CN101983073B - 与其它抗糖尿病药组合的dpp-iv抑制剂、包含此类制剂的片剂,和其用途和制备方法 - Google Patents
与其它抗糖尿病药组合的dpp-iv抑制剂、包含此类制剂的片剂,和其用途和制备方法 Download PDFInfo
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- CN101983073B CN101983073B CN2009801120281A CN200980112028A CN101983073B CN 101983073 B CN101983073 B CN 101983073B CN 2009801120281 A CN2009801120281 A CN 2009801120281A CN 200980112028 A CN200980112028 A CN 200980112028A CN 101983073 B CN101983073 B CN 101983073B
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- LTXREWYXXSTFRX-QGZVFWFLSA-N Cc1nc(CN(C(c([n]2CC#CC)c(N3C)nc2N(CCC2)C[C@@H]2N)=O)C3=O)nc2ccccc12 Chemical compound Cc1nc(CN(C(c([n]2CC#CC)c(N3C)nc2N(CCC2)C[C@@H]2N)=O)C3=O)nc2ccccc12 LTXREWYXXSTFRX-QGZVFWFLSA-N 0.000 description 1
- QGJUIPDUBHWZPV-SGTAVMJGSA-N N[C@@H](C(CC(C1)C2)(CC1C1)CC21O)C(N([C@@H](C1)[C@@H]1C1)[C@@H]1C#N)=O Chemical compound N[C@@H](C(CC(C1)C2)(CC1C1)CC21O)C(N([C@@H](C1)[C@@H]1C1)[C@@H]1C#N)=O QGJUIPDUBHWZPV-SGTAVMJGSA-N 0.000 description 1
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- A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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- Transplantation (AREA)
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- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
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- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
Description
Claims (51)
Priority Applications (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CN201610649449.XA CN106215190A (zh) | 2008-04-03 | 2009-04-02 | 与其它抗糖尿病药组合的dpp‑iv抑制剂、包含此类制剂的片剂,和其用途和制备方法 |
CN201310013538.1A CN103083672B (zh) | 2008-04-03 | 2009-04-02 | 与其它抗糖尿病药组合的dpp-iv抑制剂、包含此类制剂的片剂,和其用途和制备方法 |
CN202110764372.1A CN113648422A (zh) | 2008-04-03 | 2009-04-02 | 与其它抗糖尿病药组合的dpp-iv抑制剂、包含此类制剂的片剂,和其用途和制备方法 |
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP08154039.5 | 2008-04-03 | ||
EP08154039 | 2008-04-03 | ||
US8734308P | 2008-08-08 | 2008-08-08 | |
US61/087,343 | 2008-08-08 | ||
PCT/EP2009/053978 WO2009121945A2 (en) | 2008-04-03 | 2009-04-02 | New formulations, tablets comprising such formulations, their use and process for their preparation |
Related Child Applications (3)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CN201610649449.XA Division CN106215190A (zh) | 2008-04-03 | 2009-04-02 | 与其它抗糖尿病药组合的dpp‑iv抑制剂、包含此类制剂的片剂,和其用途和制备方法 |
CN202110764372.1A Division CN113648422A (zh) | 2008-04-03 | 2009-04-02 | 与其它抗糖尿病药组合的dpp-iv抑制剂、包含此类制剂的片剂,和其用途和制备方法 |
CN201310013538.1A Division CN103083672B (zh) | 2008-04-03 | 2009-04-02 | 与其它抗糖尿病药组合的dpp-iv抑制剂、包含此类制剂的片剂,和其用途和制备方法 |
Publications (2)
Publication Number | Publication Date |
---|---|
CN101983073A CN101983073A (zh) | 2011-03-02 |
CN101983073B true CN101983073B (zh) | 2013-06-26 |
Family
ID=39714040
Family Applications (4)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CN202110764372.1A Pending CN113648422A (zh) | 2008-04-03 | 2009-04-02 | 与其它抗糖尿病药组合的dpp-iv抑制剂、包含此类制剂的片剂,和其用途和制备方法 |
CN201610649449.XA Pending CN106215190A (zh) | 2008-04-03 | 2009-04-02 | 与其它抗糖尿病药组合的dpp‑iv抑制剂、包含此类制剂的片剂,和其用途和制备方法 |
CN201310013538.1A Active CN103083672B (zh) | 2008-04-03 | 2009-04-02 | 与其它抗糖尿病药组合的dpp-iv抑制剂、包含此类制剂的片剂,和其用途和制备方法 |
CN2009801120281A Active CN101983073B (zh) | 2008-04-03 | 2009-04-02 | 与其它抗糖尿病药组合的dpp-iv抑制剂、包含此类制剂的片剂,和其用途和制备方法 |
Family Applications Before (3)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CN202110764372.1A Pending CN113648422A (zh) | 2008-04-03 | 2009-04-02 | 与其它抗糖尿病药组合的dpp-iv抑制剂、包含此类制剂的片剂,和其用途和制备方法 |
CN201610649449.XA Pending CN106215190A (zh) | 2008-04-03 | 2009-04-02 | 与其它抗糖尿病药组合的dpp‑iv抑制剂、包含此类制剂的片剂,和其用途和制备方法 |
CN201310013538.1A Active CN103083672B (zh) | 2008-04-03 | 2009-04-02 | 与其它抗糖尿病药组合的dpp-iv抑制剂、包含此类制剂的片剂,和其用途和制备方法 |
Country Status (26)
Country | Link |
---|---|
US (9) | US9155705B2 (zh) |
EP (3) | EP4144374A1 (zh) |
JP (2) | JP5588428B2 (zh) |
KR (3) | KR101611314B1 (zh) |
CN (4) | CN113648422A (zh) |
AR (1) | AR071175A1 (zh) |
AU (1) | AU2009232043B2 (zh) |
BR (1) | BRPI0911273B8 (zh) |
CA (1) | CA2720450C (zh) |
CO (1) | CO6251277A2 (zh) |
DK (1) | DK2285410T3 (zh) |
EA (2) | EA038435B1 (zh) |
EC (1) | ECSP10010489A (zh) |
ES (1) | ES2696124T3 (zh) |
HK (1) | HK1149485A1 (zh) |
IL (2) | IL207497A0 (zh) |
MA (1) | MA32200B1 (zh) |
MX (2) | MX351232B (zh) |
NZ (1) | NZ587747A (zh) |
PE (2) | PE20091730A1 (zh) |
PL (1) | PL2285410T3 (zh) |
TW (2) | TW201509941A (zh) |
UA (1) | UA104136C2 (zh) |
UY (1) | UY31747A (zh) |
WO (1) | WO2009121945A2 (zh) |
ZA (1) | ZA201005664B (zh) |
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