CS208164B2 - Method of making the d-2-halogene-6-methyl-8-kyan/carboxamido/methylergolines - Google Patents

Method of making the d-2-halogene-6-methyl-8-kyan/carboxamido/methylergolines Download PDF

Info

Publication number: CS208164B2
Authority: CS; Czechoslovakia
Prior art keywords: methyl; ergoline; formula; compounds; compound
Prior art date: 1972-07-21

Application number

CS735239A

Other languages

Czech (cs)

English (en)

Inventor

James A Clemens

Edmund C Kornfeld

Nicholas J Bach

Original Assignee

Lilly Co Eli

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1972-07-21

Filing date

1973-07-20

Publication date

1981-08-31

1973-07-20 Application filed by Lilly Co Eli filed Critical Lilly Co Eli

1977-10-13 Priority to CS776672A priority Critical patent/CS208165B2/cs

1981-08-31 Publication of CS208164B2 publication Critical patent/CS208164B2/cs

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D457/00—Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid
- C07D457/02—Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid with hydrocarbon or substituted hydrocarbon radicals, attached in position 8
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

CS735239A 1972-07-21 1973-07-20 Method of making the d-2-halogene-6-methyl-8-kyan/carboxamido/methylergolines CS208164B2 (en)

Priority Applications (1)

Application Number	Priority Date	Filing Date	Title
CS776672A CS208165B2 (cs)	1972-07-21	1977-10-13	Způsob výroby D-6-methyl-8-mesyIoxymethylergoIinu

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US27390272A	1972-07-21	1972-07-21

Publications (1)

Publication Number	Publication Date
CS208164B2 true CS208164B2 (en)	1981-08-31

Family

ID=23045910

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
CS735239A CS208164B2 (en)	1972-07-21	1973-07-20	Method of making the d-2-halogene-6-methyl-8-kyan/carboxamido/methylergolines

Country Status (24)

Country	Link
JP (2)	JPS576431B2 (ru)
AR (3)	AR206772A1 (ru)
AT (1)	AT331425B (ru)
BE (1)	BE802531A (ru)
BG (3)	BG22400A3 (ru)
CA (1)	CA1006159A (ru)
CH (5)	CH580625A5 (ru)
CS (1)	CS208164B2 (ru)
DD (1)	DD107690A5 (ru)
DE (2)	DE2335750C3 (ru)
DK (1)	DK140986B (ru)
ES (5)	ES417078A1 (ru)
FR (1)	FR2193606B1 (ru)
GB (1)	GB1423065A (ru)
HU (1)	HU167274B (ru)
IE (1)	IE37936B1 (ru)
IL (3)	IL48288A (ru)
NL (1)	NL7309969A (ru)
PH (1)	PH11229A (ru)
RO (2)	RO63792A (ru)
SE (3)	SE393111B (ru)
SU (3)	SU645581A3 (ru)
YU (1)	YU36953B (ru)
ZA (1)	ZA734627B (ru)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1517971A (en) *	1974-07-19	1978-07-19	Sandoz Ltd	8alpha-substituted ergoline i derivatives
US3968111A (en) *	1974-12-06	1976-07-06	Eli Lilly And Company	8,8-Disubstituted-6-methylergolines and related compounds
US4166182A (en) *	1978-02-08	1979-08-28	Eli Lilly And Company	6-n-propyl-8-methoxymethyl or methylmercaptomethylergolines and related compounds
AU526764B2 (en) *	1978-09-08	1983-01-27	Farmitalia Carlo Erba S.P.A.	Ergoline derivatives
ATE107647T1 (de) *	1984-04-09	1994-07-15	Schering Ag	2-substituierte ergolin-derivate, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel.
HU196598B (en) *	1986-04-25	1988-12-28	Richter Gedeon Vegyeszet	Process for producing 1- and/or 8-substituted 2-halogenated ergoline derivatives and pharmaceutics comprising such compounds
DE3620293A1 (de) *	1986-06-16	1987-12-17	Schering Ag	1-und/oder 2-substituierte ergolinderivate
JPH0596382U (ja) *	1992-05-28	1993-12-27	イビデン株式会社	ドアユニット

