EA201691857A1 - Соединения, применимые в качестве иммуномодуляторов - Google Patents
Соединения, применимые в качестве иммуномодуляторовInfo
- Publication number
- EA201691857A1 EA201691857A1 EA201691857A EA201691857A EA201691857A1 EA 201691857 A1 EA201691857 A1 EA 201691857A1 EA 201691857 A EA201691857 A EA 201691857A EA 201691857 A EA201691857 A EA 201691857A EA 201691857 A1 EA201691857 A1 EA 201691857A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- immunomodulators
- compounds
- applicable
- compounds applicable
- present
- Prior art date
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D319/00—Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D319/10—1,4-Dioxanes; Hydrogenated 1,4-dioxanes
- C07D319/14—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems
- C07D319/16—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D319/18—Ethylenedioxybenzenes, not substituted on the hetero ring
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- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
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- A61K31/275—Nitriles; Isonitriles
- A61K31/277—Nitriles; Isonitriles having a ring, e.g. verapamil
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- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/357—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having two or more oxygen atoms in the same ring, e.g. crown ethers, guanadrel
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- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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- A61K31/4015—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil having oxo groups directly attached to the heterocyclic ring, e.g. piracetam, ethosuximide
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- A61K31/4164—1,3-Diazoles
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Abstract
Изобретение в целом относится к соединениям, применимым в качестве иммуномодуляторов. В настоящем изобретении представлены соединения, композиции, содержащие такие соединения, и способы их применения. Раскрытие дополнительно относится к фармацевтическим композициям, содержащим по меньшей мере одно соединение по настоящему изобретению, которые применимы для лечения различных заболеваний, включая злокачественную опухоль и инфекционные заболевания.
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EA030811B1 (ru) | 2018-09-28 |
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