ATE253918T1
(de)
|
1999-12-08 |
2003-11-15 |
Centre Nat Rech Scient |
Verwendung von hymenialdisin und dessen derivaten zur herstellung therapeutischer mittel
|
TWI297335B
(en)
|
2001-07-10 |
2008-06-01 |
Synta Pharmaceuticals Corp |
Taxol enhancer compounds
|
TWI332943B
(en)
|
2001-07-10 |
2010-11-11 |
Synta Pharmaceuticals Corp |
Taxol enhancer compounds
|
TWI252847B
(en)
|
2001-07-10 |
2006-04-11 |
Synta Pharmaceuticals Corp |
Synthesis of taxol enhancers
|
TWI329105B
(en)
|
2002-02-01 |
2010-08-21 |
Rigel Pharmaceuticals Inc |
2,4-pyrimidinediamine compounds and their uses
|
TWI330079B
(en)
|
2003-01-15 |
2010-09-11 |
Synta Pharmaceuticals Corp |
Treatment for cancers
|
CN1849318B
(zh)
|
2003-07-30 |
2011-10-12 |
里格尔药品股份有限公司 |
用2,4-嘧啶二胺化合物预防和治疗自体免疫疾病的方法
|
US7557113B2
(en)
*
|
2003-08-26 |
2009-07-07 |
Teijin Pharma Limited |
Substituted pyrrolo[3,2-d]pyrimidine derivatives
|
US7572914B2
(en)
*
|
2003-12-19 |
2009-08-11 |
Takeda Pharmaceutical Company Limited |
Kinase inhibitors
|
AR048454A1
(es)
|
2004-03-30 |
2006-04-26 |
Vertex Pharma |
Azaindoles utiles como inhibidores de las proteinas quinasas jak u otras proteinas quinasas
|
JP5019612B2
(ja)
|
2004-04-02 |
2012-09-05 |
バーテックス ファーマシューティカルズ インコーポレイテッド |
Rockの阻害剤として有用なアザインドールおよび他のプロテインキナーゼ
|
JP2007533753A
(ja)
*
|
2004-04-23 |
2007-11-22 |
タケダ サン ディエゴ インコーポレイテッド |
インドール誘導体及びキナーゼ阻害剤としてのその使用
|
EP1781604B1
(en)
|
2004-06-23 |
2013-08-07 |
Synta Pharmaceuticals Corp. |
Bis(thio-hydrazide amide) salts for treatment of cancers
|
AU2005260689B2
(en)
*
|
2004-06-30 |
2012-05-10 |
Vertex Pharmaceuticals Incorporated |
Azaindoles useful as inhibitors of protein kinases
|
NZ553267A
(en)
|
2004-07-27 |
2010-09-30 |
Sgx Pharmaceuticals Inc |
Pyrrolo-pyridine kinase modulators
|
US7626021B2
(en)
|
2004-07-27 |
2009-12-01 |
Sgx Pharmaceuticals, Inc. |
Fused ring heterocycle kinase modulators
|
MX2007001126A
(es)
|
2004-07-27 |
2007-09-25 |
Sgx Pharmaceuticals Inc |
Moduladores de heterociclo cinasa de anillo fusionado.
