HN2002000156A - Derivados de benzamida tiazol y composiciones farmaceuticas para inhibir la proliferacion de celulas y metodos para su utilización. - Google Patents

Derivados de benzamida tiazol y composiciones farmaceuticas para inhibir la proliferacion de celulas y metodos para su utilización.

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Publication number
HN2002000156A
HN2002000156A HN2002000156A HN2002000156A HN2002000156A HN 2002000156 A HN2002000156 A HN 2002000156A HN 2002000156 A HN2002000156 A HN 2002000156A HN 2002000156 A HN2002000156 A HN 2002000156A HN 2002000156 A HN2002000156 A HN 2002000156A
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HN
Honduras
Prior art keywords
benzamide
proliferation
inhibit
cells
methods
Prior art date
Application number
HN2002000156A
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English (en)
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Inc Agouron Pharmaceuticals
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Publication date
Application filed by Inc Agouron Pharmaceuticals filed Critical Inc Agouron Pharmaceuticals
Publication of HN2002000156A publication Critical patent/HN2002000156A/es

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    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
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    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
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    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
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    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38—Nitrogen atoms
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    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/10—Spiro-condensed systems

Abstract

LA PRESENTE INVENCIÓN SE REFIERE A COMPUESTOS AMINOTIAZOL CON BENZAMIDA MONO - DI/SUSTITUIDOS ESTAN REPRESENTADOS POR LA FORMULA (I), Y SE DESCRIBEN SUS SALES FARMACEUTICAMENTE ACEPTABLES, PRO DROGAS FARMACEUTICAMENTE ACEPTABLES, METABOLITOS FARMACEUTICAMENTE ACTIVOS Y SALES FARMACEUTICAMENTE ACEPTABLES DE DICHOS METABOLITOS.
HN2002000156A 2001-07-06 2002-06-26 Derivados de benzamida tiazol y composiciones farmaceuticas para inhibir la proliferacion de celulas y metodos para su utilización. HN2002000156A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US30367901P 2001-07-06 2001-07-06
US30527401P 2001-07-13 2001-07-13

Publications (1)

Publication Number Publication Date
HN2002000156A true HN2002000156A (es) 2003-11-27

Family

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HN2002000156A HN2002000156A (es) 2001-07-06 2002-06-26 Derivados de benzamida tiazol y composiciones farmaceuticas para inhibir la proliferacion de celulas y metodos para su utilización.

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Country Link
US (1) US6720346B2 (es)
EP (1) EP1438046A4 (es)
JP (1) JP2005521631A (es)
AU (1) AU2002354801A1 (es)
BR (1) BR0210874A (es)
CA (1) CA2452609A1 (es)
HN (1) HN2002000156A (es)
MX (1) MXPA04000069A (es)
PA (1) PA8550101A1 (es)
PE (1) PE20030269A1 (es)
SV (1) SV2003001148A (es)
UY (1) UY27370A1 (es)
WO (1) WO2003004467A2 (es)

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CA2452609A1 (en) 2003-01-16
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WO2003004467A3 (en) 2004-05-06
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