SE0001899D0 - New compounds - Google Patents

New compounds

Info

Publication number
SE0001899D0
SE0001899D0 SE0001899A SE0001899A SE0001899D0 SE 0001899 D0 SE0001899 D0 SE 0001899D0 SE 0001899 A SE0001899 A SE 0001899A SE 0001899 A SE0001899 A SE 0001899A SE 0001899 D0 SE0001899 D0 SE 0001899D0
Authority
SE
Sweden
Prior art keywords
compounds
new compounds
preparation
medicament
beta
Prior art date
Application number
SE0001899A
Other languages
English (en)
Inventor
Tjeerd Barf
Original Assignee
Pharmacia & Upjohn Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia & Upjohn Ab filed Critical Pharmacia & Upjohn Ab
Priority to SE0001899A priority Critical patent/SE0001899D0/sv
Publication of SE0001899D0 publication Critical patent/SE0001899D0/sv
Priority to PE2001000450A priority patent/PE20020100A1/es
Priority to EP01934782A priority patent/EP1283832B1/en
Priority to ES01937063T priority patent/ES2333846T3/es
Priority to KR1020027015743A priority patent/KR20030016272A/ko
Priority to NZ522506A priority patent/NZ522506A/en
Priority to EP01934781A priority patent/EP1283831A1/en
Priority to CN01809979A priority patent/CN1430614A/zh
Priority to AU6283101A priority patent/AU6283101A/xx
Priority to AT01934782T priority patent/ATE485283T1/de
Priority to IL15275301A priority patent/IL152753A0/xx
Priority to US10/276,954 priority patent/US7125900B2/en
Priority to PCT/SE2001/001157 priority patent/WO2001090094A1/en
Priority to CA2409697A priority patent/CA2409697C/en
Priority to CN01811609A priority patent/CN1437588A/zh
Priority to US10/296,132 priority patent/US7030135B2/en
Priority to KR1020027015741A priority patent/KR20030011341A/ko
Priority to PCT/SE2001/001155 priority patent/WO2001090090A1/en
Priority to DE60139931T priority patent/DE60139931D1/de
Priority to ARP010102421A priority patent/AR033534A1/es
Priority to JP2001586279A priority patent/JP2003534337A/ja
Priority to BR0111099-3A priority patent/BR0111099A/pt
Priority to CNB018099661A priority patent/CN1188403C/zh
Priority to DE60143293T priority patent/DE60143293D1/de
Priority to DE1283831T priority patent/DE1283831T1/de
Priority to EP01938885A priority patent/EP1283833A1/en
Priority to KR1020027015742A priority patent/KR20030016271A/ko
Priority to CA002408144A priority patent/CA2408144C/en
Priority to IL15267001A priority patent/IL152670A0/xx
Priority to AU2001262831A priority patent/AU2001262831B9/en
Priority to NZ522507A priority patent/NZ522507A/en
Priority to NZ522538A priority patent/NZ522538A/en
Priority to HU0302435A priority patent/HUP0302435A3/hu
Priority to AU6093101A priority patent/AU6093101A/xx
Priority to JP2001586280A priority patent/JP2003534338A/ja
Priority to KR1020027015703A priority patent/KR20030016269A/ko
Priority to IL15279001A priority patent/IL152790A0/xx
Priority to AU6445601A priority patent/AU6445601A/xx
Priority to AU6093201A priority patent/AU6093201A/xx
Priority to IL15266901A priority patent/IL152669A0/xx
Priority to US10/296,553 priority patent/US7618961B2/en
Priority to AU2001262830A priority patent/AU2001262830A1/en
Priority to EP01937063A priority patent/EP1283834B1/en