|
US7709645B2
(en)
|
2004-07-27 |
2010-05-04 |
Sgx Pharmaceuticals, Inc. |
Pyrrolo-pyridine kinase modulators
|
WO2006023931A2
(en)
*
|
2004-08-18 |
2006-03-02 |
Takeda San Diego, Inc. |
Kinase inhibitors
|
EP1812439B2
(en)
|
2004-10-15 |
2017-12-06 |
Takeda Pharmaceutical Company Limited |
Kinase inhibitors
|
CA2587926A1
(en)
*
|
2004-11-22 |
2006-06-01 |
Vertex Pharmaceuticals Incorporated |
Bicyclic inhibitors or rho kinase
|
WO2006089177A2
(en)
|
2005-02-17 |
2006-08-24 |
Synta Pharmaceuticals Corp. |
Isoxazole combretastin derivatives for the treatment of disorders
|
BRPI0610219A2
(pt)
|
2005-04-15 |
2010-06-08 |
Synta Pharmaceuticals Corp |
métodos de tratamento de um ser humano com cáncer e composição de farmacêutica
|
CN101228161B
(zh)
*
|
2005-05-20 |
2012-10-10 |
沃泰克斯药物股份有限公司 |
适用作蛋白激酶抑制剂的吡咯并吡啶类
|
US20070203161A1
(en)
|
2006-02-24 |
2007-08-30 |
Rigel Pharmaceuticals, Inc. |
Compositions and methods for inhibition of the jak pathway
|
US7491732B2
(en)
|
2005-06-08 |
2009-02-17 |
Rigel Pharmaceuticals, Inc. |
Compositions and methods for inhibition of the JAK pathway
|
EP2251341A1
(en)
*
|
2005-07-14 |
2010-11-17 |
Astellas Pharma Inc. |
Heterocyclic Janus kinase 3 inhibitors
|
KR20080026654A
(ko)
|
2005-07-14 |
2008-03-25 |
아스텔라스세이야쿠 가부시키가이샤 |
헤테로시클릭 야누스 키나제 3 억제제
|
EP1928437A2
(en)
|
2005-08-26 |
2008-06-11 |
Braincells, Inc. |
Neurogenesis by muscarinic receptor modulation
|
EP2258359A3
(en)
|
2005-08-26 |
2011-04-06 |
Braincells, Inc. |
Neurogenesis by muscarinic receptor modulation with sabcomelin
|
WO2007043287A1
(ja)
*
|
2005-09-20 |
2007-04-19 |
Nihon University |
高親和性IgE受容体γ鎖転写調節
|
RU2008117151A
(ru)
*
|
2005-09-30 |
2009-11-10 |
Вертекс Фармасьютикалз Инкорпорейтед (Us) |
Деазапурины, пригодные в качестве ингибиторов янус-киназ
|
US8119655B2
(en)
|
2005-10-07 |
2012-02-21 |
Takeda Pharmaceutical Company Limited |
Kinase inhibitors
|
US8247556B2
(en)
*
|
2005-10-21 |
2012-08-21 |
Amgen Inc. |
Method for preparing 6-substituted-7-aza-indoles
|
JP2009512711A
(ja)
|
2005-10-21 |
2009-03-26 |
ブレインセルス,インコーポレイティド |
Pde阻害による神経新生の調節
|
EP2314289A1
(en)
|
2005-10-31 |
2011-04-27 |
Braincells, Inc. |
Gaba receptor mediated modulation of neurogenesis
|
CA2630079A1
(en)
*
|
2005-11-16 |
2007-05-24 |
Sgx Pharmaceuticals, Inc. |
Pyrazolothiazole protein kinase modulators
|
WO2007076348A2
(en)
*
|
2005-12-23 |
2007-07-05 |
Smithkline Beecham Corporation |
Azaindole inhibitors of aurora kinases
|
CN104650077A
(zh)
|
2006-01-17 |
2015-05-27 |
沃泰克斯药物股份有限公司 |
适用作詹纳斯激酶抑制剂的吖吲哚类
|
WO2007098507A2
(en)
|
2006-02-24 |
2007-08-30 |
Rigel Pharmaceuticals, Inc. |
Compositions and methods for inhibition of the jak pathway
|
US20100216734A1
(en)
|
2006-03-08 |
2010-08-26 |
Braincells, Inc. |
Modulation of neurogenesis by nootropic agents
|
RU2008143361A
(ru)
*
|
2006-04-05 |
2010-05-10 |
Вертекс Фармасьютикалз Инкорпорейтед (Us) |
Деазапурины в качестве ингибиторов янус-киназ
|
WO2007134077A2
(en)
|
2006-05-09 |
2007-11-22 |
Braincells, Inc. |
5 ht receptor mediated neurogenesis
|
WO2007134136A2
(en)
|
2006-05-09 |
2007-11-22 |
Braincells, Inc. |
Neurogenesis by modulating angiotensin
|
EP2046119A2
(en)
*
|
2006-07-07 |
2009-04-15 |
Myriad Genetics, Inc. |
Treatment of psychiatric disorders
|
CA2660836A1
(en)
|
2006-08-07 |
2008-02-21 |
Incyte Corporation |
Triazolotriazines as kinase inhibitors
|
CA2660524A1
(en)
|
2006-08-21 |
2008-02-28 |
Synta Pharmaceutical Corp. |
Compounds for treating proliferative disorders
|
WO2008027445A2
(en)
|
2006-08-31 |
2008-03-06 |
Synta Pharmaceuticals Corp. |
Combination with bis(thiohydrazide amides) for treating cancer
|
EP2068872A1
(en)
|
2006-09-08 |
2009-06-17 |
Braincells, Inc. |
Combinations containing a 4-acylaminopyridine derivative
|
CA2662554A1
(en)
*
|
2006-09-14 |
2008-03-20 |
Synta Pharmaceuticals Corp. |
Compounds for the treatment of angiogenesis
|
US20100184806A1
(en)
|
2006-09-19 |
2010-07-22 |
Braincells, Inc. |
Modulation of neurogenesis by ppar agents
|
MX2009003793A
(es)
|
2006-10-09 |
2009-12-14 |
Takeda Pharmaceutical |
Inhibidores de cinasa.
