NO20081592L - Dipeptidylpeptidaseinhibitorer for behandling av diabetes - Google Patents

Dipeptidylpeptidaseinhibitorer for behandling av diabetes

Info

Publication number
NO20081592L
NO20081592L NO20081592A NO20081592A NO20081592L NO 20081592 L NO20081592 L NO 20081592L NO 20081592 A NO20081592 A NO 20081592A NO 20081592 A NO20081592 A NO 20081592A NO 20081592 L NO20081592 L NO 20081592L
Authority
NO
Norway
Prior art keywords
diabetes
treatment
dipeptidyl peptidase
peptidase inhibitors
pharmaceutical compositions
Prior art date
Application number
NO20081592A
Other languages
English (en)
Other versions
NO340910B1 (no
Inventor
Ronald J Christopher
Paul Covington
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37564046&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20081592(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of NO20081592L publication Critical patent/NO20081592L/no
Publication of NO340910B1 publication Critical patent/NO340910B1/no

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/426—1,3-Thiazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22—Hormones
    • A61K38/26—Glucagons
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
    • A61P5/50—Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin

Abstract

Farmasøytiske sammensetninger som innbefatter 2-[6-(3-amino-piperidin-1-yl)-3-metyl-2,4-diokso-3,4-dihydro-2H-pyrimidin-1-ylmetyl]-4-fluor-benzonitril og farmasøytisk akseptable salter derav er tilveiebrakt så vel som kits og fremstilte artikler som innbefatter de farmasøytiske sammensetningene så vel som fremgangsmåter for anvendelse av de farmasøytiske sammensetningene. Sammensetningene kan anvendes for behandling av diabetes.
NO20081592A 2005-09-14 2008-03-31 Farmasøytiske sammensetninger, fremstilt artikkel og anvendelse av de farmasøytiske sammensetninger NO340910B1 (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US71756005P 2005-09-14 2005-09-14
US74728006P 2006-05-15 2006-05-15
PCT/US2006/035958 WO2007033350A1 (en) 2005-09-14 2006-09-13 Dipeptidyl peptidase inhibitors for treating diabetes

Publications (2)

Publication Number Publication Date
NO20081592L true NO20081592L (no) 2008-05-23
NO340910B1 NO340910B1 (no) 2017-07-10

Family

ID=37564046

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20081592A NO340910B1 (no) 2005-09-14 2008-03-31 Farmasøytiske sammensetninger, fremstilt artikkel og anvendelse av de farmasøytiske sammensetninger

Country Status (31)

Country Link
US (3) US20070060530A1 (no)
EP (1) EP1942898B2 (no)
JP (1) JP5027137B2 (no)
KR (1) KR101345316B1 (no)
CN (1) CN101374523B (no)
AR (1) AR055435A1 (no)
AT (1) ATE532518T1 (no)
AU (1) AU2006290205B2 (no)
CA (1) CA2622472C (no)
CR (1) CR9874A (no)
CY (1) CY1112281T1 (no)
DK (1) DK1942898T4 (no)
EA (1) EA015169B1 (no)
ES (1) ES2376351T5 (no)
GE (1) GEP20135838B (no)
HK (1) HK1119086A1 (no)
HR (1) HRP20120004T4 (no)
IL (1) IL190131A (no)
MA (1) MA29795B1 (no)
ME (2) ME02005B (no)
MY (1) MY147393A (no)
NO (1) NO340910B1 (no)
NZ (1) NZ566799A (no)
PE (1) PE20070522A1 (no)
PL (1) PL1942898T5 (no)
PT (1) PT1942898E (no)
RS (1) RS52110B2 (no)
SI (1) SI1942898T2 (no)
TW (1) TWI432200B (no)
WO (1) WO2007033350A1 (no)
ZA (2) ZA200802857B (no)

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