NO159531C - Analogifremgangsmaate for fremstilling av farmasoeytisk aktive karbostyrilderivater. - Google Patents

Analogifremgangsmaate for fremstilling av farmasoeytisk aktive karbostyrilderivater.

Info

Publication number
NO159531C
NO159531C NO810765A NO810765A NO159531C NO 159531 C NO159531 C NO 159531C NO 810765 A NO810765 A NO 810765A NO 810765 A NO810765 A NO 810765A NO 159531 C NO159531 C NO 159531C
Authority
NO
Norway
Prior art keywords
pharmasoyytic
carbostyric
derivatives
active
preparation
Prior art date
Application number
NO810765A
Other languages
English (en)
Norwegian (no)
Other versions
NO810765L (no
NO159531B (no
Inventor
Kazuo Banno
Takafumi Fujioka
Masaaki Osaki
Kazuyuki Nakagawa
Original Assignee
Otsuka Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP2880580A external-priority patent/JPS56125370A/ja
Priority claimed from JP11502280A external-priority patent/JPS5738772A/ja
Application filed by Otsuka Pharma Co Ltd filed Critical Otsuka Pharma Co Ltd
Publication of NO810765L publication Critical patent/NO810765L/no
Publication of NO159531B publication Critical patent/NO159531B/no
Publication of NO159531C publication Critical patent/NO159531C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20Oxygen atoms
    • C07D215/22Oxygen atoms attached in position 2 or 4
    • C07D215/227Oxygen atoms attached in position 2 or 4 only one oxygen atom which is attached in position 2

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
NO810765A 1980-03-06 1981-03-05 Analogifremgangsmaate for fremstilling av farmasoeytisk aktive karbostyrilderivater. NO159531C (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2880580A JPS56125370A (en) 1980-03-06 1980-03-06 Carbostyril derivative
JP11502280A JPS5738772A (en) 1980-08-20 1980-08-20 Carbostyril derivative

Publications (3)

Publication Number Publication Date
NO810765L NO810765L (no) 1981-09-07
NO159531B NO159531B (no) 1988-10-03
NO159531C true NO159531C (no) 1989-01-11

Family

ID=26366952

Family Applications (1)

Application Number Title Priority Date Filing Date
NO810765A NO159531C (no) 1980-03-06 1981-03-05 Analogifremgangsmaate for fremstilling av farmasoeytisk aktive karbostyrilderivater.

Country Status (21)

Country Link
US (4) US4567187A (es)
AT (1) AT381307B (es)
AU (1) AU523005B2 (es)
BE (1) BE887800A (es)
CA (1) CA1155119A (es)
CH (1) CH647775A5 (es)
DE (2) DE3152880C2 (es)
DK (1) DK155282C (es)
ES (4) ES500137A0 (es)
FI (1) FI76323C (es)
FR (1) FR2477542A1 (es)
GB (1) GB2071094B (es)
IT (1) IT1144315B (es)
MX (1) MX6980E (es)
NL (1) NL184364C (es)
NO (1) NO159531C (es)
PH (1) PH17194A (es)
PT (1) PT72622B (es)
RU (1) RU1779249C (es)
SE (1) SE447255B (es)
SU (1) SU1367857A3 (es)

