AR122505A1 - Procesos para preparar un inhibidor de jak1 - Google Patents
Procesos para preparar un inhibidor de jak1Info
- Publication number
- AR122505A1 AR122505A1 ARP210101500A ARP210101500A AR122505A1 AR 122505 A1 AR122505 A1 AR 122505A1 AR P210101500 A ARP210101500 A AR P210101500A AR P210101500 A ARP210101500 A AR P210101500A AR 122505 A1 AR122505 A1 AR 122505A1
- Authority
- AR
- Argentina
- Prior art keywords
- prepare
- processes
- jak1 inhibitor
- compound
- jak1
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
- A61K31/4155—1,2-Diazoles non condensed and containing further heterocyclic rings
-
- B—PERFORMING OPERATIONS; TRANSPORTING
- B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
- B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
- B01J31/00—Catalysts comprising hydrides, coordination complexes or organic compounds
- B01J31/26—Catalysts comprising hydrides, coordination complexes or organic compounds containing in addition, inorganic metal compounds not provided for in groups B01J31/02 - B01J31/24
- B01J31/28—Catalysts comprising hydrides, coordination complexes or organic compounds containing in addition, inorganic metal compounds not provided for in groups B01J31/02 - B01J31/24 of the platinum group metals, iron group metals or copper
Abstract
Reivindicación 1: Un proceso para preparar (base libre del Compuesto 1) o una sal de este, caracterizado porque comprende hacer reaccionar (Compuesto 1x) con (Compuesto 2x) para formar la base libre del Compuesto 1, o una sal de este.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US202063033618P | 2020-06-02 | 2020-06-02 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR122505A1 true AR122505A1 (es) | 2022-09-14 |
Family
ID=76601838
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP210101500A AR122505A1 (es) | 2020-06-02 | 2021-06-02 | Procesos para preparar un inhibidor de jak1 |
Country Status (18)
Country | Link |
---|---|
US (1) | US11685731B2 (es) |
EP (1) | EP4157831A1 (es) |
JP (1) | JP2023528868A (es) |
KR (1) | KR20230027086A (es) |
CN (1) | CN115836065A (es) |
AR (1) | AR122505A1 (es) |
AU (1) | AU2021283271A1 (es) |
BR (1) | BR112022024632A2 (es) |
CA (1) | CA3184275A1 (es) |
CL (1) | CL2022003363A1 (es) |
CO (1) | CO2022017344A2 (es) |
CR (1) | CR20220612A (es) |
EC (1) | ECSP22091930A (es) |
IL (1) | IL298118A (es) |
MX (1) | MX2022015221A (es) |
PE (1) | PE20231102A1 (es) |
TW (1) | TW202210471A (es) |
WO (1) | WO2021247668A1 (es) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
PE20160126A1 (es) | 2013-05-17 | 2016-02-24 | Incyte Corp | Derivados del bipirazol como inhibidores jak |
SG11202007805SA (en) | 2018-02-16 | 2020-09-29 | Incyte Corp | Jak1 pathway inhibitors for the treatment of cytokine-related disorders |
KR20230118118A (ko) | 2020-12-08 | 2023-08-10 | 인사이트 코포레이션 | 백반증의 치료를 위한 jak1 경로 저해제 |
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GB9905075D0 (en) | 1999-03-06 | 1999-04-28 | Zeneca Ltd | Chemical compounds |
GB0004890D0 (en) | 2000-03-01 | 2000-04-19 | Astrazeneca Uk Ltd | Chemical compounds |
CN1321628C (zh) | 2000-06-28 | 2007-06-20 | 史密斯克莱·比奇曼公司 | 湿磨方法 |