Priority to JP2001586282A priority patent/JP2003534339A/ja
Priority to PCT/SE2001/001156 priority patent/WO2001090091A1/en
Priority to CNB018116787A priority patent/CN1249039C/zh
Priority to PCT/SE2001/001154 priority patent/WO2001090093A1/en
Priority to JP2001586278A priority patent/JP2003534336A/ja
Priority to AT01937063T priority patent/ATE443055T1/de
Priority to MXPA02011632A priority patent/MXPA02011632A/es
Priority to PCT/SE2001/001158 priority patent/WO2001090092A1/en
Priority to CA002408783A priority patent/CA2408783A1/en
Priority to CA002408142A priority patent/CA2408142C/en
Priority to EA200201271A priority patent/EA005274B1/ru
Priority to NZ522591A priority patent/NZ522591A/en
Priority to US10/296,552 priority patent/US7132436B2/en
Priority to PL36013701A priority patent/PL360137A1/xx
Priority to ZA200209360A priority patent/ZA200209360B/en
Priority to ZA200209364A priority patent/ZA200209364B/en
Priority to ZA200209359A priority patent/ZA200209359B/en
Priority to ZA200209362A priority patent/ZA200209362B/en
Priority to NO20025585A priority patent/NO323831B1/no
Priority to NO20025588A priority patent/NO20025588L/no
Priority to NO20025586A priority patent/NO323832B1/no
Priority to NO20025587A priority patent/NO323779B1/no
Priority to HK03109254A priority patent/HK1056878A1/xx
Priority to US11/289,634 priority patent/US20060160797A1/en
Priority to US11/511,224 priority patent/US20060287374A1/en
Priority to US12/619,216 priority patent/US20100113435A1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/12—Drugs for disorders of the metabolism for electrolyte homeostasis
    • A61P3/14—Drugs for disorders of the metabolism for electrolyte homeostasis for calcium homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A61P31/06—Antibacterial agents for tuberculosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A61P31/08—Antibacterial agents for leprosy
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
    • A61P5/46—Drugs for disorders of the endocrine system of the suprarenal hormones for decreasing, blocking or antagonising the activity of glucocorticosteroids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38—Nitrogen atoms
    • C07D277/50—Nitrogen atoms bound to hetero atoms
    • C07D277/52—Nitrogen atoms bound to hetero atoms to sulfur atoms, e.g. sulfonamides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/84—Naphthothiazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/08—Bridged systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
SE0001899A 2000-05-22 2000-05-22 New compounds SE0001899D0 (sv)

Priority Applications (69)

Application Number Priority Date Filing Date Title
SE0001899A SE0001899D0 (sv) 2000-05-22 2000-05-22 New compounds
PE2001000450A PE20020100A1 (es) 2000-05-22 2001-05-18 DERIVADOS DE 2-SULFONIL AMINO-1,3-TIAZOL COMO INHIBIDORES DE 11-ß-HIDROXI ESTEROIDE DESHIDROGENASA TIPO 1 (11ßHSD1)
EP01934782A EP1283832B1 (en) 2000-05-22 2001-05-22 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
ES01937063T ES2333846T3 (es) 2000-05-22 2001-05-22 Inhibidores de la 11-beta-hidroxiesteroide deshidrogenada tipo1.
