PL2173752T5 - Sole (r)-3-(4-(7h-pirolo(2,3-d)pirymidyn-4-ylo)-1h-pirazol-1-ilo)-3-cyklopentylopropanonitrylu inhibitora kinazy janusowej - Google Patents

Sole (r)-3-(4-(7h-pirolo(2,3-d)pirymidyn-4-ylo)-1h-pirazol-1-ilo)-3-cyklopentylopropanonitrylu inhibitora kinazy janusowej

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Publication number
PL2173752T5
PL2173752T5 PL08770794.9T PL08770794T PL2173752T5 PL 2173752 T5 PL2173752 T5 PL 2173752T5 PL 08770794 T PL08770794 T PL 08770794T PL 2173752 T5 PL2173752 T5 PL 2173752T5
Authority
PL
Poland
Prior art keywords
cyclopentylpropanenitrile
pyrrolo
pyrazol
pyrimidin
salts
Prior art date
Application number
PL08770794.9T
Other languages
English (en)
Other versions
PL2173752T3 (pl
Inventor
Hui-Yin Li
James D. Rodgers
Original Assignee
Incyte Holdings Corporation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40029273&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PL2173752(T5) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Incyte Holdings Corporation filed Critical Incyte Holdings Corporation
Publication of PL2173752T3 publication Critical patent/PL2173752T3/pl
Publication of PL2173752T5 publication Critical patent/PL2173752T5/pl

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    • A—HUMAN NECESSITIES
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
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    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
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PL08770794.9T 2007-06-13 2008-06-12 Sole (r)-3-(4-(7h-pirolo(2,3-d)pirymidyn-4-ylo)-1h-pirazol-1-ilo)-3-cyklopentylopropanonitrylu inhibitora kinazy janusowej PL2173752T5 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US94370507P 2007-06-13 2007-06-13
PCT/US2008/066662 WO2008157208A2 (en) 2007-06-13 2008-06-12 Salts of the janus kinase inhibitor (r)-3-(4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl)-3-cyclopentylpropanenitrile
EP08770794.9A EP2173752B2 (en) 2007-06-13 2008-06-12 Salts of the janus kinase inhibitor (r)-3-(4-(7h-pyrrolo(2,3-d)pyrimidin-4-yl)-1h-pyrazol-1-yl)-3-cyclopentylpropanenitrile

Publications (2)

Publication Number Publication Date
PL2173752T3 PL2173752T3 (pl) 2014-08-29
PL2173752T5 true PL2173752T5 (pl) 2022-12-05

Family

ID=40029273

Family Applications (3)

Application Number Title Priority Date Filing Date
PL16152794T PL3070090T3 (pl) 2007-06-13 2008-06-12 Zastosowanie soli inhibitora kinazy janusowej (r)-3-(4-(7h-pirolo[2,3- d]pirymidyn-4-ylo)-1h-pirazol-1-ilo)-3-cyklopentylopropanonitrylu
PL13198120.1T PL2740731T3 (pl) 2007-06-13 2008-06-12 Krystaliczne sole (R)-3-(4-(7H-pirolo[2,3-d]pirymidyn-4-ylo)-1H-pirazol-1-ilo)-3-cyklopentylopropanonitrylu jako inhibitory kinazy Janusowej
PL08770794.9T PL2173752T5 (pl) 2007-06-13 2008-06-12 Sole (r)-3-(4-(7h-pirolo(2,3-d)pirymidyn-4-ylo)-1h-pirazol-1-ilo)-3-cyklopentylopropanonitrylu inhibitora kinazy janusowej

Family Applications Before (2)

Application Number Title Priority Date Filing Date
PL16152794T PL3070090T3 (pl) 2007-06-13 2008-06-12 Zastosowanie soli inhibitora kinazy janusowej (r)-3-(4-(7h-pirolo[2,3- d]pirymidyn-4-ylo)-1h-pirazol-1-ilo)-3-cyklopentylopropanonitrylu
PL13198120.1T PL2740731T3 (pl) 2007-06-13 2008-06-12 Krystaliczne sole (R)-3-(4-(7H-pirolo[2,3-d]pirymidyn-4-ylo)-1H-pirazol-1-ilo)-3-cyklopentylopropanonitrylu jako inhibitory kinazy Janusowej

Country Status (42)

Country Link
US (10) US20080312259A1 (pl)
EP (5) EP2173752B2 (pl)
JP (1) JP5475653B2 (pl)
KR (2) KR20150036210A (pl)
CN (2) CN101932582B (pl)
AU (1) AU2008266183B2 (pl)
BR (1) BRPI0814254B8 (pl)
CA (1) CA2689663C (pl)
CO (1) CO6251256A2 (pl)
CR (1) CR11151A (pl)
CU (2) CU24179B1 (pl)
CY (3) CY1115145T1 (pl)
DK (3) DK3070090T3 (pl)
DO (1) DOP2009000280A (pl)
EA (1) EA019784B1 (pl)
EC (1) ECSP099802A (pl)
ES (4) ES2575797T3 (pl)
GE (1) GEP20125533B (pl)
GT (1) GT200900314A (pl)
HK (2) HK1143161A1 (pl)
HR (3) HRP20140541T4 (pl)
HU (2) HUE043732T2 (pl)
IL (5) IL202524A (pl)
LT (1) LT3070090T (pl)
MA (1) MA31517B1 (pl)
ME (1) ME00960B (pl)
MX (2) MX342814B (pl)
MY (1) MY154969A (pl)
NI (1) NI200900216A (pl)
NO (1) NO2019025I1 (pl)
NZ (1) NZ581803A (pl)
PL (3) PL3070090T3 (pl)
PT (2) PT3070090T (pl)
RS (3) RS58449B1 (pl)
SG (3) SG10201912675VA (pl)
SI (3) SI2173752T2 (pl)
SM (1) SMP201000002B (pl)
TN (1) TN2009000514A1 (pl)
TR (1) TR201903488T4 (pl)
UA (1) UA99467C2 (pl)
WO (1) WO2008157208A2 (pl)
ZA (1) ZA200908826B (pl)

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