ZA200504339B - 2-(1H-indazol-6-ylamino)-benzamide compounds as protein kinases inhibitors useful for the treatment of ophtalmic diseases - Google Patents
2-(1H-indazol-6-ylamino)-benzamide compounds as protein kinases inhibitors useful for the treatment of ophtalmic diseases Download PDFInfo
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- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
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- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
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- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
Landscapes
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- Urology & Nephrology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
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JPWO2005094823A1 (ja) * | 2004-03-30 | 2007-08-16 | 協和醗酵工業株式会社 | Flt−3阻害剤 |
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WO2006043172A1 (en) * | 2004-10-19 | 2006-04-27 | Pfizer Inc. | Pharmaceutical compositions and methods for sub-tenon delivery |
CA2586176A1 (en) * | 2004-11-02 | 2006-05-11 | Srinivasan Babu | Methods for preparing indazole compounds |
US20060160863A1 (en) * | 2005-01-05 | 2006-07-20 | Agouron Pharmaceuticals, Inc. | Polymorphic and amorphous forms of 2-{3-[(E)-2-(4,6-dimethyl-pyridin-2-yl)-vinyl]-1H-indazol-6-ylamino}-N-(4-hydroxy-but-2-ynyl)benzamide |
WO2006117666A2 (en) * | 2005-04-29 | 2006-11-09 | Pfizer Inc. | Dosage forms, pharmaceutical compositions and methods for sub-tenon delivery |
US8340944B2 (en) | 2005-11-30 | 2012-12-25 | The Invention Science Fund I, Llc | Computational and/or control systems and methods related to nutraceutical agent selection and dosing |
US10296720B2 (en) | 2005-11-30 | 2019-05-21 | Gearbox Llc | Computational systems and methods related to nutraceuticals |
US7827042B2 (en) | 2005-11-30 | 2010-11-02 | The Invention Science Fund I, Inc | Methods and systems related to transmission of nutraceutical associated information |
US8297028B2 (en) | 2006-06-14 | 2012-10-30 | The Invention Science Fund I, Llc | Individualized pharmaceutical selection and packaging |
US8000981B2 (en) | 2005-11-30 | 2011-08-16 | The Invention Science Fund I, Llc | Methods and systems related to receiving nutraceutical associated information |
US20080103746A1 (en) * | 2005-11-30 | 2008-05-01 | Searete Llc, A Limited Liability Corporation | Systems and methods for pathogen detection and response |
US7974856B2 (en) | 2005-11-30 | 2011-07-05 | The Invention Science Fund I, Llc | Computational systems and methods related to nutraceuticals |
US7927787B2 (en) | 2006-06-28 | 2011-04-19 | The Invention Science Fund I, Llc | Methods and systems for analysis of nutraceutical associated components |
CA2641884A1 (en) * | 2006-02-10 | 2007-08-16 | Summit Corporation Plc | Treatment of duchenne muscular dystrophy |
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CN101677979A (zh) * | 2007-04-19 | 2010-03-24 | 利奥制药有限公司 | Src家族激酶抑制剂 |
RU2494089C2 (ru) | 2007-04-20 | 2013-09-27 | Акьюсела Инк. | Соединения, представляющие собой стиролильные производные, для лечения офтальмических заболеваний и расстройств |
US20090081277A1 (en) * | 2007-09-21 | 2009-03-26 | Allergan, Inc. | Pharmaceutical formulations and methods for treating ocular conditions |
CA2734551A1 (en) | 2008-08-27 | 2010-03-04 | Leo Pharma A/S | Pyridine derivatives as vegfr-2 receptor and protein tyrosine kinase inhibitors |
CN103804349A (zh) * | 2012-11-01 | 2014-05-21 | 杨子娇 | 一类治疗青光眼的化合物及其用途 |
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CN109942544B (zh) * | 2017-12-21 | 2021-06-11 | 中国科学院合肥物质科学研究院 | 一类新型吲唑类衍生物激酶抑制剂 |
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-
2003
- 2003-12-08 NZ NZ540340A patent/NZ540340A/en unknown
- 2003-12-08 AU AU2003286321A patent/AU2003286321A1/en not_active Abandoned
- 2003-12-08 SI SI200330833T patent/SI1585743T1/sl unknown
- 2003-12-08 WO PCT/IB2003/005854 patent/WO2004056806A1/en active IP Right Grant
- 2003-12-08 BR BR0317548-0A patent/BR0317548A/pt not_active IP Right Cessation
- 2003-12-08 PL PL377713A patent/PL377713A1/pl not_active Application Discontinuation
- 2003-12-08 AP AP2005003341A patent/AP2005003341A0/xx unknown
- 2003-12-08 CN CNA2003801096976A patent/CN1747950A/zh active Pending
- 2003-12-08 JP JP2004561821A patent/JP3814285B2/ja not_active Expired - Fee Related
- 2003-12-08 OA OA1200500188A patent/OA12977A/en unknown
- 2003-12-08 DK DK03777064T patent/DK1585743T3/da active
- 2003-12-08 CA CA002510850A patent/CA2510850A1/en not_active Abandoned
- 2003-12-08 KR KR1020057011551A patent/KR100730267B1/ko not_active IP Right Cessation
- 2003-12-08 EA EA200500811A patent/EA008501B1/ru not_active IP Right Cessation
- 2003-12-08 AT AT03777064T patent/ATE362928T1/de not_active IP Right Cessation
- 2003-12-08 RS YUP-2005/0430A patent/RS20050430A/sr unknown
- 2003-12-08 MX MXPA05006676A patent/MXPA05006676A/es unknown
- 2003-12-08 DE DE60314013T patent/DE60314013T2/de not_active Expired - Fee Related
- 2003-12-08 EP EP03777064A patent/EP1585743B1/en not_active Expired - Lifetime
- 2003-12-08 PT PT03777064T patent/PT1585743E/pt unknown
- 2003-12-11 PE PE2003001269A patent/PE20041006A1/es not_active Application Discontinuation
- 2003-12-15 US US10/737,655 patent/US7053107B2/en not_active Expired - Fee Related
- 2003-12-17 PA PA20038592901A patent/PA8592901A1/es unknown
- 2003-12-17 AR ARP030104683A patent/AR042510A1/es unknown
- 2003-12-17 UY UY28130A patent/UY28130A1/es not_active Application Discontinuation
- 2003-12-18 NL NL1025073A patent/NL1025073C2/nl not_active IP Right Cessation
- 2003-12-18 GT GT200300294A patent/GT200300294A/es unknown
- 2003-12-18 TW TW092135955A patent/TW200424193A/zh unknown
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2005
- 2005-05-23 IS IS7859A patent/IS7859A/is unknown
- 2005-05-27 ZA ZA200504339A patent/ZA200504339B/en unknown
- 2005-06-15 EC EC2005005858A patent/ECSP055858A/es unknown
- 2005-06-16 HR HR20050559A patent/HRP20050559A2/hr not_active Application Discontinuation
- 2005-06-17 CO CO05059483A patent/CO5580767A2/es not_active Application Discontinuation
- 2005-06-17 MA MA28348A patent/MA27570A1/fr unknown
- 2005-06-17 TN TNP2005000164A patent/TNSN05164A1/fr unknown
- 2005-06-17 CR CR7882A patent/CR7882A/es not_active Application Discontinuation
- 2005-07-18 NO NO20053486A patent/NO20053486L/no not_active Application Discontinuation
- 2005-12-16 US US11/305,811 patent/US20060160858A1/en not_active Abandoned
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