KR1020027015743A KR20030016272A (ko) 2000-05-22 2001-05-22 11-베타-히드록시 스테로이드 탈수소효소 타입 1의 억제제
NZ522506A NZ522506A (en) 2000-05-22 2001-05-22 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1, pharmaceutical use and preparation process thereof
EP01934781A EP1283831A1 (en) 2000-05-22 2001-05-22 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
CN01809979A CN1430614A (zh) 2000-05-22 2001-05-22 1型11－β－羟基类固醇脱氢酶的抑制剂
AU6283101A AU6283101A (en) 2000-05-22 2001-05-22 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
AT01934782T ATE485283T1 (de) 2000-05-22 2001-05-22 Inhibitoren der 11-beta-hydroxy-steroid- dehydrogenase des typs 1
IL15275301A IL152753A0 (en) 2000-05-22 2001-05-22 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
US10/276,954 US7125900B2 (en) 2000-05-22 2001-05-22 Inhibitors of 11-β-hydroxy steroid dehydrogenase type 1
PCT/SE2001/001157 WO2001090094A1 (en) 2000-05-22 2001-05-22 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
CA2409697A CA2409697C (en) 2000-05-22 2001-05-22 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
CN01811609A CN1437588A (zh) 2000-05-22 2001-05-22 1型11－β－羟基类固醇脱氢酶抑制剂
US10/296,132 US7030135B2 (en) 2000-05-22 2001-05-22 Inhibitors of 11-β-hydroxy steroid dehydrogenase type 1
KR1020027015741A KR20030011341A (ko) 2000-05-22 2001-05-22 11-베타-히드록시 스테로이드 탈수소효소 타입 1의 억제제
PCT/SE2001/001155 WO2001090090A1 (en) 2000-05-22 2001-05-22 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
DE60139931T DE60139931D1 (de) 2000-05-22 2001-05-22 Inhibitoren der 11-beta-hydroxy-steroid-dehydrogenase des typs 1
ARP010102421A AR033534A1 (es) 2000-05-22 2001-05-22 Derivados de (hetero) arilsulfonil-1,3-tiazol-2-ilamina, utiles como inhibidores de 11-beta-hidroxi esteroide deshidrogenasa tipo 1, procedimiento para prepararlos, el uso de los mismos para la preparacion de medicamentos y las composiciones farmaceuticas que las contienen
JP2001586279A JP2003534337A (ja) 2000-05-22 2001-05-22 １１−β−ヒドロキシステロイドデヒドロゲナーゼ１型の阻害剤
BR0111099-3A BR0111099A (pt) 2000-05-22 2001-05-22 Composto, processo para a preparação de um composto, método para o tratamento ou prevenção de diabetes, sìndrome x, obesidade, glaucoma, hiperlipidemia, hiperglicemia, hiperinsulinemia, osteoporose, tuberculose, demência, depressão, doenças virais e distúrbios inflamatórios, uso de um composto e composição farmacêutica
CNB018099661A CN1188403C (zh) 2000-05-22 2001-05-22 1型11－β－羟基类固醇脱氢酶的抑制剂
DE60143293T DE60143293D1 (de) 2000-05-22 2001-05-22 Inhibitoren der 11-beta-hydroxy-steroid-dehydrogenase des typs 1
DE1283831T DE1283831T1 (de) 2000-05-22 2001-05-22 Inhibitoren der 11-beta-hydroxy-steroid-dehydrogenase des typs 1
EP01938885A EP1283833A1 (en) 2000-05-22 2001-05-22 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
KR1020027015742A KR20030016271A (ko) 2000-05-22 2001-05-22 11-베타-히드록시 스테로이드 탈수소효소 타입 1의 억제제
CA002408144A CA2408144C (en) 2000-05-22 2001-05-22 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
IL15267001A IL152670A0 (en) 2000-05-22 2001-05-22 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
AU2001262831A AU2001262831B9 (en) 2000-05-22 2001-05-22 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
NZ522507A NZ522507A (en) 2000-05-22 2001-05-22 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
NZ522538A NZ522538A (en) 2000-05-22 2001-05-22 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 their use and preparation
HU0302435A HUP0302435A3 (en) 2000-05-22 2001-05-22 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 and pharmaceutical compositions containing them
AU6093101A AU6093101A (en) 2000-05-22 2001-05-22 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
JP2001586280A JP2003534338A (ja) 2000-05-22 2001-05-22 １１−β−ヒドロキシステロイドデヒドロゲナーゼ１型の阻害剤