DE60230890D1 (de) | 2001-09-19 | 2009-03-05 | Aventis Pharma Sa | Indolizine als kinaseproteinhemmer |
IL161156A0 (en) | 2001-10-30 | 2004-08-31 | Novartis Ag | Staurosporine derivatives as inhibitors of flt3 receptor tyrosine kinase activity |
PE20040522A1 (es) | 2002-05-29 | 2004-09-28 | Novartis Ag | Derivados de diarilurea dependientes de la cinasa de proteina |
GB0215676D0 (en) | 2002-07-05 | 2002-08-14 | Novartis Ag | Organic compounds |
AR042052A1 (es) | 2002-11-15 | 2005-06-08 | Vertex Pharma | Diaminotriazoles utiles como inhibidores de proteinquinasas |
UA80767C2 (en) | 2002-12-20 | 2007-10-25 | Pfizer Prod Inc | Pyrimidine derivatives for the treatment of abnormal cell growth |
GB0305929D0 (en) | 2003-03-14 | 2003-04-23 | Novartis Ag | Organic compounds |
PE20050952A1 (es) | 2003-09-24 | 2005-12-19 | Novartis Ag | Derivados de isoquinolina como inhibidores de b-raf |
AU2005309019A1 (en) | 2004-11-24 | 2006-06-01 | Novartis Ag | Combinations of JAK inhibitors and at least one of Bcr-Abl, Flt-3, FAK or RAF kinase inhibitors |
MY162590A (en) | 2005-12-13 | 2017-06-30 | Incyte Holdings Corp | Heteroaryl substituted pyrrolo[2,3-b] pyridines and pyrrolo[2,3-b] pyrimidines as janus kinase inhibitors |
EP3495369B1 (en) | 2007-06-13 | 2021-10-27 | Incyte Holdings Corporation | Use of salts of the janus kinase inhibitor (r)-3-(4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h- pyrazol-1-yl)-3- cyclopentylpropanenitrile |
CL2008001709A1 (es) | 2007-06-13 | 2008-11-03 | Incyte Corp | Compuestos derivados de pirrolo [2,3-b]pirimidina, moduladores de quinasas jak; composicion farmaceutica; y uso en el tratamiento de enfermedades tales como cancer, psoriasis, artritis reumatoide, entre otras. |
CA2704599C (en) | 2007-11-16 | 2015-05-12 | Incyte Corporation | 4-pyrazolyl-n-arylpyrimidin-2-amines and 4-pyrazolyl-n-heteroarylpyrimidin-2-amines as janus kinase inhibitors |
SI2288610T1 (sl) | 2008-03-11 | 2016-11-30 | Incyte Holdings Corporation | Derivati azetidina in ciklobutana kot inhibitorji jak |
CL2009001884A1 (es) | 2008-10-02 | 2010-05-14 | Incyte Holdings Corp | Uso de 3-ciclopentil-3-[4-(7h-pirrolo[2,3-d]pirimidin-4-il)-1h-pirazol-1-il)propanonitrilo, inhibidor de janus quinasa, y uso de una composición que lo comprende para el tratamiento del ojo seco. |
JOP20190230A1 (ar) | 2009-01-15 | 2017-06-16 | Incyte Corp | طرق لاصلاح مثبطات انزيم jak و المركبات الوسيطة المتعلقة به |
MX2011012262A (es) | 2009-05-22 | 2012-01-25 | Incyte Corp | 3-[4-(7h-pirrolo[2,3-d]pirimidin-4-il)-1h-pirazol-1-il] octano-o heptano-nitrilo como inhibidores de cinasas janus (jak). |
EA025520B1 (ru) | 2009-05-22 | 2017-01-30 | Инсайт Холдингс Корпорейшн | N-(ГЕТЕРО)АРИЛПИРРОЛИДИНОВЫЕ ПРОИЗВОДНЫЕ ПИРАЗОЛ-4-ИЛ-ПИРРОЛО[2,3-d]ПИРИМИДИНОВ И ПИРРОЛ-3-ИЛ-ПИРРОЛО[2,3-d]ПИРИМИДИНОВ В КАЧЕСТВЕ ИНГИБИТОРОВ ЯНУС-КИНАЗЫ |
TW201113285A (en) | 2009-09-01 | 2011-04-16 | Incyte Corp | Heterocyclic derivatives of pyrazol-4-yl-pyrrolo[2,3-d]pyrimidines as janus kinase inhibitors |
PT2486041E (pt) | 2009-10-09 | 2013-11-14 | Incyte Corp | Derivados hidroxilo, ceto e glucuronido de 3-(4-(7h-pirrolo[2,3-d]pirimidin-4-il)-1h-pirazol-1-il)-3-ciclopentil-propanonitrilo |
