ID28032A - TRISIKLIK PIPERIDIN-Δ3-SEBAGAI ANTAGONIS-α2 - Google Patents

TRISIKLIK PIPERIDIN-Δ3-SEBAGAI ANTAGONIS-α2

Info

Publication number
ID28032A
ID28032A IDW20010780A ID20010780A ID28032A ID 28032 A ID28032 A ID 28032A ID W20010780 A IDW20010780 A ID W20010780A ID 20010780 A ID20010780 A ID 20010780A ID 28032 A ID28032 A ID 28032A
Authority
ID
Indonesia
Prior art keywords
triciclic
antagonis
piperidin
Prior art date
Application number
IDW20010780A
Other languages
English (en)
Inventor
Ludo E J Kennis
Frans M A Van Den Keybus
Josephus C Mertens
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of ID28032A publication Critical patent/ID28032A/id

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
IDW20010780A 1998-10-06 1999-10-01 TRISIKLIK PIPERIDIN-Δ3-SEBAGAI ANTAGONIS-α2 ID28032A (id)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP98203370 1998-10-06

Publications (1)

Publication Number Publication Date
ID28032A true ID28032A (id) 2001-05-03

Family

ID=8234191

Family Applications (1)

Application Number Title Priority Date Filing Date
IDW20010780A ID28032A (id) 1998-10-06 1999-10-01 TRISIKLIK PIPERIDIN-Δ3-SEBAGAI ANTAGONIS-α2

Country Status (31)

Country Link
US (1) US6495555B1 (id)
EP (1) EP1119571B1 (id)
JP (1) JP4590101B2 (id)
KR (1) KR20010071843A (id)
CN (1) CN1131230C (id)
AR (1) AR024216A1 (id)
AT (1) ATE232869T1 (id)
AU (1) AU760502B2 (id)
BG (1) BG64872B1 (id)
BR (1) BR9913507A (id)
CA (1) CA2345622C (id)
CZ (1) CZ20011104A3 (id)
DE (1) DE69905478T2 (id)
DK (1) DK1119571T3 (id)
EE (1) EE04770B1 (id)
ES (1) ES2193751T3 (id)
HK (1) HK1038010A1 (id)
HU (1) HUP0104002A3 (id)
ID (1) ID28032A (id)
IL (1) IL142443A0 (id)
NO (1) NO20011270D0 (id)
NZ (1) NZ510115A (id)
PL (1) PL347894A1 (id)
PT (1) PT1119571E (id)
RU (1) RU2230744C2 (id)
SI (1) SI1119571T1 (id)
SK (1) SK285585B6 (id)
TR (1) TR200100952T2 (id)
TW (1) TWI248441B (id)
UA (1) UA69420C2 (id)
WO (1) WO2000020421A2 (id)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE69918148T2 (de) * 1998-10-06 2005-07-28 Janssen Pharmaceutica N.V. Trizyclische delta3-pyridine als arzneimittel
ATE521593T1 (de) * 2002-04-03 2011-09-15 Orion Corp Verwendung eines alfa2-adrenorezeptorantagonisten bei mit dem zns zusammenhängenden erkrankungen
WO2005100355A1 (ja) 2004-04-12 2005-10-27 Taisho Pharmaceutical Co., Ltd. 環状アミン化合物
WO2006006740A1 (ja) * 2004-07-14 2006-01-19 Japan Tobacco Inc. ３−アミノベンズアミド化合物及びバニロイド受容体１型(ｖｒ１)活性阻害剤
CA2571133C (en) * 2004-07-15 2011-04-19 Japan Tobacco Inc. Fused benzamide compound and vanilloid receptor 1 (vr1) activity inhibitor
US7906508B2 (en) 2005-12-28 2011-03-15 Japan Tobacco Inc. 3,4-dihydrobenzoxazine compounds and inhibitors of vanilloid receptor subtype 1 (VRI) activity
NZ596137A (en) 2009-05-14 2013-08-30 Janssen Pharmaceutica Nv Compounds with two fused bicyclic heteroaryl moieties as modulators of leukotriene a4 hydrolase
US9624199B2 (en) 2013-12-19 2017-04-18 Bayer Pharma Aktiengesellschaft Substituted bipiperidinyl derivatives
JOP20200052A1 (ar) 2013-12-19 2017-06-16 Bayer Pharma AG بيبريدينيل تتراهيدرو كوينولينات مستبدلة واستخدامها كمعضدات مستقبل أدريني ألفا- 2c
WO2015091417A1 (de) * 2013-12-19 2015-06-25 Bayer Pharma Aktiengesellschaft Substituierte piperidinyl-tetrahydrochinoline
CN114276359B (zh) * 2022-01-05 2023-05-05 浙江大学 一种1,2,3,4-四氢苯并[4,5]呋喃[2,3-c]吡啶衍生物的制备方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3522959A1 (de) 1985-06-27 1987-01-08 Merck Patent Gmbh Indolderivate
US4673680A (en) * 1985-09-18 1987-06-16 Pendleton Robert G α2 -adrenergic receptor antagonists as modifiers of gastrointestinal motility
EP0339959A3 (en) * 1988-04-27 1991-03-20 Glaxo Group Limited Lactam derivatives
US4971974A (en) 1988-06-16 1990-11-20 Neurex Corporation Benzothiophenes as appetite suppressants
US5100891A (en) * 1991-01-18 1992-03-31 Hoechst-Roussel Pharmaceuticals Inc. Substituted 1,2,3,4-tetrahydrocyclopent[b]indoles, 1,2,3,3a,4,8a-hexahydrocyclopent[B]indoles and related compounds
KR20000057418A (ko) * 1996-12-06 2000-09-15 스티븐 에프. 웨인스톡 벤조피라노피롤 및 벤조피라노피리딘 알파-1 아드레날린성화합물
DE69829317T2 (de) 1997-12-25 2006-04-06 Meiji Seika Kaisha Ltd. Tetrahydrobenzindol-derivate
DE69918148T2 (de) * 1998-10-06 2005-07-28 Janssen Pharmaceutica N.V. Trizyclische delta3-pyridine als arzneimittel

