EA201300987A1 - Фармацевтические композиции, включающие метформин и ингибитор dpp-4 или ингибитор sglt-2 - Google Patents

Фармацевтические композиции, включающие метформин и ингибитор dpp-4 или ингибитор sglt-2

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Publication number
EA201300987A1
EA201300987A1 EA201300987A EA201300987A EA201300987A1 EA 201300987 A1 EA201300987 A1 EA 201300987A1 EA 201300987 A EA201300987 A EA 201300987A EA 201300987 A EA201300987 A EA 201300987A EA 201300987 A1 EA201300987 A1 EA 201300987A1
Authority
EA
Eurasian Patent Office
Prior art keywords
inhibitor
sglt
dpp
pharmaceutical compositions
methormene
Prior art date
Application number
EA201300987A
Other languages
English (en)
Inventor
Масанори Ито
Кенджи Эгуса
Роман Мессершмид
Петер Шнайдер
Original Assignee
Бёрингер Ингельхайм Интернациональ Гмбх
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=45808965&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA201300987(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Бёрингер Ингельхайм Интернациональ Гмбх filed Critical Бёрингер Ингельхайм Интернациональ Гмбх
Publication of EA201300987A1 publication Critical patent/EA201300987A1/ru

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52—Purines, e.g. adenine
    • A61K31/522—Purines, e.g. adenine having oxo groups directly attached to the heterocyclic ring, e.g. hypoxanthine, guanine, acyclovir
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    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
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  • Molecular Biology (AREA)
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  • Urology & Nephrology (AREA)
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  • Child & Adolescent Psychology (AREA)
  • Dermatology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Hospice & Palliative Care (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

В настоящем изобретении описаны фармацевтические композиции, включающие комбинации лекарственных средств с фиксированными дозами, ингибитора DPP-4 и/или ингибитора SGLT-2 и метформина с замедленным высвобождением (XR), способы их получения, а также их применение при лечении некоторых заболеваний.
EA201300987A 2011-03-07 2012-03-07 Фармацевтические композиции, включающие метформин и ингибитор dpp-4 или ингибитор sglt-2 EA201300987A1 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP11157240 2011-03-07
EP11158358 2011-03-15
PCT/EP2012/053910 WO2012120040A1 (en) 2011-03-07 2012-03-07 Pharmaceutical compositions comprising metformin and a dpp-4 inhibitor or a sglt-2 inhibitor

Publications (1)

Publication Number Publication Date
EA201300987A1 true EA201300987A1 (ru) 2014-03-31

Family

ID=45808965

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201300987A EA201300987A1 (ru) 2011-03-07 2012-03-07 Фармацевтические композиции, включающие метформин и ингибитор dpp-4 или ингибитор sglt-2

Country Status (15)

Country Link
US (5) US20130064887A1 (ru)
EP (1) EP2683366A1 (ru)
JP (2) JP2014507456A (ru)
KR (1) KR20140052970A (ru)
CN (1) CN103391771A (ru)
AR (1) AR085689A1 (ru)
BR (1) BR112013022789A2 (ru)
CA (1) CA2826640A1 (ru)
CL (1) CL2013002505A1 (ru)
EA (1) EA201300987A1 (ru)
IL (1) IL227528A0 (ru)
MX (1) MX2013010187A (ru)
SG (1) SG193338A1 (ru)
UY (1) UY33937A (ru)
WO (1) WO2012120040A1 (ru)

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