RU2017123878A - Пиколинамидные соединения с фунгицидной активностью - Google Patents
Пиколинамидные соединения с фунгицидной активностью Download PDFInfo
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- RU2017123878A RU2017123878A RU2017123878A RU2017123878A RU2017123878A RU 2017123878 A RU2017123878 A RU 2017123878A RU 2017123878 A RU2017123878 A RU 2017123878A RU 2017123878 A RU2017123878 A RU 2017123878A RU 2017123878 A RU2017123878 A RU 2017123878A
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- alkyl
- hydrogen
- optionally substituted
- aryl
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
- C07C271/06—Esters of carbamic acids
- C07C271/08—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
- C07C271/10—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C271/22—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of hydrocarbon radicals substituted by carboxyl groups
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
- A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
- A01N47/10—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
- A01N47/18—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof containing a —O—CO—N< group, or a thio analogue thereof, directly attached to a heterocyclic or cycloaliphatic ring
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N37/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids
- A01N37/44—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids containing at least one carboxylic group or a thio analogue, or a derivative thereof, and a nitrogen atom attached to the same carbon skeleton by a single or double bond, this nitrogen atom not being a member of a derivative or of a thio analogue of a carboxylic group, e.g. amino-carboxylic acids
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
- A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/81—Amides; Imides
Claims (45)
1. Соединение формулы I
I
где X представляет собой водород или C(О)R5;
Y представляет собой водород, C(O)R5 или Q;
Q представляет собой
R1 и R11 независимо выбраны из водорода или алкила, необязательно замещенного 0, 1 или несколькими R8; альтернативно, R1 и R11 могут быть взяты вместе с образованием 3-6-членного насыщенного или частично насыщенного карбоцикла или гетероцикла, необязательно замещенного 0, 1 или несколькими R8;
R2 и R12 независимо выбраны из водорода, алкила, арила или алкенила, каждый необязательно замещен 0, 1 или несколькими R8;
R3 выбран из водорода, C2-C6 алкила, арила или алкенила, каждый необязательно замещен 0, 1 или несколькими R8;
R4 выбран из алкила, арила или ацила, каждый необязательно замещен 0, 1 или несколькими R8;
R5 выбран из алкокси или бензилокси, каждый необязательно замещен 0, 1 или несколькими R8;
R6 выбран из водорода, алкокси или галогена, каждый необязательно замещен 0, 1 или несколькими R8;
R7 выбран из водорода, -С(О)R9 или -CH2OC(О)R9;
R8 выбран из водорода, алкила, арила, ацила, галогена, алкенила, алкокси или гетероциклила, каждый необязательно замещен 0, 1 или несколькими R10;
R9 выбран из алкила, алкокси или арила, каждый необязательно замещен 0, 1 или несколькими R8;
R10 выбран из водорода, алкила, арила, ацила, галогена, алкенила, алкокси или гетероциклила.
2. Соединение по п.1, где Х и Y представляют собой водород.
3. Соединение по п.2, где R1 и R11 независимо выбраны из водорода или алкила.
4. Соединение по п.2, где R2 и R12 независимо выбраны из водорода или алкила.
5. Соединение по п.2, где R3 выбран из C2-C6 алкила, арила или алкенила, каждый необязательно замещен 0, 1 или несколькими R8.
6. Соединение по п.2, где R4 выбран из алкила или арила, каждый необязательно замещен 0, 1 или несколькими R8.
7. Соединение по п.2, где R1 и R11 независимо выбраны из водорода или алкила, R2 и R12 независимо выбраны из водорода или алкила, R3 выбран из C2-C6 алкила, арила или алкенила, каждый необязательно замещен 0, 1 или несколькими R8, и R4 выбран из алкила или арила, каждый необязательно замещен 0, 1 или несколькими R8.
8. Соединение по п.1, где Х представляет собой C(O)R5, и Y представляет собой водород.
9. Соединение по п.8, где R1 и R11 независимо выбраны из водорода или алкила.
10. Соединение по п.8, где R2 и R12 независимо выбраны из водорода или алкила.
11. Соединение по п.8, где R3 выбран из C2-C6 алкила, арила или алкенила, каждый необязательно замещен 0, 1 или несколькими R8.
12. Соединение по п.8, где R4 выбран из алкила или арила, каждый необязательно замещен 0, 1 или несколькими R8.
