocyclic rings other than cyclohexane rings; Bicyclic carbocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/06—Antigout agents, e.g. antihyperuricemic or uricosuric agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/10—Antioedematous agents; Diuretics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/02—Heterocyclic radicals containing only nitrogen as ring hetero atoms
DE60230591T 2001-02-26 2002-02-26 Glykopyranosyloxypyrazolderivate und deren medizinische verwendung Expired - Lifetime DE60230591D1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2001051278 2001-02-26
JP2001052903 2001-02-27
PCT/JP2002/001707 WO2002068439A1 (fr) 2001-02-26 2002-02-26 Derives de glycopyranosyloxypyrazole et utilisation medicinale de ceux-ci

Publications (1)

Publication Number Publication Date
DE60230591D1 true DE60230591D1 (de) 2009-02-12

Family

ID=26610141

Family Applications (1)

Application Number Title Priority Date Filing Date
DE60230591T Expired - Lifetime DE60230591D1 (de) 2001-02-26 2002-02-26 Glykopyranosyloxypyrazolderivate und deren medizinische verwendung

Country Status (8)

Country Link
US (2) US7087579B2 (de)
EP (1) EP1364957B1 (de)
JP (1) JP4141258B2 (de)
CA (1) CA2438593C (de)
DE (1) DE60230591D1 (de)
ES (1) ES2319263T3 (de)
TW (1) TW593329B (de)
WO (1) WO2002068439A1 (de)

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CN1020944C (zh) 1990-01-30 1993-05-26 阿图尔-费希尔股份公司费希尔厂 紧固件
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AU2002210990A1 (en) * 2000-11-02 2002-05-15 Ajinomoto Co. Inc. Novel pyrazole derivatives and diabetes remedies containing the same
PL209375B1 (pl) * 2000-12-28 2011-08-31 Kissei Pharmaceutical Pochodne glukopiranozyloksypirazolu, kompozycja farmaceutyczna zawierająca takie pochodne i zastosowanie tych pochodnych do wytwarzania kompozycji farmaceutycznej
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EP1389621A4 (de) 2001-04-27 2005-05-11 Ajinomoto Kk N-substituierte pyrazolyl-o-glykosidderivate und diese enthaltendes diabetesmittel
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Also Published As

Publication number Publication date
TW593329B (en) 2004-06-21
ES2319263T3 (es) 2009-05-06
US7087579B2 (en) 2006-08-08
EP1364957A4 (de) 2004-05-06
US7189702B2 (en) 2007-03-13
EP1364957B1 (de) 2008-12-31
EP1364957A1 (de) 2003-11-26
CA2438593A1 (en) 2002-09-06
JP4141258B2 (ja) 2008-08-27
WO2002068439A1 (fr) 2002-09-06
US20060142209A1 (en) 2006-06-29
JPWO2002068439A1 (ja) 2004-06-24
US20040132669A1 (en) 2004-07-08
CA2438593C (en) 2010-09-21

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