|
TWI432427B
(zh)
|
2006-10-23 |
2014-04-01 |
Cephalon Inc |
作為ALK及c-MET抑制劑之2,4-二胺基嘧啶之融合雙環衍生物
|
WO2008063888A2
(en)
|
2006-11-22 |
2008-05-29 |
Plexxikon, Inc. |
Compounds modulating c-fms and/or c-kit activity and uses therefor
|
MY188335A
(en)
|
2006-11-22 |
2021-11-30 |
Incyte Holdings Corp |
Imidazotriazines and imidazopyrimidines as kinase inhibitors
|
MX2009006700A
(es)
|
2006-12-21 |
2009-06-30 |
Vertex Pharma |
Derivados de 5-ciano-4-(pirolo)[2,3b]piridina-3-il)-pirimidinas utiles como inhibidores de proteina-cinasas.
|
GB0702265D0
(en)
*
|
2007-02-06 |
2007-03-14 |
Eisai London Res Lab Ltd |
7-Azaindole derivatives
|
AU2008237019A1
(en)
*
|
2007-04-10 |
2008-10-16 |
Sgx Pharmaceuticals, Inc. |
Fused ring heterocycle kinase modulators
|
WO2009012283A1
(en)
|
2007-07-17 |
2009-01-22 |
Plexxikon Inc. |
Compounds and methods for kinase modulation, and indications therefor
|
RS53144B
(en)
*
|
2007-08-22 |
2014-06-30 |
Astrazeneca Ab. |
DERIVATES CYCLOPROPIL AMIDA
|
US8193177B2
(en)
*
|
2007-11-13 |
2012-06-05 |
Angion Biomedica Corp. |
Hepatocyte growth factor pathway activators in fibrotic connective tissue diseases
|
EP2231282A1
(en)
*
|
2008-01-22 |
2010-09-29 |
Merck Patent GmbH |
Protein kinase inhibitors and use thereof
|
PL2265607T3
(pl)
|
2008-02-15 |
2017-07-31 |
Rigel Pharmaceuticals, Inc. |
Związki pirymidyno-2-aminowe i ich zastosowanie jako inhibitory kinaz JAK
|
BRPI0910921B1
(pt)
|
2008-04-16 |
2022-06-21 |
Portola Pharmaceuticals, Inc |
Inibidores de proteína syk quinase, composição farmacêutica, kit e usos dos referidos inibidores
|
US8138339B2
(en)
|
2008-04-16 |
2012-03-20 |
Portola Pharmaceuticals, Inc. |
Inhibitors of protein kinases
|
CA2723185A1
(en)
|
2008-04-22 |
2009-10-29 |
Portola Pharmaceuticals, Inc. |
Inhibitors of protein kinases
|
ES2643363T3
(es)
|
2008-05-21 |
2017-11-22 |
Incyte Holdings Corporation |
Sales de 2-fluoro-N-metil-4-[7-(quinolin-6-il-metil)-imidazo[1,2-b][1,2,4]triazin-2-il]benzamida y procesos relacionados con la preparación de las mismas
|
AR072008A1
(es)
*
|
2008-06-13 |
2010-07-28 |
Merck & Co Inc |
Compuestos heterobiciclicos como agentes de inhibicion de quinasa p38
|
JPWO2009157196A1
(ja)
|
2008-06-25 |
2011-12-08 |
武田薬品工業株式会社 |
アミド化合物
|
EP2328896B1
(en)
*
|
2008-07-23 |
2013-10-23 |
Vertex Pharmaceuticals Incorporated |
Tri-cyclic pyrazolopyridine kinase inhibitors
|
DE102008038221A1
(de)
*
|
2008-08-18 |
2010-02-25 |
Merck Patent Gmbh |
7-Azaindolderivate
|
EP2370424A1
(en)
|
2008-11-10 |
2011-10-05 |
Vertex Pharmaceuticals Incorporated |
Compounds useful as inhibitors of atr kinase
|
EP2379561B1
(en)
|
2008-11-25 |
2015-11-04 |
University Of Rochester |
Mlk inhibitors and methods of use
|
CN102300862B
(zh)
|
2008-12-19 |
2016-11-23 |
沃泰克斯药物股份有限公司 |
用作atr激酶抑制剂的化合物
|
TW201039825A
(en)
|
2009-02-20 |
2010-11-16 |
Astrazeneca Ab |