13. Соединение по п.8, где R1 и R11 независимо выбраны из водорода или алкила, R2 и R12 независимо выбраны из водорода или алкила, R3 выбран из C2-C6 алкила, арила или алкенила, каждый необязательно замещен 0, 1 или несколькими R8, и R4 выбран из алкила или арила, каждый необязательно замещен 0, 1 или несколькими R8.
14. Соединение по п.1, где X представляет собой водород и Y представляет собой Q.
15. Соединение по п.14, где R6 представляет собой алкокси.
16. Соединение по п.15, где R7 представляет собой водород.
17. Соединение по п.16, где R1 и R11 независимо выбраны из водорода или алкила.
18. Соединение по п.16, где R2 и R12 независимо выбраны из водорода или алкила.
19. Соединение по п.16, где R3 выбран из C2-C6 алкила, арила или алкенила, каждый необязательно замещен 0, 1 или несколькими R8.
20. Соединение по п.16, где R4 выбран из алкила или арила, каждый необязательно замещен 0, 1 или несколькими R8.
21. Соединение по п.16, где R1 и R11 независимо выбраны из водорода или алкила, R2 и R12 независимо выбраны из водорода или алкила, R3 выбран из C2-C6 алкила, арила или алкенила, каждый необязательно замещен 0, 1 или несколькими R8, и R4 выбран из алкила или арила, каждый необязательно замещен 0, 1 или несколькими R8.
22. Соединение по п.15, где R7 выбран из -C(O)R9 или -CH2OC(O)R9.
23. Соединение по п.22, где R9 представляет собой алкил, необязательно замещенный 0, 1 или несколькими R8.
24. Соединение по п.23, где R1 и R11 независимо выбраны из водорода или алкила.
25. Соединение по п.23, где R2 и R12 независимо выбраны из водорода или алкила.
26. Соединение по п.23, где R3 выбран из алкила, арила или алкенила, каждый необязательно замещен 0, 1 или несколькими R8.
27. Соединение по п.23, где R4 выбран из алкила или арила, каждый необязательно замещен 0, 1 или несколькими R8.
28. Соединение по п.23, где R1 и R11 независимо выбраны из водорода или алкила, R2 и R12 независимо выбраны из водорода или алкила, R3 выбран из C2-C6 алкила, арила или алкенила, каждый необязательно замещен 0, 1 или несколькими R8, и R4 выбран из алкила или арила, каждый необязательно замещен 0, 1 или несколькими R8.
29. Соединение по п.28, где R9 выбран из -CH3, -CH2OCH2CH3, -CH2CH2OCH3, -CH(CH3)2, -CH2CH2CH2CH3, -циклопропила.
Applications Claiming Priority (17)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201462098097P | 2014-12-30 | 2014-12-30 | |
US201462098089P | 2014-12-30 | 2014-12-30 | |
US62/098,097 | 2014-12-30 | ||
US62/098,089 | 2014-12-30 | ||
US201562255168P | 2015-11-13 | 2015-11-13 | |
US201562255152P | 2015-11-13 | 2015-11-13 | |
US201562255163P | 2015-11-13 | 2015-11-13 | |
US201562255125P | 2015-11-13 | 2015-11-13 | |
US201562255131P | 2015-11-13 | 2015-11-13 | |
US201562255144P | 2015-11-13 | 2015-11-13 | |
US62/255,152 | 2015-11-13 | ||
US62/255,163 | 2015-11-13 | ||
US62/255,131 | 2015-11-13 | ||
US62/255,144 | 2015-11-13 | ||
US62/255,125 | 2015-11-13 | ||
US62/255,168 | 2015-11-13 | ||
PCT/US2015/067113 WO2016109289A1 (en) | 2014-12-30 | 2015-12-21 | Picolinamide compounds with fungicidal activity |
Publications (3)
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RU2017123878A true RU2017123878A (ru) | 2019-01-31 |
RU2017123878A3 RU2017123878A3 (ru) | 2019-02-20 |
RU2687160C2 RU2687160C2 (ru) | 2019-05-07 |
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RU2017123854A RU2704867C2 (ru) | 2014-12-30 | 2015-12-21 | Применение соединений пиколинамида с фунгицидным действием |