KR1020027015703A KR20030016269A (ko) 2000-05-22 2001-05-22 11-베타-히드록시 스테로이드 탈수소효소 타입 1의 억제제
IL15279001A IL152790A0 (en) 2000-05-22 2001-05-22 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
AU6445601A AU6445601A (en) 2000-05-22 2001-05-22 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
AU6093201A AU6093201A (en) 2000-05-22 2001-05-22 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
IL15266901A IL152669A0 (en) 2000-05-22 2001-05-22 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
US10/296,553 US7618961B2 (en) 2000-05-22 2001-05-22 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
AU2001262830A AU2001262830A1 (en) 2000-05-22 2001-05-22 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
EP01937063A EP1283834B1 (en) 2000-05-22 2001-05-22 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
JP2001586282A JP2003534339A (ja) 2000-05-22 2001-05-22 １１−ベータヒドロキシステロイドデヒドロゲナーゼタイプ１の阻害剤
PCT/SE2001/001156 WO2001090091A1 (en) 2000-05-22 2001-05-22 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
CNB018116787A CN1249039C (zh) 2000-05-22 2001-05-22 11β－羟基类固醇Ⅰ型脱氢酶抑制剂
PCT/SE2001/001154 WO2001090093A1 (en) 2000-05-22 2001-05-22 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
JP2001586278A JP2003534336A (ja) 2000-05-22 2001-05-22 １１−ベータ−ヒドロキシステロイド・デヒドロゲナーゼタイプ１の阻害因子
AT01937063T ATE443055T1 (de) 2000-05-22 2001-05-22 Inhibitoren der 11-beta-hydroxy-steroid- dehydrogenase des typs 1
MXPA02011632A MXPA02011632A (es) 2000-05-22 2001-05-22 Inhibidores de 11-beta-hidroxiesteroide deshidrogenasa tipo 1.
PCT/SE2001/001158 WO2001090092A1 (en) 2000-05-22 2001-05-22 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
CA002408783A CA2408783A1 (en) 2000-05-22 2001-05-22 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
CA002408142A CA2408142C (en) 2000-05-22 2001-05-22 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
EA200201271A EA005274B1 (ru) 2000-05-22 2001-05-22 Ингибиторы 11-бета-гидроксистероиддегидрогеназы типа 1
NZ522591A NZ522591A (en) 2000-05-22 2001-05-22 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
US10/296,552 US7132436B2 (en) 2000-05-22 2001-05-22 Inhibitors of 11-β-hydroxy steroid dehydrogenase type 1
PL36013701A PL360137A1 (en) 2000-05-22 2001-05-22 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
ZA200209360A ZA200209360B (en) 2000-05-22 2002-11-18 Inhibitors of 11-Beta-hydroxy steroid dehydrogenase type 1.
ZA200209364A ZA200209364B (en) 2000-05-22 2002-11-18 Inhibitors of 11-Beta-hydroxy steroid dehydrogenase type 1.
ZA200209359A ZA200209359B (en) 2000-05-22 2002-11-18 Inhibitors of 11-Beta-hydroxy steroid dehydrogenase type 1.
ZA200209362A ZA200209362B (en) 2000-05-22 2002-11-18 Inhibitors of 11-Beta-hydroxy steroid dehydrogenase type 1.
NO20025585A NO323831B1 (no) 2000-05-22 2002-11-21 Inhibitorer for 11-beta-hydroxy steroid dehydrogenase type 1
NO20025588A NO20025588L (no) 2000-05-22 2002-11-21 Inhibitorer for 11-beta-hydroxy steroid dehydrogenase type 1
NO20025586A NO323832B1 (no) 2000-05-22 2002-11-21 Inhibitorer for 11-beta-hydroxy steroid dehydrogenase type 1
NO20025587A NO323779B1 (no) 2000-05-22 2002-11-21 Inhibitorer for 11-beta-hydroxy steroid dehydrogenase type 1
HK03109254A HK1056878A1 (en) 2000-05-22 2003-12-19 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1.
US11/289,634 US20060160797A1 (en) 2000-05-22 2005-11-30 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
US11/511,224 US20060287374A1 (en) 2000-05-22 2006-08-29 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
US12/619,216 US20100113435A1 (en) 2000-05-22 2009-11-16 Inhibitors of 11-beta-hydroxy steriod dehydrogenase type 1

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