Also Published As

Publication number Publication date
DE69905478T2 (de) 2004-03-18
EE04770B1 (et) 2007-02-15
PT1119571E (pt) 2003-06-30
UA69420C2 (uk) 2004-09-15
HUP0104002A2 (hu) 2002-03-28
JP4590101B2 (ja) 2010-12-01
CN1131230C (zh) 2003-12-17
AU6334199A (en) 2000-04-26
HK1038010A1 (en) 2002-03-01
EP1119571A2 (en) 2001-08-01
KR20010071843A (ko) 2001-07-31
SK285585B6 (sk) 2007-04-05
SK4322001A3 (en) 2002-01-07
EE200100209A (et) 2002-06-17
DK1119571T3 (da) 2003-05-26
BG105332A (en) 2001-11-30
NZ510115A (en) 2002-11-26
CN1332744A (zh) 2002-01-23
US6495555B1 (en) 2002-12-17
AU760502B2 (en) 2003-05-15
CZ20011104A3 (cs) 2001-12-12
ES2193751T3 (es) 2003-11-01
BR9913507A (pt) 2001-06-05
TWI248441B (en) 2006-02-01
WO2000020421A2 (en) 2000-04-13
WO2000020421A3 (en) 2000-08-03
DE69905478D1 (de) 2003-03-27
RU2230744C2 (ru) 2004-06-20
BG64872B1 (bg) 2006-07-31
EP1119571B1 (en) 2003-02-19
CA2345622A1 (en) 2000-04-13
PL347894A1 (en) 2002-04-22
NO20011270L (no) 2001-03-13
HUP0104002A3 (en) 2003-12-29
NO20011270D0 (no) 2001-03-13
SI1119571T1 (en) 2003-08-31
AR024216A1 (es) 2002-09-25
IL142443A0 (en) 2002-03-10
CA2345622C (en) 2007-12-04
ATE232869T1 (de) 2003-03-15
TR200100952T2 (tr) 2001-10-22
JP2002526545A (ja) 2002-08-20

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