AP2005003341A0 - 2-(1H-indazole-6-ylamino)-benzamide compounds as protein kinases inhibitors useful for the treatmentof ophthalmic diseases - Google Patents
2-(1H-indazole-6-ylamino)-benzamide compounds as protein kinases inhibitors useful for the treatmentof ophthalmic diseasesInfo
- Publication number
- AP2005003341A0 AP2005003341A0 AP2005003341A AP2005003341A AP2005003341A0 AP 2005003341 A0 AP2005003341 A0 AP 2005003341A0 AP 2005003341 A AP2005003341 A AP 2005003341A AP 2005003341 A AP2005003341 A AP 2005003341A AP 2005003341 A0 AP2005003341 A0 AP 2005003341A0
- Authority
- AP
- ARIPO
- Prior art keywords
- treatmentof
- ylamino
- indazole
- protein kinases
- inhibitors useful
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
- A61K31/416—1,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/10—Antioedematous agents; Diuretics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
- C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US43490202P | 2002-12-19 | 2002-12-19 | |
PCT/IB2003/005854 WO2004056806A1 (en) | 2002-12-19 | 2003-12-08 | 2-(1h-indazol-6-ylamino)-benzamide compounds as protein kinases inhibitors useful for the treatment of ophtalmic diseases |
Publications (1)
Publication Number | Publication Date |
---|---|
AP2005003341A0 true AP2005003341A0 (en) | 2005-06-30 |
Family
ID=32682122
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AP2005003341A AP2005003341A0 (en) | 2002-12-19 | 2003-12-08 | 2-(1H-indazole-6-ylamino)-benzamide compounds as protein kinases inhibitors useful for the treatmentof ophthalmic diseases |
Country Status (37)
Country | Link |
---|---|
US (2) | US7053107B2 (nl) |
EP (1) | EP1585743B1 (nl) |
JP (1) | JP3814285B2 (nl) |
KR (1) | KR100730267B1 (nl) |
CN (1) | CN1747950A (nl) |
AP (1) | AP2005003341A0 (nl) |
AR (1) | AR042510A1 (nl) |
AT (1) | ATE362928T1 (nl) |
AU (1) | AU2003286321A1 (nl) |
BR (1) | BR0317548A (nl) |
CA (1) | CA2510850A1 (nl) |
CO (1) | CO5580767A2 (nl) |
CR (1) | CR7882A (nl) |
DE (1) | DE60314013T2 (nl) |
DK (1) | DK1585743T3 (nl) |
EA (1) | EA008501B1 (nl) |
EC (1) | ECSP055858A (nl) |
GT (1) | GT200300294A (nl) |
HR (1) | HRP20050559A2 (nl) |
IS (1) | IS7859A (nl) |
MA (1) | MA27570A1 (nl) |
MX (1) | MXPA05006676A (nl) |
NL (1) | NL1025073C2 (nl) |
NO (1) | NO20053486L (nl) |
NZ (1) | NZ540340A (nl) |
OA (1) | OA12977A (nl) |
PA (1) | PA8592901A1 (nl) |
PE (1) | PE20041006A1 (nl) |
PL (1) | PL377713A1 (nl) |
PT (1) | PT1585743E (nl) |
RS (1) | RS20050430A (nl) |
SI (1) | SI1585743T1 (nl) |
TN (1) | TNSN05164A1 (nl) |
TW (1) | TW200424193A (nl) |
UY (1) | UY28130A1 (nl) |
WO (1) | WO2004056806A1 (nl) |
ZA (1) | ZA200504339B (nl) |
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US8000981B2 (en) | 2005-11-30 | 2011-08-16 | The Invention Science Fund I, Llc | Methods and systems related to receiving nutraceutical associated information |
US8068991B2 (en) * | 2005-11-30 | 2011-11-29 | The Invention Science Fund I, Llc | Systems and methods for transmitting pathogen related information and responding |
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UA75055C2 (uk) | 1999-11-30 | 2006-03-15 | Пфайзер Продактс Інк. | Похідні бензоімідазолу, що використовуються як антипроліферативний засіб, фармацевтична композиція на їх основі |
