GB0411056D0 - Organic compounds - Google Patents

Organic compounds

Info

Publication number
GB0411056D0
GB0411056D0 GBGB0411056.5A GB0411056A GB0411056D0 GB 0411056 D0 GB0411056 D0 GB 0411056D0 GB 0411056 A GB0411056 A GB 0411056A GB 0411056 D0 GB0411056 D0 GB 0411056D0
Authority
GB
United Kingdom
Prior art keywords
sup
organic compounds
glycopyrrolate
meanings
inflammatory
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
GBGB0411056.5A
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Novartis AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=32607514&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=GB0411056(D0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis AG filed Critical Novartis AG
Priority to GBGB0411056.5A priority Critical patent/GB0411056D0/en
Publication of GB0411056D0 publication Critical patent/GB0411056D0/en
Priority to US11/568,559 priority patent/US20080267886A1/en
Priority to HUE10164976A priority patent/HUE048936T2/en
Priority to SI200532271T priority patent/SI2228064T1/en
Priority to EP10164976.2A priority patent/EP2228064B1/en
Priority to NZ550369A priority patent/NZ550369A/en
Priority to ES10164976T priority patent/ES2775979T3/en
Priority to RU2006144810/15A priority patent/RU2388465C2/en
Priority to LTEP10164976.2T priority patent/LT2228064T/en
Priority to ES05749635T priority patent/ES2370647T3/en
Priority to BRPI0511327A priority patent/BRPI0511327B8/en
Priority to PT05749635T priority patent/PT1755590E/en
Priority to PL10164976T priority patent/PL2228064T3/en
Priority to JP2007517074A priority patent/JP5567252B2/en
Priority to CNA2005800159322A priority patent/CN1953745A/en
Priority to PL05749635T priority patent/PL1755590T3/en
Priority to PCT/EP2005/005354 priority patent/WO2005110402A1/en
Priority to DK05749635.8T priority patent/DK1755590T3/en
Priority to SE05749635T priority patent/SE1755590T5/xx
Priority to KR1020067024115A priority patent/KR101360556B1/en
Priority to SG200904196-3A priority patent/SG153836A1/en
Priority to MXPA06013382A priority patent/MXPA06013382A/en
Priority to KR1020137000008A priority patent/KR20130018429A/en
Priority to CA2563302A priority patent/CA2563302C/en
Priority to PT101649762T priority patent/PT2228064T/en
Priority to EP19180535.7A priority patent/EP3603634A1/en
Priority to AU2005244439A priority patent/AU2005244439C1/en
Priority to SI200531407T priority patent/SI1755590T1/en
Priority to AT05749635T priority patent/ATE521348T1/en
Priority to EP05749635A priority patent/EP1755590B1/en
Priority to DK10164976.2T priority patent/DK2228064T3/en
Priority to ZA200608123A priority patent/ZA200608123B/en
Priority to EC2006006950A priority patent/ECSP066950A/en
Priority to IL179013A priority patent/IL179013A/en
Priority to TNP2006000377A priority patent/TNSN06377A1/en
Priority to MA29475A priority patent/MA28598B1/en
Priority to NO20065787A priority patent/NO334760B1/en
Priority to HK07107762.4A priority patent/HK1105579A1/en
Priority to CY20111101145T priority patent/CY1112086T1/en
Priority to JP2012156212A priority patent/JP2012236833A/en
Priority to US13/862,529 priority patent/US20130237564A1/en
Priority to LTPA2014015C priority patent/LTC1755590I2/en
Priority to HUS1400013C priority patent/HUS1400013I1/en
Priority to CY2014014C priority patent/CY2014014I1/en
Priority to NO2014020C priority patent/NO2014020I1/en
Priority to US14/973,778 priority patent/US20160101097A1/en
Priority to US15/818,991 priority patent/US20180071276A1/en
Priority to US16/429,382 priority patent/US20190282561A1/en
Priority to CY20201100208T priority patent/CY1122863T1/en
Priority to FR20C1018C priority patent/FR20C1018I2/en
Priority to LU00155C priority patent/LUC00155I2/fr
Priority to HUS2000014C priority patent/HUS2000014I1/en
Priority to CY2020013C priority patent/CY2020013I1/en
Priority to LTPA2020509C priority patent/LTC2228064I2/en
Priority to US17/237,350 priority patent/US20210236478A1/en
Ceased legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4704—2-Quinolinones, e.g. carbostyril
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/4015—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil having oxo groups directly attached to the heterocyclic ring, e.g. piracetam, ethosuximide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/402—1-aryl substituted, e.g. piretanide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/428—Thiazoles condensed with carbocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system