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PH17194A (en) * 1980-03-06 1984-06-19 Otsuka Pharma Co Ltd Novel carbostyril derivatives,and pharmaceutical composition containing the same
FI77852C (fi) * 1981-02-17 1989-05-10 Otsuka Pharma Co Ltd Foerfarande foer framstaellning av nya, saosom hjaertmediciner anvaendbara substituerade amid- och (maettad heterocykel)karbonylkarbostyrilderivat.
AU532361B2 (en) * 1981-09-01 1983-09-29 Otsuka Pharmaceutical Co., Ltd. Carbostyril derivatives
US4578381A (en) * 1982-07-05 1986-03-25 Otsuka Pharmaceutical Co., Ltd. Carbostyril derivatives
CH655110A5 (de) * 1982-09-03 1986-03-27 Otsuka Pharma Co Ltd Carbostyrilderivate, verfahren zu deren herstellung und arzneimittel, welche diese enthalten.
DE3434271A1 (de) * 1984-09-19 1986-03-20 Beiersdorf Ag, 2000 Hamburg Substituierte 3,4-dihydro-chinolin-2(1h)-one verfahren zu ihrer herstellung und ihre verwendung sowie diese verbindungen enthaltende zubereitungen
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US6255322B1 (en) 1992-06-19 2001-07-03 Pfizer Inc. 2-(4-hydroxypiperidino)-1-alkanol derivatives as antiischemic agents
DE69430861T2 (de) * 1993-04-07 2003-01-23 Otsuka Pharma Co Ltd N-acylierte 4-aminopiperidin derivate als aktive bestandteile von peripher gefässerweiternden wikstoffen
DK0709384T3 (da) * 1994-10-31 1999-08-23 Merck Patent Gmbh Benzylpiperidinderivater med høj affinitet til aminosyrereceptorers bindingssteder
ZA9610738B (en) 1995-12-22 1997-06-24 Warner Lambert Co Subtype selective nmda receptor ligands and the use thereof
ZA9610745B (en) * 1995-12-22 1997-06-24 Warner Lambert Co 4-Subsituted piperidine analogs and their use as subtype selective nmda receptor antagonists
ZA9610736B (en) * 1995-12-22 1997-06-27 Warner Lambert Co 2-Substituted piperidine analogs and their use as subtypeselective nmda receptor antagonists
ZA9610741B (en) 1995-12-22 1997-06-24 Warner Lambert Co 4-Substituted piperidine analogs and their use as subtype selective nmda receptor antagonists
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FR2823749B1 (fr) * 2001-04-20 2004-02-20 Sanofi Synthelabo Phenyl- et pyridyl-piperidines, procede pour leur preparation et compositions pharmaceutiques les contenant
MY129350A (en) * 2001-04-25 2007-03-30 Bristol Myers Squibb Co Aripiprazole oral solution
DE10210779A1 (de) * 2002-03-12 2003-10-09 Merck Patent Gmbh Cyclische Amide
AU2003212335B8 (en) * 2002-03-13 2009-04-23 Janssen Pharmaceutica N.V. Aminocarbonyl-derivatives as novel inhibitors of histone deacetylase
NZ534831A (en) 2002-03-13 2007-01-26 Janssen Pharmaceutica Nv Carbonylamino-derivatives having histone deacetylase (HDAC) inhibiting enzymatic activity
DK1485354T3 (da) 2002-03-13 2008-09-01 Janssen Pharmaceutica Nv Sulfonylamino-derivater som nye inhibitorer af histandeacetylase
BR0307606A (pt) * 2002-03-13 2004-12-21 Janssen Pharmaceutica Nv Derivados de piperazinila, piperidinila e morfolinila como inibidores de histona desacetilase
MY142362A (en) * 2004-01-29 2010-11-30 Otsuka Pharma Co Ltd Pharmaceutical composition for promoting angiogenesis
ES2327253T3 (es) * 2004-07-28 2009-10-27 Janssen Pharmaceutica Nv Derivados de propenil piperazina sustituidos como nuevos inhibidores de histona deacetilasa.
WO2006010750A1 (en) 2004-07-28 2006-02-02 Janssen Pharmaceutica N.V. Substituted indolyl alkyl amino derivatives as novel inhibitors of histone deacetylase
RS51189B (sr) * 2004-07-28 2010-10-31 Janssen Pharmaceutica N.V. Supstituisani derivati propenil piperazina kao novi inhibitori histonske deacetilaze
TWI320783B (en) 2005-04-14 2010-02-21 Otsuka Pharma Co Ltd Heterocyclic compound
EP1885710B1 (en) 2005-05-18 2015-08-19 Janssen Pharmaceutica N.V. Substituted aminopropenyl piperidine or morpholine derivatives as novel inhibitors of histone deacetylase
SI1981874T1 (sl) * 2006-01-19 2009-10-31 Janssen Pharmaceutica Nv Aminofenilni derivati kot novi inhibitorji histon deacetilaze
AU2007206944B2 (en) * 2006-01-19 2012-08-23 Janssen Pharmaceutica N.V. Pyridine and pyrimidine derivatives as inhibitors of histone deacetylase
AU2007206942B2 (en) 2006-01-19 2012-08-23 Janssen Pharmaceutica N.V. Pyridine and pyrimidine derivatives as inhibitors of histone deacetylase
JP5137849B2 (ja) * 2006-01-19 2013-02-06 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ ヒストンデアセチラーゼのインヒビターとしての置換インドリル−アルキル−アミノ−誘導体
US7935706B2 (en) * 2006-02-23 2011-05-03 Shionogi & Co., Ltd. Nitrogen-containing heterocycle derivatives substituted with cyclic group
WO2009034029A2 (de) * 2007-09-07 2009-03-19 Boehringer Ingelheim International Gmbh 1-substituierte 4 -heterocyclylpiperidine als cgrp antagonisten
KR101705727B1 (ko) 2009-02-26 2017-02-10 레비바 파마슈티칼스, 아이엔씨. 아릴피페라진 유도체의 조성물, 합성, 및 사용 방법
US9951088B2 (en) * 2012-05-09 2018-04-24 Sunovion Pharmaceuticals Inc. D2 receptor modulators and methods of use thereof in the treatment of diseases and disorders
CN106608875A (zh) 2015-10-26 2017-05-03 江苏恩华药业股份有限公司 一种稠和杂环类衍生物合成及其应用
CN108031471A (zh) * 2017-10-27 2018-05-15 苏州盖德精细材料有限公司 一种静电纺丝制备的负载型纳米纤维催化剂及其在3,5-二羟基甲苯制备中的应用
CN114409680B (zh) * 2018-01-19 2023-11-21 上海怡立舍生物技术有限公司 Ppar激动剂及其应用
CN116554127A (zh) * 2022-01-28 2023-08-08 成都麻沸散医药科技有限公司 哌嗪取代苯酚类衍生物及其用途

