AU2016233568A1 - Alpha-cinnamide compounds and compositions as HDAC8 inhibitors - Google Patents
Alpha-cinnamide compounds and compositions as HDAC8 inhibitors Download PDFInfo
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- AU2016233568A1 AU2016233568A1 AU2016233568A AU2016233568A AU2016233568A1 AU 2016233568 A1 AU2016233568 A1 AU 2016233568A1 AU 2016233568 A AU2016233568 A AU 2016233568A AU 2016233568 A AU2016233568 A AU 2016233568A AU 2016233568 A1 AU2016233568 A1 AU 2016233568A1
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- phenyl
- hydroxy
- acrylamide
- oxoprop
- hydroxyacrylamide
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- C07C259/04—Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups without replacement of the other oxygen atom of the carboxyl group, e.g. hydroxamic acids
- C07C259/06—Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups without replacement of the other oxygen atom of the carboxyl group, e.g. hydroxamic acids having carbon atoms of hydroxamic groups bound to hydrogen atoms or to acyclic carbon atoms
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TWI659949B (zh) | 2016-05-16 | 2019-05-21 | 臺北醫學大學 | 組蛋白去乙醯酶6抑制劑及其用途 |
TW201821105A (zh) | 2016-10-20 | 2018-06-16 | 美商弗瑪治療公司 | 使用hdac11抑制劑之方法 |
CN107056631A (zh) * | 2017-04-14 | 2017-08-18 | 六盘水师范学院 | 一种基于Heck反应的2‑烯基苯胺类化合物制备方法 |
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US11535607B2 (en) | 2018-04-20 | 2022-12-27 | Valo Health, Inc. | Isoindolines as HDAC inhibitors |
KR102055369B1 (ko) * | 2018-08-09 | 2019-12-12 | 충북대학교 산학협력단 | 신규한 3/4-((치환된 벤즈아미도페녹시)메틸)-n-히드록시 벤즈아미드/프로펜아미드 화합물 및 이의 용도 |
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CN113493407A (zh) * | 2020-04-03 | 2021-10-12 | 中国医学科学院药物研究所 | 一种吡啶类化合物及其制法和药物用途 |
CN111728961B (zh) * | 2020-08-05 | 2021-06-15 | 牡丹江医学院 | 一种用于治疗老年痴呆的药物组合物及其用途 |
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KR20230141506A (ko) | 2022-03-31 | 2023-10-10 | 재단법인 대구경북첨단의료산업진흥재단 | 3,4-다이하이드로퀴녹살린-2-카복사미드 유도체 화합물 및 이를 포함하는 암 질환 예방 또는 치료용 약학적 조성물 |
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PH12017501669A1 (en) | 2018-03-19 |
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US20180044282A1 (en) | 2018-02-15 |
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HK1249104A1 (zh) | 2018-10-26 |
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US20220073452A1 (en) | 2022-03-10 |
MA41677A (fr) | 2021-06-02 |
SG11201707418WA (en) | 2017-10-30 |
ECSP17064695A (es) | 2017-10-31 |
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US9745253B2 (en) | 2017-08-29 |
CA2979391C (en) | 2023-10-17 |
US20190241506A1 (en) | 2019-08-08 |
CO2017009298A2 (es) | 2018-01-31 |
CN107531660A (zh) | 2018-01-02 |
US11919839B2 (en) | 2024-03-05 |
EP3932914A1 (en) | 2022-01-05 |
CR20170420A (es) | 2017-10-03 |
BR112017019453A2 (pt) | 2018-05-15 |
US10988441B2 (en) | 2021-04-27 |
TW201639811A (zh) | 2016-11-16 |
US10266487B2 (en) | 2019-04-23 |
PE20171517A1 (es) | 2017-10-20 |
IL254383A0 (en) | 2017-11-30 |
MX2017011778A (es) | 2017-12-04 |
US20180297939A1 (en) | 2018-10-18 |
EA201792028A1 (ru) | 2018-04-30 |
EP3268358A1 (en) | 2018-01-17 |
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