1973
- 1973-01-01 AR AR249167A patent/AR206772A1/es active
- 1973-07-10 GB GB3289073A patent/GB1423065A/en not_active Expired
- 1973-07-10 ZA ZA734627A patent/ZA734627B/xx unknown
- 1973-07-12 SE SE7309781A patent/SE393111B/xx unknown
- 1973-07-12 IL IL48288A patent/IL48288A/en unknown
- 1973-07-12 IL IL42730A patent/IL42730A/en unknown
- 1973-07-13 DE DE2335750A patent/DE2335750C3/de not_active Expired
- 1973-07-13 DE DE2365974A patent/DE2365974A1/de not_active Withdrawn
- 1973-07-17 NL NL7309969A patent/NL7309969A/xx not_active Application Discontinuation
- 1973-07-17 YU YU1945/73A patent/YU36953B/xx unknown
- 1973-07-18 PH PH14835A patent/PH11229A/en unknown
- 1973-07-19 HU HUEI485A patent/HU167274B/hu unknown
- 1973-07-19 BE BE1005246A patent/BE802531A/xx not_active IP Right Cessation
- 1973-07-19 DK DK399873AA patent/DK140986B/da unknown
- 1973-07-20 BG BG28443A patent/BG22400A3/xx unknown
- 1973-07-20 CH CH391076A patent/CH580625A5/xx not_active IP Right Cessation
- 1973-07-20 CA CA177,021A patent/CA1006159A/en not_active Expired
- 1973-07-20 BG BG24148A patent/BG21410A3/xx unknown
- 1973-07-20 DD DD172402A patent/DD107690A5/xx unknown
- 1973-07-20 JP JP8074973A patent/JPS576431B2/ja not_active Expired
- 1973-07-20 BG BG26855A patent/BG21411A3/xx not_active Expired
- 1973-07-20 CH CH391276A patent/CH580626A5/xx not_active IP Right Cessation
- 1973-07-20 RO RO7300083213A patent/RO63792A/ro unknown
- 1973-07-20 IE IE1238/73A patent/IE37936B1/xx unknown
- 1973-07-20 ES ES417078A patent/ES417078A1/es not_active Expired
- 1973-07-20 SU SU731948966A patent/SU645581A3/ru active
- 1973-07-20 AT AT643473A patent/AT331425B/de not_active IP Right Cessation
- 1973-07-20 CH CH391176A patent/CH578563A5/xx not_active IP Right Cessation
- 1973-07-20 CS CS735239A patent/CS208164B2/cs unknown
- 1973-07-20 CH CH391376A patent/CH578564A5/xx not_active IP Right Cessation
- 1973-07-20 CH CH1067873A patent/CH581135A5/xx not_active IP Right Cessation
- 1973-07-20 FR FR7326708A patent/FR2193606B1/fr not_active Expired
- 1973-07-20 RO RO7375548A patent/RO71305A/ro unknown
1974
- 1974-01-01 AR AR252738A patent/AR206887A1/es active
- 1974-12-04 SU SU7402080295A patent/SU584780A3/ru active
1975
- 1975-01-14 SU SU7502098198A patent/SU575029A3/ru active
- 1975-01-30 AR AR257473A patent/AR210072A1/es active
- 1975-10-13 IL IL48288A patent/IL48288A0/xx unknown
- 1975-11-21 ES ES442886A patent/ES442886A1/es not_active Expired
- 1975-11-21 ES ES442887A patent/ES442887A1/es not_active Expired
- 1975-11-21 ES ES442885A patent/ES442885A1/es not_active Expired
1976
- 1976-04-07 ES ES446789A patent/ES446789A1/es not_active Expired
- 1976-10-15 SE SE7611466A patent/SE410459B/xx unknown
- 1976-10-15 SE SE7611467A patent/SE410603B/xx unknown
1981
- 1981-08-07 JP JP56123937A patent/JPS5813541B2/ja not_active Expired

Also Published As

Publication number	Publication date
HU167274B (ru)	1975-09-27
CH580625A5 (ru)	1976-10-15
IL42730A0 (en)	1973-10-25
DK140986C (ru)	1980-07-21
YU194573A (en)	1982-06-18
ZA734627B (en)	1974-06-26
ES442886A1 (es)	1977-04-16
BG21410A3 (ru)	1976-05-20
JPS576431B2 (ru)	1982-02-04
SE393111B (sv)	1977-05-02
CH580626A5 (ru)	1976-10-15
AT331425B (de)	1976-08-25
SE410459B (sv)	1979-10-15
DE2335750A1 (de)	1974-02-14
CH578563A5 (ru)	1976-08-13
IL42730A (en)	1976-06-30
ATA643473A (de)	1975-11-15
GB1423065A (en)	1976-01-28
DE2335750C3 (de)	1978-10-19
PH11229A (en)	1977-10-28
ES446789A1 (es)	1977-06-01
IL48288A (en)	1976-06-30
AU5792673A (en)	1975-01-16
DK140986B (da)	1979-12-17
FR2193606A1 (ru)	1974-02-22
CH581135A5 (ru)	1976-10-29
BG22400A3 (ru)	1977-02-20
SU575029A3 (ru)	1977-09-30
ES442885A1 (es)	1977-04-16
CA1006159A (en)	1977-03-01
DE2335750B2 (de)	1978-02-23
SU584780A3 (ru)	1977-12-15
CH578564A5 (ru)	1976-08-13
SE7611467L (sv)	1976-10-15
DE2365974A1 (de)	1977-03-24
ES417078A1 (es)	1976-05-01
SE7611466L (sv)	1976-10-15
JPS5813541B2 (ja)	1983-03-14
BG21411A3 (ru)	1976-05-20
FR2193606B1 (ru)	1977-07-15
ES442887A1 (es)	1977-05-16
IL48288A0 (en)	1975-12-31
IE37936B1 (en)	1977-11-23
AR210072A1 (es)	1977-06-30
RO63792A (fr)	1978-12-15
YU36953B (en)	1984-08-31
JPS4985099A (ru)	1974-08-15
AR206887A1 (es)	1976-08-31
RO71305A (ro)	1982-03-24
NL7309969A (ru)	1974-01-23
DD107690A5 (ru)	1974-08-12
JPS5781487A (en)	1982-05-21
SE410603B (sv)	1979-10-22
BE802531A (fr)	1974-01-21
SU645581A3 (ru)	1979-01-30
IE37936L (en)	1974-01-21
AR206772A1 (es)	1976-08-23

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