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Also Published As

Publication number Publication date
ES8306141A1 (es) 1983-05-01
ES8301962A1 (es) 1982-11-01
FI76323B (fi) 1988-06-30
SE447255B (sv) 1986-11-03
DE3107601A1 (de) 1982-02-04
US4567187A (en) 1986-01-28
ES500137A0 (es) 1982-11-01
IT1144315B (it) 1986-10-29
CH647775A5 (de) 1985-02-15
ES509659A0 (es) 1983-05-01
DE3107601C2 (es) 1989-07-20
US4455422A (en) 1984-06-19
FR2477542A1 (fr) 1981-09-11
CA1155119A (en) 1983-10-11
FI76323C (fi) 1988-10-10
FI810669L (fi) 1981-09-07
GB2071094B (en) 1984-09-26
AT381307B (de) 1986-09-25
PH17194A (en) 1984-06-19
DE3152880C2 (es) 1990-03-22
RU1779249C (ru) 1992-11-30
GB2071094A (en) 1981-09-16
NL184364B (nl) 1989-02-01
SE8101409L (sv) 1981-09-07
ES518667A0 (es) 1984-06-16
DK155282B (da) 1989-03-20
SU1367857A3 (ru) 1988-01-15
US4619932A (en) 1986-10-28
NO810765L (no) 1981-09-07
PT72622A (en) 1981-04-01
AU6797381A (en) 1981-09-10
DK99781A (da) 1981-09-07
ES8405782A1 (es) 1984-06-16
IT8167311A0 (it) 1981-03-05
NO159531B (no) 1988-10-03
NL8101099A (nl) 1981-10-01
NL184364C (nl) 1989-07-03
MX6980E (es) 1987-01-19
FR2477542B1 (es) 1983-09-09
ATA98481A (de) 1986-02-15
ES8305356A1 (es) 1983-04-01
US4460593A (en) 1984-07-17
PT72622B (en) 1982-06-15
AU523005B2 (en) 1982-07-08
DK155282C (da) 1989-08-07
BE887800A (fr) 1981-09-07
ES509658A0 (es) 1983-04-01

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