Abstract

A pharmaceutical composition containing (A) glycopyrrolate; and (B) a compound of formula Iin free or salt or solvate form, wherein W, R<sup>x</sup>, R<sup>y</sup>, R<sup>1</sup>, R<sup>2</sup>, R<sup>3</sup>, R<sup>4</sup>, R<sup>5</sup>, R<sup>6</sup>and R<sup>7</sup>have the meanings as indicated in the specification, together with at least one pharmaceutically acceptable carrier. The composition is useful in the treatment of inflammatory or obstructive airways diseases.
GBGB0411056.5A 2004-05-18 2004-05-18 Organic compounds Ceased GB0411056D0 (en)

Priority Applications (55)

Application Number Priority Date Filing Date Title
GBGB0411056.5A GB0411056D0 (en) 2004-05-18 2004-05-18 Organic compounds
US11/568,559 US20080267886A1 (en) 2004-05-18 2005-05-17 Combinations of Glycopyrrolate and Beta2 Adrenoceptor Agonists
HUE10164976A HUE048936T2 (en) 2004-05-18 2005-05-17 Pharmaceutical composition containing glycopyrrolate and a beta2 adrenoceptor agonist
SI200532271T SI2228064T1 (en) 2004-05-18 2005-05-17 Pharmaceutical composition containing glycopyrrolate and a beta2 adrenoceptor agonist
EP10164976.2A EP2228064B1 (en) 2004-05-18 2005-05-17 Pharmaceutical composition containing glycopyrrolate and a beta2 adrenoceptor agonist
NZ550369A NZ550369A (en) 2004-05-18 2005-05-17 Combinations of glycopyrrolate and beta2 adrenoceptor agonists
ES10164976T ES2775979T3 (en) 2004-05-18 2005-05-17 Pharmaceutical composition containing glycopyrrolate and a beta-2 adrenergic receptor agonist
RU2006144810/15A RU2388465C2 (en) 2004-05-18 2005-05-17 Combinations of glucopyrrolate and b-2 adrenoceptor antogonists
LTEP10164976.2T LT2228064T (en) 2004-05-18 2005-05-17 Pharmaceutical composition containing glycopyrrolate and a beta2 adrenoceptor agonist
ES05749635T ES2370647T3 (en) 2004-05-18 2005-05-17 COMBINATION OF GLUCOPIRROLATE AND A BETA2 ADRENORECEPTOR AGONIST.
BRPI0511327A BRPI0511327B8 (en) 2004-05-18 2005-05-17 combinations of glycopyrrolate and beta2 adrenoreceptor agonists
PT05749635T PT1755590E (en) 2004-05-18 2005-05-17 Combination of glycopyrrolate and a beta2 adrenoceptor agonist
PL10164976T PL2228064T3 (en) 2004-05-18 2005-05-17 Pharmaceutical composition containing glycopyrrolate and a beta2 adrenoceptor agonist
JP2007517074A JP5567252B2 (en) 2004-05-18 2005-05-17 Combination of glycopyrrolate and beta-2 adrenergic receptor agonist
CNA2005800159322A CN1953745A (en) 2004-05-18 2005-05-17 Combinations of glycopyrrolate and beta2 adrenoceptor agonists
PL05749635T PL1755590T3 (en) 2004-05-18 2005-05-17 Combination of glycopyrrolate and a beta2 adrenoceptor agonist
PCT/EP2005/005354 WO2005110402A1 (en) 2004-05-18 2005-05-17 Combinations of glycopyrrolate and beta2 adrenoceptor agonists
DK05749635.8T DK1755590T3 (en) 2004-05-18 2005-05-17 Combination of glycopyrrolate and a beta2-adrenoceptor agonist
SE05749635T SE1755590T5 (en) 2004-05-18 2005-05-17
KR1020067024115A KR101360556B1 (en) 2004-05-18 2005-05-17 Combinations of glycopyrrolate and beta2 adrenoceptor agonists
SG200904196-3A SG153836A1 (en) 2004-05-18 2005-05-17 Combination of glycopyrrolate and a beta2 adrenoceptor agonist
MXPA06013382A MXPA06013382A (en) 2004-05-18 2005-05-17 Combinations of glycopyrrolate and beta2 adrenoceptor agonists.
KR1020137000008A KR20130018429A (en) 2004-05-18 2005-05-17 Combinations of glycopyrrolate and beta2 adrenoceptor agonists
CA2563302A CA2563302C (en) 2004-05-18 2005-05-17 Combinations of glycopyrrolate and beta2 adrenoceptor agonists
PT101649762T PT2228064T (en) 2004-05-18 2005-05-17 Pharmaceutical composition containing glycopyrrolate and a beta2 adrenoceptor agonist