DE60008206T2 (de) | 1999-11-30 | 2004-12-02 | Pfizer Products Inc., Groton | Chinolinderivate verwendbar zur Hemmung der Farnesyl-Protein Transferase |
YU54202A (sh) * | 2000-01-18 | 2006-01-16 | Agouron Pharmaceuticals Inc. | Jedinjenja indazola, farmaceutske smeše i postupci za stimulisanje i inhibiranje ćelijske proliferacije |
HN2000000266A (es) * | 2000-01-21 | 2001-05-21 | Pfizer Prod Inc | Compuesto anticanceroso y metodo de separacion de enantiomeros util para sintetizar dicho compuesto. |
US6844357B2 (en) * | 2000-05-01 | 2005-01-18 | Pfizer Inc. | Substituted quinolin-2-one derivatives useful as antiproliferative agents |
AR038957A1 (es) | 2001-08-15 | 2005-02-02 | Pharmacia Corp | Terapia de combinacion para el tratamiento del cancer |
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2003
- 2003-12-08 PT PT03777064T patent/PT1585743E/pt unknown
- 2003-12-08 CN CNA2003801096976A patent/CN1747950A/zh active Pending
- 2003-12-08 JP JP2004561821A patent/JP3814285B2/ja not_active Expired - Fee Related
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- 2003-12-08 EA EA200500811A patent/EA008501B1/ru not_active IP Right Cessation
- 2003-12-08 PL PL377713A patent/PL377713A1/pl not_active Application Discontinuation
- 2003-12-08 KR KR1020057011551A patent/KR100730267B1/ko not_active IP Right Cessation
- 2003-12-08 CA CA002510850A patent/CA2510850A1/en not_active Abandoned
- 2003-12-08 DK DK03777064T patent/DK1585743T3/da active
- 2003-12-08 EP EP03777064A patent/EP1585743B1/en not_active Expired - Lifetime
- 2003-12-08 BR BR0317548-0A patent/BR0317548A/pt not_active IP Right Cessation
- 2003-12-08 WO PCT/IB2003/005854 patent/WO2004056806A1/en active IP Right Grant
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- 2003-12-08 AU AU2003286321A patent/AU2003286321A1/en not_active Abandoned
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- 2003-12-08 MX MXPA05006676A patent/MXPA05006676A/es unknown
- 2003-12-08 AP AP2005003341A patent/AP2005003341A0/xx unknown
- 2003-12-08 RS YUP-2005/0430A patent/RS20050430A/sr unknown
- 2003-12-08 DE DE60314013T patent/DE60314013T2/de not_active Expired - Fee Related
- 2003-12-08 SI SI200330833T patent/SI1585743T1/sl unknown
- 2003-12-11 PE PE2003001269A patent/PE20041006A1/es not_active Application Discontinuation
- 2003-12-15 US US10/737,655 patent/US7053107B2/en not_active Expired - Fee Related
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- 2003-12-18 NL NL1025073A patent/NL1025073C2/nl not_active IP Right Cessation
- 2003-12-18 TW TW092135955A patent/TW200424193A/zh unknown
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2005
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- 2005-05-27 ZA ZA200504339A patent/ZA200504339B/en unknown
- 2005-06-15 EC EC2005005858A patent/ECSP055858A/es unknown
- 2005-06-16 HR HR20050559A patent/HRP20050559A2/hr not_active Application Discontinuation
- 2005-06-17 MA MA28348A patent/MA27570A1/fr unknown
- 2005-06-17 TN TNP2005000164A patent/TNSN05164A1/fr unknown
- 2005-06-17 CR CR7882A patent/CR7882A/es not_active Application Discontinuation
- 2005-06-17 CO CO05059483A patent/CO5580767A2/es not_active Application Discontinuation
- 2005-07-18 NO NO20053486A patent/NO20053486L/no not_active Application Discontinuation
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