SG11201407851RA - Synthesis of pyrrolo [2, 3 - b] pyridines - Google Patents

Synthesis of pyrrolo [2, 3 - b] pyridines

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Publication number
SG11201407851RA
SG11201407851RA SG11201407851RA SG11201407851RA SG11201407851RA SG 11201407851R A SG11201407851R A SG 11201407851RA SG 11201407851R A SG11201407851R A SG 11201407851RA SG 11201407851R A SG11201407851R A SG 11201407851RA SG 11201407851R A SG11201407851R A SG 11201407851RA
Authority
SG
Singapore
Prior art keywords
international
synthesis
california
pct
applicant
Prior art date
Application number
SG11201407851RA
Inventor
Prabha N Ibrahim
Original Assignee
Plexxikon Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=48577959&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SG11201407851R(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Plexxikon Inc filed Critical Plexxikon Inc
Publication of SG11201407851RA publication Critical patent/SG11201407851RA/en

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings

Abstract

(12) INTERNATIONAL APPLICATION PUBLISHED UNDER THE PATENT COOPERATION TREATY (PCT) (19) World Intellectual Property Organization International Bureau (43) International Publication Date 5 December 2013 (05.12.2013) WIPOIPCT (10) International Publication Number WO 2013/181415 A1 (51) International Patent Classification: C07D 471/04 (2006.01) (21) International Application Number: (22) International Filing Date: (25) Filing Language: (26) Publication Language: PCT/US2013/043400 30 May 2013 (30.05.2013) English English (30) Priority Data: 61/653,994 13/793,917 31 May 2012 (31.05.2012) US 11 March 2013 (11.03.2013) US (71) Applicant: PLEXXIKON INC. [US/US]; 91 Bolivar Drive, Berkeley, California 947140 (US). (72) Inventor: IBRAHIM, Prabha, N.; 3380 Lubich Drive, Mountain View, California 94040 (US). (74) Agents: TANNER, Lorna, L. et al.; Foley & Lardner LLP, 3000 K Street N.W., Suite 600, Washington, DC 20007-5109 (US). (81) Designated States (unless otherwise indicated, for every kind of national protection available)'. AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW. (84) Designated States (unless otherwise indicated, for every kind of regional protection available)'. ARIPO (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, SZ, TZ, UG, ZM, ZW), Eurasian (AM, AZ, BY, KG, KZ, RU, TJ, TM), European (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR), OAPI (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, KM, ML, MR, NE, SN, TD, TG). Declarations under Rule 4.17: — as to applicant's entitlement to apply for and be granted a patent (Rule 4.17(H)) Published: — with international search report (Art. 21(3)) •H •t i-H 00 i-H o CJ 0 (54) Title: SYNTHESIS OF PYRROLO [2, 3 - B] PYRIDINES ^ (57) Abstract: Provided herein are intermediates and processes useful for facile synthesis of biologically active molecules.
SG11201407851RA 2012-05-31 2013-05-30 Synthesis of pyrrolo [2, 3 - b] pyridines SG11201407851RA (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261653994P 2012-05-31 2012-05-31
US13/793,917 US9150570B2 (en) 2012-05-31 2013-03-11 Synthesis of heterocyclic compounds
PCT/US2013/043400 WO2013181415A1 (en) 2012-05-31 2013-05-30 Synthesis of pyrrolo [2, 3 - b] pyridines

Publications (1)

Publication Number Publication Date
SG11201407851RA true SG11201407851RA (en) 2014-12-30

Family

ID=48577959

Family Applications (1)

Application Number Title Priority Date Filing Date
SG11201407851RA SG11201407851RA (en) 2012-05-31 2013-05-30 Synthesis of pyrrolo [2, 3 - b] pyridines

Country Status (25)

Country Link
US (2) US9150570B2 (en)
EP (1) EP2861591B1 (en)
JP (1) JP6258301B2 (en)
KR (1) KR102078429B1 (en)
CN (2) CN109608450A (en)
AR (1) AR091159A1 (en)
AU (1) AU2013267325B2 (en)
BR (1) BR112014029454B1 (en)
CA (1) CA2874555C (en)
CL (1) CL2014003228A1 (en)
CR (1) CR20140576A (en)
EA (1) EA027928B1 (en)
EC (1) ECSP14033037A (en)
ES (1) ES2687300T3 (en)
HK (1) HK1206010A1 (en)
IL (1) IL235819B (en)
MX (1) MX2014014465A (en)
MY (1) MY168935A (en)
NZ (1) NZ630453A (en)
PE (1) PE20142335A1 (en)
PH (1) PH12014502613B1 (en)
SG (1) SG11201407851RA (en)
TW (1) TWI603970B (en)
UY (1) UY34825A (en)
WO (1) WO2013181415A1 (en)

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