NO20050650L - Fremgangsmate for selektiv fremstilling av aryl-5-tio- -D-aldoheksopyranosider - Google Patents

Fremgangsmate for selektiv fremstilling av aryl-5-tio- -D-aldoheksopyranosider

Info

Publication number
NO20050650L
NO20050650L NO20050650A NO20050650A NO20050650L NO 20050650 L NO20050650 L NO 20050650L NO 20050650 A NO20050650 A NO 20050650A NO 20050650 A NO20050650 A NO 20050650A NO 20050650 L NO20050650 L NO 20050650L
Authority
NO
Norway
Prior art keywords
thio
aryl
general formula
aldohexopyranosides
selective preparation
Prior art date
Application number
NO20050650A
Other languages
English (en)
Inventor
Masakazu Sato
Hiroyuki Kakinuma
Hajime Asanuma
Original Assignee
Taisho Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Taisho Pharmaceutical Co Ltd filed Critical Taisho Pharmaceutical Co Ltd
Publication of NO20050650L publication Critical patent/NO20050650L/no

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/203—Monocyclic carbocyclic rings other than cyclohexane rings; Bicyclic carbocyclic ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/06—Antigout agents, e.g. antihyperuricemic or uricosuric agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
    • A61P5/50—Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings

Abstract

Fremgangsmåte for fremstilling av aryl 5-tio-p-D- aldoheksopyranosid-derivater representert ved. den generelle formel (III), ved å reagere, i samsvar med det følgende skjema, et 5-tio-D-aldoheksopyranose-derivat med den generelle formel (I) med Ar-OH (II) i nærvær av et fosfin representert ved den generelle formel: PR^^R^^R^^ og en azo- reagens representert ved den generelle formel: R^-'--H=H-R^^.
NO20050650A 2002-08-09 2005-02-07 Fremgangsmate for selektiv fremstilling av aryl-5-tio- -D-aldoheksopyranosider NO20050650L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2002233015 2002-08-09
JP2003097839 2003-04-01
PCT/JP2003/010159 WO2004014930A1 (ja) 2002-08-09 2003-08-08 選択的なアリール５−チオ−β−Ｄ−アルドヘキソピラノシドの製造法

Publications (1)

Publication Number Publication Date
NO20050650L true NO20050650L (no) 2005-03-04

Family

ID=31719867

Family Applications (2)

Application Number Title Priority Date Filing Date
NO20043733A NO20043733L (no) 2002-08-09 2004-09-07 Aryl-5-tio-Β-D-glukopyranosid-derivater og legemidler for diabetes inneholdende de samme
NO20050650A NO20050650L (no) 2002-08-09 2005-02-07 Fremgangsmate for selektiv fremstilling av aryl-5-tio- -D-aldoheksopyranosider

Family Applications Before (1)

Application Number Title Priority Date Filing Date
NO20043733A NO20043733L (no) 2002-08-09 2004-09-07 Aryl-5-tio-Β-D-glukopyranosid-derivater og legemidler for diabetes inneholdende de samme

Country Status (19)

Country Link
US (2) US7250522B2 (no)
EP (2) EP1528066A4 (no)
JP (2) JP3813160B2 (no)
KR (2) KR20050056194A (no)
CN (2) CN1312165C (no)
AU (2) AU2003254903B9 (no)
BR (1) BR0310006A (no)
CA (2) CA2493491A1 (no)
HK (2) HK1077582A1 (no)
HR (1) HRP20040814A2 (no)
MX (2) MXPA05000725A (no)
NO (2) NO20043733L (no)
NZ (1) NZ535229A (no)
PL (2) PL372865A1 (no)
RU (1) RU2322449C2 (no)
TW (2) TWI274055B (no)
UA (1) UA77300C2 (no)
WO (2) WO2004014931A1 (no)
ZA (1) ZA200407187B (no)

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KR20050018642A (ko) 2005-02-23
KR100588457B1 (ko) 2006-06-12
TW200406396A (en) 2004-05-01
CN1675233A (zh) 2005-09-28
NO20043733L (no) 2004-10-20
CN100341885C (zh) 2007-10-10
JPWO2004014930A1 (ja) 2005-12-02
WO2004014930A1 (ja) 2004-02-19
NZ535229A (en) 2006-05-26
AU2003254903B2 (en) 2008-07-31
EP1541578A1 (en) 2005-06-15
UA77300C2 (en) 2006-11-15
EP1528066A4 (en) 2007-05-02
US7414072B2 (en) 2008-08-19
HRP20040814A2 (en) 2005-06-30
PL375298A1 (en) 2005-11-28
TW200409778A (en) 2004-06-16
CN1639180A (zh) 2005-07-13
HK1077582A1 (en) 2006-02-17
MXPA04009265A (es) 2005-01-25
BR0310006A (pt) 2005-02-15
US7250522B2 (en) 2007-07-31
US20050209309A1 (en) 2005-09-22
ZA200407187B (en) 2006-02-22
WO2004014931A1 (ja) 2004-02-19
AU2003254903A1 (en) 2004-02-25
TWI274055B (en) 2007-02-21
JP3813160B2 (ja) 2006-08-23
PL372865A1 (en) 2005-08-08
AU2003254903B9 (en) 2008-08-21
EP1528066A1 (en) 2005-05-04
US20050256317A1 (en) 2005-11-17
CN1312165C (zh) 2007-04-25
HK1079532A1 (en) 2006-04-07
RU2004135914A (ru) 2005-05-10
KR20050056194A (ko) 2005-06-14
AU2003254904A1 (en) 2004-02-25
MXPA05000725A (es) 2005-04-08
CA2493491A1 (en) 2004-02-19
CA2478889A1 (en) 2004-02-19
JPWO2004014931A1 (ja) 2005-12-02
RU2322449C2 (ru) 2008-04-20

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