Cyclopropyl amide derivatives 983
|
WO2010099217A1
(en)
|
2009-02-25 |
2010-09-02 |
Braincells, Inc. |
Modulation of neurogenesis using d-cycloserine combinations
|
CN110269838A
(zh)
|
2009-04-03 |
2019-09-24 |
豪夫迈罗氏公司 |
丙烷-1-磺酸{3-[5-(4-氯-苯基)-1H-吡咯并[2,3-b]吡啶-3-羰基]-2,4-二氟-苯基}-酰胺组合物及其用途
|
ES2604667T3
(es)
|
2009-06-17 |
2017-03-08 |
Vertex Pharmaceuticals Incorporated |
Inhibidores de la replicación de virus de influenza
|
US8329724B2
(en)
|
2009-08-03 |
2012-12-11 |
Hoffmann-La Roche Inc. |
Process for the manufacture of pharmaceutically active compounds
|
MX2012005284A
(es)
|
2009-11-06 |
2012-06-28 |
Plexxikon Inc |
Compuestos y metodos para la modulacion de cinasas. e indicaciones para ello.
|
JP5714030B2
(ja)
|
2010-02-03 |
2015-05-07 |
インサイト コーポレーションIncyte Corporation |
C−Met阻害剤としてのイミダゾ[1,2−b][1,2,4]トリアジン
|
AU2011218492B2
(en)
|
2010-02-18 |
2014-11-13 |
Astrazeneca Ab |
New crystalline form of a cyclopropyl benzamide derivative
|
EP2536701A4
(en)
*
|
2010-02-18 |
2014-05-07 |
Astrazeneca Ab |
SOLID FORMS WITH A CYCLOPROPYLAMID DERIVATIVE
|
JP2013526538A
(ja)
|
2010-05-12 |
2013-06-24 |
バーテックス ファーマシューティカルズ インコーポレイテッド |
Atrキナーゼ阻害剤として有用な化合物
|
JP5856151B2
(ja)
|
2010-05-12 |
2016-02-09 |
バーテックス ファーマシューティカルズ インコーポレイテッドVertex Pharmaceuticals Incorporated |
Atrキナーゼ阻害剤として有用な2−アミノピリジン誘導体
|
WO2011143426A1
(en)
|
2010-05-12 |
2011-11-17 |
Vertex Pharmaceuticals Incorporated |
Compounds useful as inhibitors of atr kinase
|
WO2011143419A1
(en)
|
2010-05-12 |
2011-11-17 |
Vertex Pharmaceuticals Incorporated |
Pyrazines useful as inhibitors of atr kinase
|
US9062008B2
(en)
|
2010-05-12 |
2015-06-23 |
Vertex Pharmaceuticals Incorporated |
Compounds useful as inhibitors of ATR kinase
|
EP2569287B1
(en)
|
2010-05-12 |
2014-07-09 |
Vertex Pharmaceuticals Inc. |
Compounds useful as inhibitors of atr kinase
|
EP2571878B1
(en)
|
2010-05-17 |
2018-10-17 |
Incozen Therapeutics Pvt. Ltd. |
Novel 3,5-disubstitued-3h-imidazo[4,5-b]pyridine and 3,5- disubstitued -3h-[1,2,3]triazolo[4,5-b]pyridine compounds as modulators of protein kinases
|
JP6086326B2
(ja)
|
2010-05-24 |
2017-03-01 |
ユニヴァーシティー オブ ロチェスター |
二環式ヘテロアリールキナーゼ阻害剤および使用方法
|
WO2011163527A1
(en)
*
|
2010-06-23 |
2011-12-29 |
Vertex Pharmaceuticals Incorporated |
Pyrrolo- pyrazine derivatives useful as inhibitors of atr kinase
|
JP5760085B2
(ja)
*
|
2010-08-04 |
2015-08-05 |
武田薬品工業株式会社 |
縮合複素環化合物
|
DE102010049877A1
(de)
*
|
2010-11-01 |
2012-05-03 |
Merck Patent Gmbh |
7-((1,2,3)Triazol-4-yl)-pyrrolo(2,3) pyrazinderivate
|
US9102625B2
(en)
|
2010-11-01 |
2015-08-11 |
Portola Pharmaceuticals, Inc. |
Nicotinamides as JAK kinase modulators
|
EP2796456A1
(en)
*
|
2010-12-09 |
2014-10-29 |
Amgen Inc. |
Bicyclic compounds as Pim inhibitors
|
MX2013006836A
(es)
|
2010-12-16 |
2013-09-26 |
Vertex Pharma |
Inhibidores de la replicacion de los virus de la influenza.