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SI3354652T1 (sl) | 2010-03-10 | 2020-08-31 | Incyte Holdings Corporation | Derivati piperidin-4-il azetidina kot inhibitorji JAK1 |
KR20130094710A (ko) | 2010-04-14 | 2013-08-26 | 어레이 바이오파마 인크. | Jak 키나아제의 억제제로서 5,7-치환된-이미다조[1,2-c]피리미딘 |
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PE20160126A1 (es) | 2013-05-17 | 2016-02-24 | Incyte Corp | Derivados del bipirazol como inhibidores jak |
CN105209470B (zh) | 2013-05-17 | 2018-02-06 | 豪夫迈·罗氏有限公司 | 用于治疗和预防乙型肝炎病毒感染的6‑桥连的杂芳基二氢嘧啶 |
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JO3603B1 (ar) | 2013-05-17 | 2020-07-05 | Janssen Sciences Ireland Uc | مشتقات سلفامويل بيرولاميد واستخدامها كادوية لمعالجة التهاب الكبد نوع بي |
ES2792549T3 (es) | 2013-08-07 | 2020-11-11 | Incyte Corp | Formas de dosificación de liberación sostenida para un inhibidor de JAK1 |
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AU2015253192B2 (en) | 2014-04-30 | 2019-05-16 | Incyte Holdings Corporation | Processes of preparing a JAK1 inhibitor and new forms thereto |
WO2015184305A1 (en) | 2014-05-30 | 2015-12-03 | Incyte Corporation | TREATMENT OF CHRONIC NEUTROPHILIC LEUKEMIA (CNL) AND ATYPICAL CHRONIC MYELOID LEUKEMIA (aCML) BY INHIBITORS OF JAK1 |
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-
2021
- 2021-06-02 US US17/337,065 patent/US11685731B2/en active Active
- 2021-06-02 BR BR112022024632A patent/BR112022024632A2/pt unknown
- 2021-06-02 AU AU2021283271A patent/AU2021283271A1/en active Pending
- 2021-06-02 TW TW110119976A patent/TW202210471A/zh unknown
- 2021-06-02 PE PE2022002824A patent/PE20231102A1/es unknown
- 2021-06-02 CR CR20220612A patent/CR20220612A/es unknown
- 2021-06-02 CN CN202180048817.4A patent/CN115836065A/zh active Pending
- 2021-06-02 IL IL298118A patent/IL298118A/en unknown
- 2021-06-02 MX MX2022015221A patent/MX2022015221A/es unknown
- 2021-06-02 WO PCT/US2021/035400 patent/WO2021247668A1/en unknown
- 2021-06-02 EP EP21734728.5A patent/EP4157831A1/en active Pending
- 2021-06-02 KR KR1020227045757A patent/KR20230027086A/ko unknown
- 2021-06-02 CA CA3184275A patent/CA3184275A1/en active Pending
- 2021-06-02 JP JP2022574313A patent/JP2023528868A/ja active Pending
- 2021-06-02 AR ARP210101500A patent/AR122505A1/es unknown
-
2022
- 2022-11-29 CL CL2022003363A patent/CL2022003363A1/es unknown
- 2022-12-01 EC ECSENADI202291930A patent/ECSP22091930A/es unknown
- 2022-12-01 CO CONC2022/0017344A patent/CO2022017344A2/es unknown
Also Published As
Publication number | Publication date |
---|---|
TW202210471A (zh) | 2022-03-16 |
IL298118A (en) | 2023-01-01 |
EP4157831A1 (en) | 2023-04-05 |
CN115836065A (zh) | 2023-03-21 |
JP2023528868A (ja) | 2023-07-06 |
CO2022017344A2 (es) | 2023-03-07 |
MX2022015221A (es) | 2023-03-08 |
CR20220612A (es) | 2023-04-11 |
WO2021247668A1 (en) | 2021-12-09 |
AU2021283271A1 (en) | 2022-12-15 |
CA3184275A1 (en) | 2021-12-09 |
US11685731B2 (en) | 2023-06-27 |
PE20231102A1 (es) | 2023-07-19 |
KR20230027086A (ko) | 2023-02-27 |
CL2022003363A1 (es) | 2023-05-19 |
US20210380563A1 (en) | 2021-12-09 |
BR112022024632A2 (pt) | 2023-02-28 |
ECSP22091930A (es) | 2023-02-28 |
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