YU44900A - Derivati 2-(purin-9-il)tetrahidrofuran-3,4-diola - Google Patents

Derivati 2-(purin-9-il)tetrahidrofuran-3,4-diola

Info

Publication number
YU44900A
YU44900A YU44900A YU44900A YU44900A YU 44900 A YU44900 A YU 44900A YU 44900 A YU44900 A YU 44900A YU 44900 A YU44900 A YU 44900A YU 44900 A YU44900 A YU 44900A
Authority
YU
Yugoslavia
Prior art keywords
purin
tetrahydrofuran
diol derivatives
diol
derivatives
Prior art date
Application number
YU44900A
Other languages
English (en)
Inventor
Chuen Chan
Richard Peter Charles Cousins
Brian Cox
Original Assignee
Glaxo Group Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Limited filed Critical Glaxo Group Limited
Priority claimed from GBGB9802066.2A external-priority patent/GB9802066D0/en
Priority claimed from GBGB9813528.8A external-priority patent/GB9813528D0/en
Publication of YU44900A publication Critical patent/YU44900A/sh

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16—Purine radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A61K31/706—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
    • A61K31/7064—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
    • A61K31/7076—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines containing purines, e.g. adenosine, adenylic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

Abstract

U skladu sa ovim pronalaskom daju se nova jedinjenja formule (I) gde su R1, R2 i R3 opisani u prijavi, postupci za njihovo dobijanje, formulacije koje ih sadrže i njihova upotreba za proizvodnju leka za lečenje inflamatornih bolesti.[There are provided according to the invention, novel compounds of formula (I) wherein R1, R2 and R3 are as described in the specification, processes for preparing them, formulations containing them and their use in therapy for the treatment of inflammatory diseases.
YU44900A 1998-01-31 1998-01-31 Derivati 2-(purin-9-il)tetrahidrofuran-3,4-diola YU44900A (sh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9802066.2A GB9802066D0 (en) 1998-01-31 1998-01-31 Chemical compounds
GBGB9813528.8A GB9813528D0 (en) 1998-06-23 1998-06-23 Chemical compounds

Publications (1)

Publication Number Publication Date
YU44900A true YU44900A (sh) 2003-01-31

Family

ID=26313042

Family Applications (1)

Application Number Title Priority Date Filing Date
YU44900A YU44900A (sh) 1998-01-31 1998-01-31 Derivati 2-(purin-9-il)tetrahidrofuran-3,4-diola

Country Status (39)

Country Link
US (1) US6762170B1 (sh)
EP (1) EP1051425B1 (sh)
JP (1) JP2002501928A (sh)
KR (1) KR20010034473A (sh)
CN (1) CN1289338A (sh)
AP (1) AP2000001875A0 (sh)
AR (1) AR014508A1 (sh)
AT (1) ATE226957T1 (sh)
AU (1) AU757183B2 (sh)
BG (1) BG63783B1 (sh)
BR (1) BR9907270A (sh)
CA (1) CA2318278A1 (sh)
CO (1) CO4980872A1 (sh)
DE (1) DE69903708T2 (sh)
DK (1) DK1051425T3 (sh)
EA (1) EA003194B1 (sh)
EE (1) EE200000441A (sh)
ES (1) ES2186330T3 (sh)
GE (1) GEP20022839B (sh)
HK (1) HK1030611A1 (sh)
HR (1) HRP20000511A2 (sh)
HU (1) HUP0101305A3 (sh)
ID (1) ID26326A (sh)
IL (1) IL137042A0 (sh)
IS (1) IS5550A (sh)
MA (1) MA26601A1 (sh)
NO (1) NO20003867D0 (sh)
NZ (1) NZ505452A (sh)
OA (1) OA11447A (sh)
PE (1) PE20000280A1 (sh)
PL (1) PL342670A1 (sh)
PT (1) PT1051425E (sh)
SI (1) SI1051425T1 (sh)
SK (1) SK11192000A3 (sh)
SV (1) SV1999000009A (sh)
TR (1) TR200002218T2 (sh)
TW (1) TW434250B (sh)
WO (1) WO1999038877A2 (sh)
YU (1) YU44900A (sh)

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GB0424284D0 (en) 2004-11-02 2004-12-01 Novartis Ag Organic compounds
GB0426164D0 (en) 2004-11-29 2004-12-29 Novartis Ag Organic compounds
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GB0601951D0 (en) 2006-01-31 2006-03-15 Novartis Ag Organic compounds
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Also Published As

Publication number Publication date
BG104729A (en) 2001-04-30
EP1051425B1 (en) 2002-10-30
TW434250B (en) 2001-05-16
WO1999038877A3 (en) 1999-09-30
WO1999038877A2 (en) 1999-08-05
BG63783B1 (bg) 2002-12-29
AU2719799A (en) 1999-08-16
MA26601A1 (fr) 2004-12-20
SI1051425T1 (en) 2003-04-30
HUP0101305A2 (hu) 2002-04-29
EE200000441A (et) 2001-12-17
CN1289338A (zh) 2001-03-28
SK11192000A3 (sk) 2001-06-11
ES2186330T3 (es) 2003-05-01
ATE226957T1 (de) 2002-11-15
NZ505452A (en) 2003-01-31
SV1999000009A (es) 2000-09-05
EP1051425A2 (en) 2000-11-15
BR9907270A (pt) 2000-10-24
DE69903708T2 (de) 2003-07-03
AP2000001875A0 (en) 2000-09-30
HK1030611A1 (en) 2001-05-11
EA200000723A1 (ru) 2001-04-23
TR200002218T2 (tr) 2000-12-21
DK1051425T3 (da) 2003-03-03
PL342670A1 (en) 2001-07-02
IS5550A (is) 2000-06-27
AR014508A1 (es) 2001-02-28
OA11447A (en) 2004-04-29
EA003194B1 (ru) 2003-02-27
PE20000280A1 (es) 2000-03-28
HUP0101305A3 (en) 2002-08-28
AU757183B2 (en) 2003-02-06
JP2002501928A (ja) 2002-01-22
ID26326A (id) 2000-12-14
CO4980872A1 (es) 2000-11-27
NO20003867L (no) 2000-07-28
US6762170B1 (en) 2004-07-13
DE69903708D1 (de) 2002-12-05
HRP20000511A2 (en) 2000-12-31
GEP20022839B (en) 2002-11-25
IL137042A0 (en) 2001-06-14
CA2318278A1 (en) 1999-08-05
KR20010034473A (ko) 2001-04-25
NO20003867D0 (no) 2000-07-28
PT1051425E (pt) 2003-03-31

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