|
CA2822062A1
(en)
*
|
2010-12-16 |
2012-06-21 |
Vertex Pharmaceuticals Incorporated |
Inhibitors of influenza viruses replication
|
DE102011008352A1
(de)
*
|
2011-01-12 |
2012-07-12 |
Merck Patent Gmbh |
5-([1,2,3]Triazol-4-yl)-7H-pyrrolo-[2,3-d]pyrimidinderivate
|
AU2012214762B2
(en)
|
2011-02-07 |
2015-08-13 |
Plexxikon Inc. |
Compounds and methods for kinase modulation, and indications therefor
|
TWI558702B
(zh)
|
2011-02-21 |
2016-11-21 |
普雷辛肯公司 |
醫藥活性物質的固態形式
|
EP2688886A1
(en)
|
2011-03-22 |
2014-01-29 |
Amgen Inc. |
Azole compounds as pim inhibitors
|
AU2012240030A1
(en)
|
2011-04-05 |
2013-10-24 |
Vertex Pharmaceuticals Incorporated |
Aminopyrazine compounds useful as inhibitors of TRA kinase
|
BR112013028900A2
(pt)
|
2011-05-10 |
2017-01-03 |
Merck Sharp & Dohe Corp |
Composto, composição farmacêutica, e, método para o tratamento ou a prevenção de doenças
|
JP2014513687A
(ja)
|
2011-05-10 |
2014-06-05 |
メルク・シャープ・アンド・ドーム・コーポレーション |
Syk阻害薬としてのピリジルアミノピリジン
|
US9145391B2
(en)
|
2011-05-10 |
2015-09-29 |
Merck Sharp & Dohme Corp. |
Bipyridylaminopyridines as Syk inhibitors
|
JP2014517079A
(ja)
|
2011-06-22 |
2014-07-17 |
バーテックス ファーマシューティカルズ インコーポレイテッド |
Atrキナーゼ阻害剤として有用な化合物
|
EP2723747A1
(en)
|
2011-06-22 |
2014-04-30 |
Vertex Pharmaceuticals Inc. |
Compounds useful as inhibitors of atr kinase
|
JP2014520161A
(ja)
|
2011-06-22 |
2014-08-21 |
バーテックス ファーマシューティカルズ インコーポレイテッド |
Atrキナーゼ阻害剤として有用な化合物
|
UA118010C2
(uk)
|
2011-08-01 |
2018-11-12 |
Вертекс Фармасьютікалз Інкорпорейтед |
Інгібітори реплікації вірусів грипу
|
ES2632443T3
(es)
*
|
2011-09-22 |
2017-09-13 |
Viiv Healthcare Uk Limited |
Compuestos de pirrolopiridinona y procedimientos de tratamiento del VIH
|
CN106496173A
(zh)
|
2011-09-30 |
2017-03-15 |
沃泰克斯药物股份有限公司 |
用于制备可用作atr激酶抑制剂的化合物的方法
|
US8846686B2
(en)
|
2011-09-30 |
2014-09-30 |
Vertex Pharmaceuticals Incorporated |
Compounds useful as inhibitors of ATR kinase
|
EP2751088B1
(en)
|
2011-09-30 |
2016-04-13 |
Vertex Pharmaceuticals Incorporated |
Compounds useful as inhibitors of atr kinase
|
US8853217B2
(en)
|
2011-09-30 |
2014-10-07 |
Vertex Pharmaceuticals Incorporated |
Compounds useful as inhibitors of ATR kinase
|
RU2018108589A
(ru)
|
2011-09-30 |
2019-02-25 |
Вертекс Фармасьютикалз Инкорпорейтед |
Лечение рака поджелудочной железы и немелкоклеточного рака легкого ингибиторами atr
|
WO2013052394A1
(en)
|
2011-10-05 |
2013-04-11 |
Merck Sharp & Dohme Corp. |
2-pyridyl carboxamide-containing spleen tyrosine kinase (syk) inhibitors
|
EP2763975B1
(en)
|
2011-10-05 |
2016-04-06 |
Merck Sharp & Dohme Corp. |
3-pyridyl carboxamide-containing spleen tyrosine kinase (syk) inhibitors
|
WO2013052391A1
(en)
|
2011-10-05 |
2013-04-11 |
Merck Sharp & Dohme Corp. |
PHENYL CARBOXAMIDE-CONTAINING SPLEEN TYROSINE KINASE (Syk) INHIBITORS
|
US8841449B2
(en)
|
2011-11-09 |
2014-09-23 |
