FR08C0051I2 - Oxazolidinones substituees et leur utilisation dans le domaine de la coagulation sanguine - Google Patents

Oxazolidinones substituees et leur utilisation dans le domaine de la coagulation sanguine

Info

Publication number
FR08C0051I2
FR08C0051I2 FR08C0051C FR08C0051C FR08C0051I2 FR 08C0051 I2 FR08C0051 I2 FR 08C0051I2 FR 08C0051 C FR08C0051 C FR 08C0051C FR 08C0051 C FR08C0051 C FR 08C0051C FR 08C0051 I2 FR08C0051 I2 FR 08C0051I2
Authority
FR
France
Prior art keywords
oxazolidinones
substitute
field
blood coagulation
coagulation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
FR08C0051C
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer AG
Original Assignee
Bayer Healthcare AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=7934434&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FR08C0051(I2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Publication of FR08C0051I1 publication Critical patent/FR08C0051I1/fr
Application filed by Bayer Healthcare AG filed Critical Bayer Healthcare AG
Application granted granted Critical
Publication of FR08C0051I2 publication Critical patent/FR08C0051I2/fr
Active legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/04—Antihaemorrhagics; Procoagulants; Haemostatic agents; Antifibrinolytic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Epidemiology (AREA)
  • Neurology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Immunology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Vascular Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
FR08C0051C 1999-12-24 2008-12-11 Oxazolidinones substituees et leur utilisation dans le domaine de la coagulation sanguine Active FR08C0051I2 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19962924A DE19962924A1 (de) 1999-12-24 1999-12-24 Substituierte Oxazolidinone und ihre Verwendung
PCT/EP2000/012492 WO2001047919A1 (fr) 1999-12-24 2000-12-11 Oxazolidinones substituees et leur utilisation dans le domaine de la coagulation sanguine

Publications (2)

Publication Number Publication Date
FR08C0051I1 FR08C0051I1 (fr) 2008-10-17
FR08C0051I2 true FR08C0051I2 (fr) 2009-12-18

Family

ID=7934434

Family Applications (1)

Application Number Title Priority Date Filing Date
FR08C0051C Active FR08C0051I2 (fr) 1999-12-24 2008-12-11 Oxazolidinones substituees et leur utilisation dans le domaine de la coagulation sanguine

Country Status (50)

Country Link
US (8) US7157456B2 (fr)
EP (2) EP1526132B1 (fr)
JP (2) JP4143297B2 (fr)
KR (3) KR20070094672A (fr)
CN (3) CN1900074B (fr)
AR (1) AR032436A1 (fr)
AT (1) ATE289605T1 (fr)
AU (2) AU775126C (fr)
BE (1) BE2008C046I2 (fr)
BG (1) BG65683B1 (fr)
BR (1) BR0017050B1 (fr)
CA (1) CA2396561C (fr)
CO (1) CO5251440A1 (fr)
CU (2) CU23208A3 (fr)
CY (2) CY2008019I2 (fr)
CZ (1) CZ301432B6 (fr)
DE (3) DE19962924A1 (fr)
DK (2) DK1261606T3 (fr)
DO (2) DOP2000000114A (fr)
EE (1) EE05169B1 (fr)
ES (2) ES2237497T3 (fr)
FR (1) FR08C0051I2 (fr)
GT (1) GT200000216A (fr)
HK (3) HK1057556A1 (fr)
HN (1) HN2000000267A (fr)
HR (2) HRP20020617B1 (fr)
HU (1) HU226522B1 (fr)
IL (2) IL149896A0 (fr)
LT (1) LTC1261606I2 (fr)
LU (1) LU91497I2 (fr)
MA (1) MA25646A1 (fr)
MX (1) MXPA02006241A (fr)
MY (1) MY140488A (fr)
NL (1) NL300370I2 (fr)
NO (4) NO323699B1 (fr)
NZ (2) NZ519730A (fr)
PE (1) PE20010963A1 (fr)
PL (2) PL200413B1 (fr)
PT (2) PT1261606E (fr)
RU (1) RU2297415C2 (fr)
SG (1) SG130939A1 (fr)
SI (2) SI1261606T1 (fr)
SK (1) SK287272B6 (fr)
SV (1) SV2002000245A (fr)
TR (2) TR200401314T2 (fr)
TW (2) TWI277615B (fr)
UA (1) UA73339C2 (fr)
UY (1) UY34152A (fr)
WO (1) WO2001047919A1 (fr)
ZA (1) ZA200204188B (fr)

Families Citing this family (247)

* Cited by examiner, † Cited by third party
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TWI226330B (en) 2005-01-11
NZ519730A (en) 2005-02-25
LTC1261606I2 (lt) 2021-05-10
US7585860B2 (en) 2009-09-08
TW200422299A (en) 2004-11-01
RU2297415C2 (ru) 2007-04-20
GT200000216A (es) 2002-06-12
CN100549008C (zh) 2009-10-14
EE200200341A (et) 2003-10-15
LU91497I9 (fr) 2019-01-02
WO2001047919A1 (fr) 2001-07-05
US20100137274A1 (en) 2010-06-03
NO2009001I1 (no) 2009-02-02
EE05169B1 (et) 2009-06-15
US8129378B2 (en) 2012-03-06
JP2003519141A (ja) 2003-06-17
LU91497I2 (fr) 2009-01-19
IL149896A0 (en) 2002-11-10
PT1261606E (pt) 2005-07-29
CN1900074B (zh) 2012-07-11
US7592339B2 (en) 2009-09-22
US8822458B2 (en) 2014-09-02
FR08C0051I1 (fr) 2008-10-17
BG65683B1 (bg) 2009-06-30
CO5251440A1 (es) 2003-02-28
CY2008019I1 (el) 2009-11-04
HK1092140A1 (en) 2007-02-02
HK1103235A1 (en) 2007-12-14
MY140488A (en) 2009-12-31
MA25646A1 (fr) 2002-12-31
NO2021009I1 (no) 2021-02-25
EP1526132A2 (fr) 2005-04-27
HRP20060251B1 (hr) 2016-08-12
SG130939A1 (en) 2007-04-26
ZA200204188B (en) 2003-05-27
CN1262551C (zh) 2006-07-05
PT1526132E (pt) 2014-04-15
SI1526132T1 (sl) 2014-07-31
PL355665A1 (en) 2004-05-04
JP2005068164A (ja) 2005-03-17
SI1261606T1 (fr) 2005-08-31
CU23208A3 (es) 2007-06-20
DOP2008000001A (es) 2010-01-15
HUP0203902A2 (hu) 2003-03-28
IL205242A0 (en) 2011-07-31
NO20070981L (no) 2002-08-14
NZ537058A (en) 2006-04-28
CA2396561A1 (fr) 2001-07-05
US20130005701A1 (en) 2013-01-03
PL200413B1 (pl) 2009-01-30
NO323699B1 (no) 2007-06-25
EP1526132B1 (fr) 2014-03-12
NO20023043L (no) 2002-08-14
DK1261606T3 (da) 2005-05-09
LTPA2008018I1 (lt) 2021-04-12
WO2001047919A9 (fr) 2002-12-19
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BG106825A (en) 2003-02-28
CY2008019I2 (el) 2009-11-04

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