ID24372A - SENYAWA-SENYAWA 4-AMINO-TIAZOL-2-IL SEBAGAI PENGHAMBAT-PENGHAMBAT CDKs - Google Patents

SENYAWA-SENYAWA 4-AMINO-TIAZOL-2-IL SEBAGAI PENGHAMBAT-PENGHAMBAT CDKs

Info

Publication number
ID24372A
ID24372A IDW20000740A ID20000740A ID24372A ID 24372 A ID24372 A ID 24372A ID W20000740 A IDW20000740 A ID W20000740A ID 20000740 A ID20000740 A ID 20000740A ID 24372 A ID24372 A ID 24372A
Authority
ID
Indonesia
Prior art keywords
compounds
cdkers
tiazol
amino
Prior art date
Application number
IDW20000740A
Other languages
English (en)
Indonesian (id)
Inventor
Wesley K M Chong
Shao Song Chu
Rohit R Duvadie
Lin Li
Wei Xiao
Yi Yang
Original Assignee
Agouron Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Agouron Pharma filed Critical Agouron Pharma
Publication of ID24372A publication Critical patent/ID24372A/id

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38Nitrogen atoms
    • C07D277/42Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
IDW20000740A 1997-10-27 1998-10-27 SENYAWA-SENYAWA 4-AMINO-TIAZOL-2-IL SEBAGAI PENGHAMBAT-PENGHAMBAT CDKs ID24372A (id)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US6363497P 1997-10-27 1997-10-27
US6366697P 1997-10-28 1997-10-28

Publications (1)

Publication Number Publication Date
ID24372A true ID24372A (id) 2000-07-13

Family

ID=26743609

Family Applications (1)

Application Number Title Priority Date Filing Date
IDW20000740A ID24372A (id) 1997-10-27 1998-10-27 SENYAWA-SENYAWA 4-AMINO-TIAZOL-2-IL SEBAGAI PENGHAMBAT-PENGHAMBAT CDKs

Country Status (34)

Country Link
US (2) US6569878B1 (de)
EP (1) EP1056732B1 (de)
JP (1) JP2004500304A (de)
KR (1) KR20010082501A (de)
CN (1) CN1158269C (de)
AP (1) AP1445A (de)
AT (2) ATE315553T1 (de)
AU (1) AU738792B2 (de)
BG (1) BG64195B1 (de)
BR (1) BR9815200A (de)
CA (1) CA2306082A1 (de)
DE (2) DE69835241T2 (de)
EA (1) EA003527B1 (de)
EE (1) EE200000289A (de)
ES (2) ES2267873T3 (de)
GE (1) GEP20032896B (de)
HR (1) HRP20000222A2 (de)
HU (1) HUP0004512A3 (de)
ID (1) ID24372A (de)
IL (1) IL135574A0 (de)
IS (1) IS5462A (de)
LT (1) LT4855B (de)
LV (1) LV12592B (de)
NO (1) NO20001955L (de)
NZ (1) NZ503788A (de)
OA (1) OA11352A (de)
PL (1) PL342447A1 (de)
RO (1) RO119463B1 (de)
SI (1) SI20324A (de)
SK (1) SK5212000A3 (de)
TR (1) TR200001081T2 (de)
UA (1) UA66810C2 (de)
WO (1) WO1999021845A2 (de)
YU (1) YU22400A (de)

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US6414156B2 (en) 1998-10-21 2002-07-02 Bristol-Myers Squibb Company Process for preparing azacycloalkanoylaminothiazoles
RU2312860C2 (ru) 1999-04-15 2007-12-20 Бристол-Маерс Сквибб Компани Циклические ингибиторы протеинтирозинкиназ
US7125875B2 (en) 1999-04-15 2006-10-24 Bristol-Myers Squibb Company Cyclic protein tyrosine kinase inhibitors
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US7141581B2 (en) 1999-07-02 2006-11-28 Agouron Pharmaceuticals, Inc. Indazole compounds and pharmaceutical compositions for inhibiting protein kinases, and methods for their use
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US6515004B1 (en) 1999-12-15 2003-02-04 Bristol-Myers Squibb Company N-[5-[[[5-alkyl-2-oxazolyl]methyl]thio]-2-thiazolyl]-carboxamide inhibitors of cyclin dependent kinases
YU54202A (sh) 2000-01-18 2006-01-16 Agouron Pharmaceuticals Inc. Jedinjenja indazola, farmaceutske smeše i postupci za stimulisanje i inhibiranje ćelijske proliferacije
HN2001000008A (es) 2000-01-21 2003-12-11 Inc Agouron Pharmaceuticals Compuesto de amida y composiciones farmaceuticas para inhibir proteinquinasas, y su modo de empleo
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EP1274706A1 (de) 2000-04-18 2003-01-15 Agouron Pharmaceuticals, Inc. Pyrazole zur inhibierung von proteinkinasen
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DE69835241D1 (de) 2006-08-24
NO20001955L (no) 2000-06-16
US6569878B1 (en) 2003-05-27
EE200000289A (et) 2001-06-15
BG104478A (en) 2001-02-28
DE69833223D1 (de) 2006-04-06
HRP20000222A2 (en) 2001-02-28
HUP0004512A2 (hu) 2002-03-28
OA11352A (en) 2003-12-23
KR20010082501A (ko) 2001-08-30
AP1445A (en) 2005-07-10
AU1366499A (en) 1999-05-17
NZ503788A (en) 2002-11-26
WO1999021845A2 (en) 1999-05-06
CN1276789A (zh) 2000-12-13
NO20001955D0 (no) 2000-04-14
EA003527B1 (ru) 2003-06-26
LV12592A (en) 2000-12-20
LV12592B (en) 2001-07-20
RO119463B1 (ro) 2004-11-30
BR9815200A (pt) 2001-10-16
EP1056732B1 (de) 2006-01-11
DE69835241T2 (de) 2007-05-31
WO1999021845A3 (en) 1999-08-19
LT4855B (lt) 2001-11-26
GEP20032896B (en) 2003-02-25
CA2306082A1 (en) 1999-05-06
AP2000001795A0 (en) 2000-06-30
ES2267873T3 (es) 2007-03-16
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ATE315553T1 (de) 2006-02-15
HUP0004512A3 (en) 2003-01-28
CN1158269C (zh) 2004-07-21
IL135574A0 (en) 2001-05-20
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US20030220326A1 (en) 2003-11-27
DE69833223T2 (de) 2006-09-14
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AU738792B2 (en) 2001-09-27
SI20324A (sl) 2001-02-28
SK5212000A3 (en) 2001-04-09
TR200001081T2 (tr) 2000-10-23
ATE332896T1 (de) 2006-08-15
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UA66810C2 (uk) 2004-06-15
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YU22400A (sh) 2003-08-29

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