Vertex Pharmaceuticals Incorporated |
Compounds useful as inhibitors of ATR kinase
|
WO2013071094A1
(en)
|
2011-11-09 |
2013-05-16 |
Vertex Pharmaceuticals Incorporated |
Compounds useful as inhibitors of atr kinase
|
WO2013071088A1
(en)
|
2011-11-09 |
2013-05-16 |
Vertex Pharmaceuticals Incorporated |
Compounds useful as inhibitors of atr kinase
|
US8841337B2
(en)
|
2011-11-09 |
2014-09-23 |
Vertex Pharmaceuticals Incorporated |
Compounds useful as inhibitors of ATR kinase
|
US8841450B2
(en)
|
2011-11-09 |
2014-09-23 |
Vertex Pharmaceuticals Incorporated |
Compounds useful as inhibitors of ATR kinase
|
US8877760B2
(en)
|
2011-11-23 |
2014-11-04 |
Portola Pharmaceuticals, Inc. |
Substituted pyrazine-2-carboxamide kinase inhibitors
|
AP3908A
(en)
|
2012-03-30 |
2016-11-24 |
Rhizen Pharmaceuticals Sa |
Novel 3,5-disubstituted-3H-imidazo[4,5-B]pyridine and 3,5-disubstituted-3H-[1,2,3]triazolo [4,5-B] pyridine compounds as modulators of C-met protein kinases
|
PT2833973T
(pt)
|
2012-04-05 |
2017-12-21 |
Vertex Pharma |
Compostos úteis como inibidores da cinase atr e terapias de combinação dos mesmos
|
US9150570B2
(en)
|
2012-05-31 |
2015-10-06 |
Plexxikon Inc. |
Synthesis of heterocyclic compounds
|
BR112014029705A2
(pt)
|
2012-06-01 |
2017-06-27 |
Takeda Pharmaceuticals Co |
composto ou sal, medicamento, métodos para inibir quinase de janus em um mamífero, e para a profilaxia ou tratamento de doenças autoimunes, e, uso de um composto ou sal
|
DK2904406T3
(en)
|
2012-10-04 |
2018-06-18 |
Vertex Pharma |
METHOD OF DETERMINING THE ATR INHIBITION, INCREASED DNA DAMAGE
|
EP2903970A4
(en)
|
2012-10-08 |
2016-11-30 |
Portola Pharm Inc |
SUBSTITUTED PYRIMIDINYL KINASE INHIBITORS
|
EP2909202A1
(en)
|
2012-10-16 |
2015-08-26 |
Vertex Pharmaceuticals Incorporated |
Compounds useful as inhibitors of atr kinase
|
WO2014085795A1
(en)
|
2012-11-30 |
2014-06-05 |
University Of Rochester |
Mixed lineage kinase inhibitors for hiv/aids therapies
|
HUE061909T2
(hu)
|
2012-12-07 |
2023-08-28 |
Vertex Pharma |
Pirazolo[1,5-a]pirimidinek alkalmazása ATR kináz inhibítorként, rákos megbetegedések kezelésére
|
BR112015022643A2
(pt)
*
|
2013-03-12 |
2017-07-18 |
Abbvie Inc |
inibidores diidro-pirrolpiridinona
|
WO2014143240A1
(en)
|
2013-03-15 |
2014-09-18 |
Vertex Pharmaceuticals Incorporated |
Fused pyrazolopyrimidine derivatives useful as inhibitors of atr kinase
|
US9206188B2
(en)
|
2013-04-18 |
2015-12-08 |
Arrien Pharmaceuticals Llc |
Substituted pyrrolo[2,3-b]pyridines as ITK and JAK inhibitors
|
AR096758A1
(es)
*
|
2013-06-28 |
2016-02-03 |
Abbvie Inc |
Inhibidores cristalinos de bromodominios
|
PT3052096T
(pt)
|
2013-10-03 |
2018-04-04 |
Kura Oncology Inc |
Inibidores de erk e métodos de utilização
|
KR102353413B1
(ko)
|
2013-11-13 |
2022-01-21 |
버텍스 파마슈티칼스 인코포레이티드 |
인플루엔자 바이러스 복제 억제제
|
LT3068782T
(lt)
|
2013-11-13 |
2018-09-10 |