EP19180535.7A EP3603634A1 (en) 2004-05-18 2005-05-17 Pharmaceutical composition containing glycopyrrolate and a beta2 adrenoceptor agonist
AU2005244439A AU2005244439C1 (en) 2004-05-18 2005-05-17 Combinations of glycopyrrolate and beta2 adrenoceptor agonists
SI200531407T SI1755590T1 (en) 2004-05-18 2005-05-17 Combination of glycopyrrolate and a beta2 adrenoceptor agonist
AT05749635T ATE521348T1 (en) 2004-05-18 2005-05-17 COMBINATION OF GLYCOPYRROLATE AND A BETA2 ADRENOCEPTOR AGONIST
EP05749635A EP1755590B1 (en) 2004-05-18 2005-05-17 Combination of glycopyrrolate and a beta2 adrenoceptor agonist
DK10164976.2T DK2228064T3 (en) 2004-05-18 2005-05-17 Pharmaceutical composition containing glycopyrrolate and a beta2-adrenoceptor agonist
ZA200608123A ZA200608123B (en) 2004-05-18 2006-09-29 Combinations of glycopyrrolate and beta2 adrenoceptor agonists
EC2006006950A ECSP066950A (en) 2004-05-18 2006-10-24 ADRENOCEPTOR-BETA2 GLICOPIRROLATE AND AGONIST COMBINATIONS
IL179013A IL179013A (en) 2004-05-18 2006-11-02 Medicaments comprising glycopyrrolate and (r)-5[ 2 -(5,6-diethyl-indan 2-ylamino)-1- hydroxy-ethyl]- 8-hydroxy-1h-quinoline-2-one for the treatment of chronic obstructive pulmonary disease
TNP2006000377A TNSN06377A1 (en) 2004-05-18 2006-11-15 Combinations of glycopyrrolate and beta2 adrenoceptor agonists
MA29475A MA28598B1 (en) 2004-05-18 2006-11-21 COMBINATIONS OF GLYCOPYRROLATE AND BETA2-ADRENERGIC RECEPTOR AGONISTS
NO20065787A NO334760B1 (en) 2004-05-18 2006-12-14 Combination of glycopyrrolate and a β-2-adrenoceptor agonist
HK07107762.4A HK1105579A1 (en) 2004-05-18 2007-07-18 Combinations of glycopyrrolate and beta2 adrenoceptor agonists
CY20111101145T CY1112086T1 (en) 2004-05-18 2011-11-24 Glycopyrrolate Salt Combination And An Adrenergic Receptor Beta2 Agent
JP2012156212A JP2012236833A (en) 2004-05-18 2012-07-12 Combination of glycopyrrolate and beta2 adrenergic receptor agonist
US13/862,529 US20130237564A1 (en) 2004-05-18 2013-04-15 Combinations of Glycopyrrolate and Beta2 Adrenoceptor Agonists
LTPA2014015C LTC1755590I2 (en) 2004-05-18 2014-03-13 A combination of glycopyrrolate and beta2 adrenoceptor agonist
HUS1400013C HUS1400013I1 (en) 2004-05-18 2014-03-13 Combination of glycopyrrolate and a beta2 adrenoceptor agonist
CY2014014C CY2014014I1 (en) 2004-05-18 2014-03-18 COMBINATION OF GLYCOPYRROLE SALT AND A BETA2 ADRENORECIPTOR AGENT
NO2014020C NO2014020I1 (en) 2004-05-18 2014-08-07 Glycopyrronium or a salt thereof and Indacaterol or a salt thereof in combination
US14/973,778 US20160101097A1 (en) 2004-05-18 2015-12-18 Combinations of Glycopyrrolate and Beta2 Adrenoceptor Agonists
US15/818,991 US20180071276A1 (en) 2004-05-18 2017-11-21 Combinations of Glycopyrrolate and Beta2 Adrenoceptor Agonists
US16/429,382 US20190282561A1 (en) 2004-05-18 2019-06-03 Combinations of Glycopyrrolate and Beta2 Adrenoceptor Agonists
CY20201100208T CY1122863T1 (en) 2004-05-18 2020-03-09 PHARMACEUTICAL COMPOSITION CONTAINING GLYCOPYRROLE AND A BETA2 ADRENOCEPTOR AGENT
FR20C1018C FR20C1018I2 (en) 2004-05-18 2020-05-27 Pharmaceutical composition comprising glycopyrrolate and a beta2 adrenergic receptor agonist
LU00155C LUC00155I2 (en) 2004-05-18 2020-05-27
HUS2000014C HUS2000014I1 (en) 2004-05-18 2020-06-05 Pharmaceutical composition containing glycopyrrolate and a beta2 adrenoceptor agonist
CY2020013C CY2020013I1 (en) 2004-05-18 2020-06-10 PHARMACEUTICAL COMPOSITION CONTAINING GLYCOPYRROLE AND A BETA2 ADRENOCEPTOR AGENT
LTPA2020509C LTC2228064I2 (en) 2004-05-18 2020-06-16 PHARMACEUTICAL COMPOSITION CONTAINING GLYCOPIROLATE AND BETA-2 ADRENOCEPTORAL ANTAGONIST
US17/237,350 US20210236478A1 (en) 2004-05-18 2021-04-22 Combinations of Glycopyrrolate and Beta2 Adrenoceptor Agonists

