AR004010A1 - Compuestos heterociclicos - Google Patents

Compuestos heterociclicos

Info

Publication number
AR004010A1
AR004010A1 ARP960104659A AR10465996A AR004010A1 AR 004010 A1 AR004010 A1 AR 004010A1 AR P960104659 A ARP960104659 A AR P960104659A AR 10465996 A AR10465996 A AR 10465996A AR 004010 A1 AR004010 A1 AR 004010A1
Authority
AR
Argentina
Prior art keywords
compounds
cyclic compounds
hetero cyclic
heteroaromatic compounds
asubstituted
Prior art date
Application number
ARP960104659A
Other languages
English (en)
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9520845.0A external-priority patent/GB9520845D0/en
Priority claimed from GBGB9614757.4A external-priority patent/GB9614757D0/en
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of AR004010A1 publication Critical patent/AR004010A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems

Abstract

La presente invención describe compuestos heteroaromáticos sustituidos, y en particular compuestos heteroaromáticos bicíclicos de la formula Asustituidos en los cuales un anillo es una piridina o pirimidina,y que son inhibidores de las tirosina cinasas proteicas. Se describen los compuestoscomo son, métodos para su preparación, composiciones farmacéuticas que incluyen esos compuestos y su uso en medicina, por ejemplo, en el tratamiento depsoriasis, fibrosis, aterosclerosis, restenosis,enfermedad autoinmune,alergia, asma, rechazo al trasplante, inflamación, trombosis, enfermedades del sistemanervioso y cáncer.
ARP960104659A 1995-10-11 1996-09-10 Compuestos heterociclicos AR004010A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9520845.0A GB9520845D0 (en) 1995-10-11 1995-10-11 Therapeutically active compounds
GBGB9614757.4A GB9614757D0 (en) 1996-07-13 1996-07-13 Therapeutically active compounds

Publications (1)

Publication Number Publication Date
AR004010A1 true AR004010A1 (es) 1998-09-30

Family

ID=26307933

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP960104659A AR004010A1 (es) 1995-10-11 1996-09-10 Compuestos heterociclicos

Country Status (8)

Country Link
US (1) US6169091B1 (es)
EP (1) EP0861253A1 (es)
JP (1) JPH11513398A (es)
AR (1) AR004010A1 (es)
AU (1) AU7289696A (es)
HR (1) HRP960465A2 (es)
ID (1) ID16345A (es)
WO (1) WO1997013771A1 (es)

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