Vertex Pharmaceuticals Incorporated |
Gripo virusų replikacijos inhibitorių paruošimo būdai
|
SG11201604519PA
(en)
|
2013-12-06 |
2016-07-28 |
Vertex Pharma |
2-amino-6-fluoro-n-[5-fluoro-pyridin-3-yl]pyrazolo[1,5-a]pyrimidin-3-carboxamide compound useful as atr kinase inhibitor, its preparation, different solid forms and radiolabelled derivatives thereof
|
WO2015095445A1
(en)
|
2013-12-20 |
2015-06-25 |
Merck Sharp & Dohme Corp. |
Thiazole-substituted aminoheteroaryls as spleen tyrosine kinase inhibitors
|
US9783531B2
(en)
|
2013-12-20 |
2017-10-10 |
Merck Sharp & Dohme Corp. |
Thiazole-substituted aminoheteroaryls as spleen tyrosine kinase inhibitors
|
WO2015095444A1
(en)
|
2013-12-20 |
2015-06-25 |
Merck Sharp & Dohme Corp. |
Thiazole-substituted aminoheteroaryls as spleen tyrosine kinase inhibitors
|
BR112016017981B1
(pt)
*
|
2014-02-04 |
2023-01-17 |
Taiho Pharmaceutical Co., Ltd. |
Compostos derivados de azaindola, inibidor de jak3, composição farmacêutica e agente compreendendo ditos compostos, e uso dos mesmos para tratar uma doença que envolve jak3
|
EP3116506B1
(en)
|
2014-03-13 |
2019-04-17 |
Merck Sharp & Dohme Corp. |
2-pyrazine carboxamides as spleen tyrosine kinase inhibitors
|
CA2945263A1
(en)
|
2014-04-09 |
2015-10-15 |
Christopher Rudd |
Use of gsk-3 inhibitors or activators which modulate pd-1 or t-bet expression to modulate t cell immunity
|
WO2015187451A1
(en)
|
2014-06-05 |
2015-12-10 |
Vertex Pharmacetucals Incorporated |
Radiolabelled derivatives of a 2-amino-6-fluoro-n-[5-fluoro-pyridin-3-yl]- pyrazolo[1,5-a]pyrimidin-3-carboxamide compound useful as atr kinase inhibitor, the preparation of said compound and different solid forms thereof
|
EP3157566B1
(en)
|
2014-06-17 |
2019-05-01 |
Vertex Pharmaceuticals Incorporated |
Method for treating cancer using a combination of chk1 and atr inhibitors
|
EP3053927A1
(en)
*
|
2015-02-05 |
2016-08-10 |
Vectura Limited |
Novel polymorphs
|
JP6704416B2
(ja)
|
2015-05-13 |
2020-06-03 |
バーテックス ファーマシューティカルズ インコーポレイテッドVertex Pharmaceuticals Incorporated |
インフルエンザウイルスの複製の阻害剤を調製する方法
|
MA42422A
(fr)
|
2015-05-13 |
2018-05-23 |
Vertex Pharma |
Inhibiteurs de la réplication des virus de la grippe
|
WO2017059357A1
(en)
|
2015-09-30 |
2017-04-06 |
Vertex Pharmaceuticals Incorporated |
Method for treating cancer using a combination of dna damaging agents and atr inhibitors
|
EP3170822A1
(en)
|
2015-11-18 |
2017-05-24 |
AGV Discovery |
Azaindole derivatives and their use as erk kinase inhibitors
|
MD3442972T2
(ro)
*
|
2016-04-15 |
2020-08-31 |
Abbvie Inc |
Inhibitori ai bromodomeniului
|
TW201811799A
(zh)
|
2016-09-09 |
2018-04-01 |
美商英塞特公司 |
吡唑并嘧啶化合物及其用途
|
MX2019002750A
(es)
|
2016-09-09 |
2019-07-04 |
Incyte Corp |
Derivados de pirazolopiridina como moduladores de cinasa 1 progenitora hematopoyetica (hpk1) y usos de los mismos para tratamiento de cancer.