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0411056.5A GB0411056D0 (en) 2004-05-18 2004-05-18 Organic compounds

Publications (1)

Publication Number Publication Date
GB0411056D0 true GB0411056D0 (en) 2004-06-23

Family

ID=32607514

Family Applications (1)

Application Number Title Priority Date Filing Date
GBGB0411056.5A Ceased GB0411056D0 (en) 2004-05-18 2004-05-18 Organic compounds

Country Status (33)

Country Link
US (6) US20080267886A1 (en)
EP (3) EP2228064B1 (en)
JP (2) JP5567252B2 (en)
KR (2) KR20130018429A (en)
CN (1) CN1953745A (en)
AT (1) ATE521348T1 (en)
AU (1) AU2005244439C1 (en)
BR (1) BRPI0511327B8 (en)
CA (1) CA2563302C (en)
CY (4) CY1112086T1 (en)
DK (2) DK2228064T3 (en)
EC (1) ECSP066950A (en)
ES (2) ES2775979T3 (en)
FR (1) FR20C1018I2 (en)
GB (1) GB0411056D0 (en)
HK (1) HK1105579A1 (en)
HU (3) HUE048936T2 (en)
IL (1) IL179013A (en)
LT (3) LT2228064T (en)
LU (1) LUC00155I2 (en)
MA (1) MA28598B1 (en)
MX (1) MXPA06013382A (en)
NO (2) NO334760B1 (en)
NZ (1) NZ550369A (en)
PL (2) PL2228064T3 (en)
PT (2) PT2228064T (en)
RU (1) RU2388465C2 (en)
SE (1) SE1755590T5 (en)
SG (1) SG153836A1 (en)
SI (2) SI1755590T1 (en)
TN (1) TNSN06377A1 (en)
WO (1) WO2005110402A1 (en)
ZA (1) ZA200608123B (en)

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GB0523656D0 (en) * 2005-11-21 2005-12-28 Novartis Ag Organic compounds
GB0523655D0 (en) * 2005-11-21 2005-12-28 Novartis Ag Organic compounds
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US8198450B2 (en) * 2006-06-30 2012-06-12 Novartis Ag Quinolinone derivatives and their pharmaceutical compositions
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