CR20140576A - Sintesis de compuestos heterociclicos - Google Patents

Sintesis de compuestos heterociclicos

Info

Publication number
CR20140576A
CR20140576A CR20140576A CR20140576A CR20140576A CR 20140576 A CR20140576 A CR 20140576A CR 20140576 A CR20140576 A CR 20140576A CR 20140576 A CR20140576 A CR 20140576A CR 20140576 A CR20140576 A CR 20140576A
Authority
CR
Costa Rica
Prior art keywords
synthesis
heterociclic compounds
heterociclic
compounds
intermediaries
Prior art date
Application number
CR20140576A
Other languages
English (en)
Inventor
Prabha N Ibrahim
Original Assignee
Plexxikon Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=48577959&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CR20140576(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Plexxikon Inc filed Critical Plexxikon Inc
Publication of CR20140576A publication Critical patent/CR20140576A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings

Abstract

Intermediarios y procesos útiles para la síntesis sencilla de moléculas biológicamente activas.
CR20140576A 2012-05-31 2014-12-15 Sintesis de compuestos heterociclicos CR20140576A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261653994P 2012-05-31 2012-05-31
US13/793,917 US9150570B2 (en) 2012-05-31 2013-03-11 Synthesis of heterocyclic compounds
PCT/US2013/043400 WO2013181415A1 (en) 2012-05-31 2013-05-30 Synthesis of pyrrolo [2, 3 - b] pyridines

Publications (1)

Publication Number Publication Date
CR20140576A true CR20140576A (es) 2015-01-30

Family

ID=48577959

Family Applications (1)

Application Number Title Priority Date Filing Date
CR20140576A CR20140576A (es) 2012-05-31 2014-12-15 Sintesis de compuestos heterociclicos

Country Status (25)

Country Link
US (2) US9150570B2 (es)
EP (1) EP2861591B1 (es)
JP (1) JP6258301B2 (es)
KR (1) KR102078429B1 (es)
CN (2) CN109608450A (es)
AR (1) AR091159A1 (es)
AU (1) AU2013267325B2 (es)
BR (1) BR112014029454B1 (es)
CA (1) CA2874555C (es)
CL (1) CL2014003228A1 (es)
CR (1) CR20140576A (es)
EA (1) EA027928B1 (es)
EC (1) ECSP14033037A (es)
ES (1) ES2687300T3 (es)
HK (1) HK1206010A1 (es)
IL (1) IL235819B (es)
MX (1) MX2014014465A (es)
MY (1) MY168935A (es)
NZ (1) NZ630453A (es)
PE (1) PE20142335A1 (es)
PH (1) PH12014502613B1 (es)
SG (1) SG11201407851RA (es)
TW (1) TWI603970B (es)
UY (1) UY34825A (es)
WO (1) WO2013181415A1 (es)

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HUE050936T2 (hu) 2015-05-22 2021-01-28 Plexxikon Inc Heterociklusos vegyületek szintézise
US10829484B2 (en) 2015-07-28 2020-11-10 Plexxikon Inc. Compounds and methods for kinase modulation, and indications therefor
TWI732785B (zh) 2015-09-21 2021-07-11 美商普雷辛肯公司 雜環化合物及其用途
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WO2017161045A1 (en) 2016-03-16 2017-09-21 Plexxikon Inc. Compounds and methods for kinase modulation and indications therefore
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US10577366B2 (en) 2017-03-20 2020-03-03 Plexxikon Inc. Crystalline forms of a compound that inhibits bromodomain
WO2018226846A1 (en) 2017-06-07 2018-12-13 Plexxikon Inc. Compounds and methods for kinase modulation
KR102051625B1 (ko) * 2017-06-30 2019-12-02 주식회사 엘지화학 신규한 헤테로 고리 화합물 및 이를 이용한 유기 발광 소자
TWI805599B (zh) 2017-07-25 2023-06-21 美商第一三共公司 激酶調節化合物之調配物
CN111194318B (zh) 2017-10-13 2023-06-09 Opna生物公司 用于调节激酶的化合物固体形式
JP7175309B2 (ja) 2017-10-27 2022-11-18 プレキシコン インコーポレーテッド キナーゼを調節する化合物の製剤
CN112119072A (zh) 2018-03-20 2020-12-22 普莱希科公司 用于ido和tdo调节的化合物和方法,以及其适应症
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