|
US20180072718A1
(en)
|
2016-09-09 |
2018-03-15 |
Incyte Corporation |
Pyrazolopyridine compounds and uses thereof
|
WO2018049191A1
(en)
|
2016-09-09 |
2018-03-15 |
Incyte Corporation |
Pyrazolopyridone derivatives as hpk1 modulators and uses thereof for the treatment of cancer
|
US20180228786A1
(en)
|
2017-02-15 |
2018-08-16 |
Incyte Corporation |
Pyrazolopyridine compounds and uses thereof
|
WO2018217766A1
(en)
|
2017-05-22 |
2018-11-29 |
Whitehead Institute For Biomedical Research |
Kcc2 expression enhancing compounds and uses thereof
|
WO2018226846A1
(en)
*
|
2017-06-07 |
2018-12-13 |
Plexxikon Inc. |
Compounds and methods for kinase modulation
|
WO2019020981A1
(en)
*
|
2017-07-24 |
2019-01-31 |
Redag Crop Protection Ltd. |
PYRAZOLE, ISOTHIAZOLE AND ISOXAZOLE DERIVATIVES USEFUL AS AGRICULTURAL FUNGICIDES
|
US10722495B2
(en)
|
2017-09-08 |
2020-07-28 |
Incyte Corporation |
Cyanoindazole compounds and uses thereof
|
KR20190043437A
(ko)
|
2017-10-18 |
2019-04-26 |
씨제이헬스케어 주식회사 |
단백질 키나제 억제제로서의 헤테로고리 화합물
|
EP3305786A3
(de)
|
2018-01-22 |
2018-07-25 |
Bayer CropScience Aktiengesellschaft |
Kondensierte bicyclische heterocyclen-derivate als schädlingsbekämpfungsmittel
|
US10752635B2
(en)
|
2018-02-20 |
2020-08-25 |
Incyte Corporation |
Indazole compounds and uses thereof
|
US10745388B2
(en)
|
2018-02-20 |
2020-08-18 |
Incyte Corporation |
Indazole compounds and uses thereof
|
MD3755703T2
(ro)
|
2018-02-20 |
2022-10-31 |
Incyte Corp |
Derivați N-(fenil)-2-(fenil)pirimidin-4-carboxamidă și compuși înrudiți ca inhibitori HPK1 pentru tratarea cancerului
|
US11299473B2
(en)
|
2018-04-13 |
2022-04-12 |
Incyte Corporation |
Benzimidazole and indole compounds and uses thereof
|
WO2019238067A1
(en)
*
|
2018-06-13 |
2019-12-19 |
Beigene, Ltd. |
Pyrrolo [2, 3-b] pyridines or pyrrolo [2, 3-b] pyrazines as hpk1 inhibitor and the use thereof
|
US10899755B2
(en)
|
2018-08-08 |
2021-01-26 |
Incyte Corporation |
Benzothiazole compounds and uses thereof
|
JP7399968B2
(ja)
|
2018-09-25 |
2023-12-18 |
インサイト・コーポレイション |
Alk2及び/またはfgfr調節剤としてのピラゾロ[4,3-d]ピリミジン化合物
|
EP3971190A4
(en)
*
|
2019-05-17 |
2023-06-14 |
Voronoi Inc. |
HETEROCYCLICALLY CONDENSED PYRIMIDIDE DERIVATE AND USE THEREOF
|
BR112022002059A2
(pt)
|
2019-08-06 |
2022-06-07 |
Incyte Corp |
Formas sólidas de um inibidor de hpk1
|
CN112625036A
(zh)
*
|
2019-10-08 |
2021-04-09 |
上海海和药物研究开发股份有限公司 |
一类具有brd4抑制活性的化合物、其制备方法及用途
|
EP4212531A1
(en)
|
2022-01-14 |
2023-07-19 |
AGV Discovery |
Azaindole derivatives and their use as erk kinase inhibitors
|