RU2017123878A RU2687160C2 (ru) | 2014-12-30 | 2015-12-21 | Пиколинамидные соединения с фунгицидной активностью |
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RU2017123854A RU2704867C2 (ru) | 2014-12-30 | 2015-12-21 | Применение соединений пиколинамида с фунгицидным действием |
Country Status (17)
Country | Link |
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US (2) | US10433555B2 (ru) |
EP (2) | EP3240413B1 (ru) |
JP (2) | JP6742319B2 (ru) |
KR (2) | KR20170099930A (ru) |
CN (2) | CN107427000A (ru) |
AU (4) | AU2015374459A1 (ru) |
BR (1) | BR112017013653A2 (ru) |
CA (2) | CA2972413A1 (ru) |
CO (2) | CO2017006852A2 (ru) |
IL (2) | IL253092A0 (ru) |
MX (2) | MX2017008407A (ru) |
NZ (2) | NZ732573A (ru) |
RU (2) | RU2704867C2 (ru) |
TW (2) | TW201625539A (ru) |
UY (2) | UY36489A (ru) |
WO (2) | WO2016109289A1 (ru) |
ZA (2) | ZA201704555B (ru) |
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BR112017013653A2 (pt) | 2014-12-30 | 2018-03-13 | Dow Agrosciences Llc | uso de compostos de picolinamida com atividade fungicida |
RU2702088C2 (ru) | 2014-12-30 | 2019-10-03 | ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи | Применение соединений пиколинамида в качестве фунгицидов |
CN107205397A (zh) | 2014-12-30 | 2017-09-26 | 美国陶氏益农公司 | 具有杀真菌活性的吡啶酰胺化合物的用途 |
CN107205385A (zh) * | 2014-12-30 | 2017-09-26 | 美国陶氏益农公司 | 吡啶酰胺作为杀真菌剂的用途 |
KR20170100547A (ko) | 2014-12-30 | 2017-09-04 | 다우 아그로사이언시즈 엘엘씨 | 살진균 활성을 갖는 피콜린아미드 |
US10173982B2 (en) | 2016-08-30 | 2019-01-08 | Dow Agrosciences Llc | Picolinamides as fungicides |
TW201808905A (zh) * | 2016-08-30 | 2018-03-16 | 美商陶氏農業科學公司 | 具有殺真菌活性的硫代吡啶醯胺化合物 |
WO2018045012A1 (en) | 2016-08-30 | 2018-03-08 | Dow Agrosciences Llc | Pyrido-1,3-oxazine-2,4-dione compounds with fungicidal activity |
US10172358B2 (en) | 2016-08-30 | 2019-01-08 | Dow Agrosciences Llc | Thiopicolinamide compounds with fungicidal activity |
WO2018045006A1 (en) | 2016-08-30 | 2018-03-08 | Dow Agrosciences Llc | Picolinamide n-oxide compounds with fungicidal activity |
BR102018000183B1 (pt) * | 2017-01-05 | 2023-04-25 | Dow Agrosciences Llc | Picolinamidas, composição para controle de um patógeno fúngico, e método para controle e prevenção de um ataque por fungos em uma planta |
EP3603668A4 (en) | 2017-03-29 | 2021-01-06 | Terumo Kabushiki Kaisha | ADDITIVE COMPOSITION, VACCINE COMPOSITION AND MEDICINAL KIT WITH IT |
TWI774761B (zh) | 2017-05-02 | 2022-08-21 | 美商科迪華農業科技有限責任公司 | 用於穀物中的真菌防治之協同性混合物 |
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UY37912A (es) | 2017-10-05 | 2019-05-31 | Syngenta Participations Ag | Derivados de picolinamida fungicidas que portan grupos terminales heteroarilo o heteroariloxi |
US11459318B2 (en) | 2017-10-06 | 2022-10-04 | Syngenta Participations Ag | Pesticidally active pyrrole derivatives |
CN111344279B (zh) * | 2017-11-15 | 2023-07-07 | 先正达参股股份有限公司 | 杀微生物的吡啶酰胺衍生物 |
WO2019121149A1 (en) | 2017-12-19 | 2019-06-27 | Syngenta Participations Ag | Microbiocidal picolinamide derivatives |
BR102019004480B1 (pt) | 2018-03-08 | 2023-03-28 | Dow Agrosciences Llc | Picolinamidas como fungicidas |
US11629129B2 (en) | 2018-05-25 | 2023-04-18 | Syngenta Participations Ag | Microbiocidal picolinamide derivatives |
BR112021006669A2 (pt) | 2018-10-15 | 2021-07-06 | Dow Agrosciences Llc | métodos para síntese de oxipicolinamidas |
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