HK1133878A1 - Inhibitors of c-fms kinase c-fms - Google Patents

Inhibitors of c-fms kinase c-fms

Info

Publication number
HK1133878A1
HK1133878A1 HK09112210.0A HK09112210A HK1133878A1 HK 1133878 A1 HK1133878 A1 HK 1133878A1 HK 09112210 A HK09112210 A HK 09112210A HK 1133878 A1 HK1133878 A1 HK 1133878A1
Authority
HK
Hong Kong
Prior art keywords
fms
inhibitors
kinase
fms kinase
Prior art date
Application number
HK09112210.0A
Other languages
English (en)
Chinese (zh)
Inventor
Carl R Illig
Shelley K Ballentine
Jinsheng Chen
Renee Louise Desjarlais
Sanath K Meegalla
Bruce E Tomczuk
Mark Wall
Kenneth Wilson
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of HK1133878A1 publication Critical patent/HK1133878A1/xx

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    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
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    • C12N9/00—Enzymes; Proenzymes; Compositions thereof; Processes for preparing, activating, inhibiting, separating or purifying enzymes
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  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Immunology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Rheumatology (AREA)
  • Zoology (AREA)
  • Genetics & Genomics (AREA)
  • Wood Science & Technology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Diabetes (AREA)
  • Oncology (AREA)
  • Molecular Biology (AREA)
  • Hematology (AREA)
  • Pulmonology (AREA)
  • Cardiology (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Microbiology (AREA)
  • General Engineering & Computer Science (AREA)
  • Vascular Medicine (AREA)
  • Psychiatry (AREA)
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HK09112210.0A 2006-04-20 2009-12-28 Inhibitors of c-fms kinase c-fms HK1133878A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US79366706P 2006-04-20 2006-04-20
PCT/US2007/066868 WO2007124319A1 (en) 2006-04-20 2007-04-18 Inhibitors of c-fms kinase

Publications (1)

Publication Number Publication Date
HK1133878A1 true HK1133878A1 (en) 2010-04-09

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Application Number Title Priority Date Filing Date
HK09112210.0A HK1133878A1 (en) 2006-04-20 2009-12-28 Inhibitors of c-fms kinase c-fms

Country Status (23)

Country Link
US (7) US8722718B2 (xx)
EP (3) EP2016070B1 (xx)
JP (3) JP5331680B2 (xx)
KR (3) KR101367646B1 (xx)
CN (1) CN101472914B (xx)
AR (3) AR060612A1 (xx)
AU (3) AU2007240443B2 (xx)
BR (1) BRPI0710548B8 (xx)
CA (3) CA2649739C (xx)
ES (3) ES2565238T3 (xx)
HK (1) HK1133878A1 (xx)
IL (1) IL194845A (xx)
MX (3) MX2008013531A (xx)
NO (1) NO20084896L (xx)
NZ (3) NZ572070A (xx)
PE (1) PE20080074A1 (xx)
RU (1) RU2475483C2 (xx)
SG (1) SG171593A1 (xx)
TW (3) TWI411612B (xx)
UA (1) UA93085C2 (xx)
UY (1) UY30297A1 (xx)
WO (3) WO2007124319A1 (xx)
ZA (1) ZA200809873B (xx)

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US20060281788A1 (en) * 2005-06-10 2006-12-14 Baumann Christian A Synergistic modulation of flt3 kinase using a flt3 inhibitor and a farnesyl transferase inhibitor
EP2705854A1 (en) * 2006-01-05 2014-03-12 Novartis AG Methods for preventing and treating cancer metastasis and bone loss associated with cancer metastasis
SG171592A1 (en) * 2006-04-20 2011-06-29 Janssen Pharmaceutica Nv Method of inhibiting c-kit kinase
EP2021335B1 (en) 2006-04-20 2011-05-25 Janssen Pharmaceutica N.V. Heterocyclic compounds as inhibitors of c-fms kinase
JP5480619B2 (ja) * 2006-04-20 2014-04-23 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ ｃ−ｆｍｓキナーゼの阻害剤
US8697716B2 (en) 2006-04-20 2014-04-15 Janssen Pharmaceutica Nv Method of inhibiting C-KIT kinase
UA93085C2 (xx) * 2006-04-20 2011-01-10 Янссен Фармацевтика Н.В. Інгібітори c-fms кінази$ингибиторы c-fms киназы
JO3240B1 (ar) * 2007-10-17 2018-03-08 Janssen Pharmaceutica Nv c-fms مثبطات كيناز
US10106798B2 (en) 2010-01-05 2018-10-23 Institut National De La Sante Et De La Recherche Medicale (Inserm) FLT3 receptor antagonists for the treatment or the prevention of pain disorders
HUE045270T2 (hu) 2010-01-05 2019-12-30 Inst Nat Sante Rech Med FLT3 receptor anatgonisták fájdalom rendellenességek kezelésére
ES2622527T3 (es) 2011-05-05 2017-07-06 Novartis Ag Inhibidores de CSF-1R para el tratamiento de tumores de cerebro
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MX2008013531A (es) 2009-01-20
BRPI0710548A2 (pt) 2012-06-05
KR101406877B1 (ko) 2014-06-13
US8722718B2 (en) 2014-05-13
SG171593A1 (en) 2011-06-29
WO2007124322A1 (en) 2007-11-01
US9403804B2 (en) 2016-08-02
US20140329815A1 (en) 2014-11-06
RU2008145763A (ru) 2010-05-27
TWI411612B (zh) 2013-10-11
EP2016074A1 (en) 2009-01-21
CA2649924A1 (en) 2007-11-01
EP2016074B1 (en) 2016-01-13

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