PH17194A - Novel carbostyril derivatives,and pharmaceutical composition containing the same - Google Patents

Novel carbostyril derivatives,and pharmaceutical composition containing the same

Info

Publication number
PH17194A
PH17194A PH25264A PH25264A PH17194A PH 17194 A PH17194 A PH 17194A PH 25264 A PH25264 A PH 25264A PH 25264 A PH25264 A PH 25264A PH 17194 A PH17194 A PH 17194A
Authority
PH
Philippines
Prior art keywords
same
pharmaceutical composition
composition containing
carbostyril derivatives
novel carbostyril
Prior art date
Application number
PH25264A
Other languages
English (en)
Inventor
Kazuo Banno
Masaaki Osaki
Kazutuki Nakagawa
Takafumi Fujioka
Original Assignee
Otsuka Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP2880580A external-priority patent/JPS56125370A/ja
Priority claimed from JP11502280A external-priority patent/JPS5738772A/ja
Application filed by Otsuka Pharma Co Ltd filed Critical Otsuka Pharma Co Ltd
Publication of PH17194A publication Critical patent/PH17194A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20—Oxygen atoms
    • C07D215/22—Oxygen atoms attached in position 2 or 4
    • C07D215/227—Oxygen atoms attached in position 2 or 4 only one oxygen atom which is attached in position 2

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
PH25264A 1980-03-06 1981-02-25 Novel carbostyril derivatives,and pharmaceutical composition containing the same PH17194A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2880580A JPS56125370A (en) 1980-03-06 1980-03-06 Carbostyril derivative
JP11502280A JPS5738772A (en) 1980-08-20 1980-08-20 Carbostyril derivative

Publications (1)

Publication Number Publication Date
PH17194A true PH17194A (en) 1984-06-19

Family

ID=26366952

Family Applications (1)

Application Number Title Priority Date Filing Date
PH25264A PH17194A (en) 1980-03-06 1981-02-25 Novel carbostyril derivatives,and pharmaceutical composition containing the same

Country Status (21)

Country Link
US (4) US4455422A (ru)
AT (1) AT381307B (ru)
AU (1) AU523005B2 (ru)
BE (1) BE887800A (ru)
CA (1) CA1155119A (ru)
CH (1) CH647775A5 (ru)
DE (2) DE3107601A1 (ru)
DK (1) DK155282C (ru)
ES (4) ES8301962A1 (ru)
FI (1) FI76323C (ru)
FR (1) FR2477542A1 (ru)
GB (1) GB2071094B (ru)
IT (1) IT1144315B (ru)
MX (1) MX6980E (ru)
NL (1) NL184364C (ru)
NO (1) NO159531C (ru)
PH (1) PH17194A (ru)
PT (1) PT72622B (ru)
RU (1) RU1779249C (ru)
SE (1) SE447255B (ru)
SU (1) SU1367857A3 (ru)

Families Citing this family (57)

* Cited by examiner, † Cited by third party
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PH17194A (en) * 1980-03-06 1984-06-19 Otsuka Pharma Co Ltd Novel carbostyril derivatives,and pharmaceutical composition containing the same
FI77852C (fi) * 1981-02-17 1989-05-10 Otsuka Pharma Co Ltd Foerfarande foer framstaellning av nya, saosom hjaertmediciner anvaendbara substituerade amid- och (maettad heterocykel)karbonylkarbostyrilderivat.
AU532361B2 (en) * 1981-09-01 1983-09-29 Otsuka Pharmaceutical Co., Ltd. Carbostyril derivatives
FI80022C (fi) * 1982-07-05 1990-04-10 Otsuka Pharma Co Ltd Foerfarande foer framstaellning av ett nytt, terapeutiskt anvaendbart karbostyrilderivat.
CH655110A5 (de) * 1982-09-03 1986-03-27 Otsuka Pharma Co Ltd Carbostyrilderivate, verfahren zu deren herstellung und arzneimittel, welche diese enthalten.
DE3434271A1 (de) * 1984-09-19 1986-03-20 Beiersdorf Ag, 2000 Hamburg Substituierte 3,4-dihydro-chinolin-2(1h)-one verfahren zu ihrer herstellung und ihre verwendung sowie diese verbindungen enthaltende zubereitungen
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US5147881A (en) * 1990-11-14 1992-09-15 Pfizer Inc 4-(1,2-benzisoxazolyl)piperidine antipsychotic agents
US5189171A (en) * 1991-06-21 1993-02-23 American Home Products Corporation Antipsychotic benzodioxan derivatives
US5166367A (en) * 1991-06-21 1992-11-24 American Home Products Corporation Antipsychotic benzodioxan derivatives
PL169884B1 (pl) * 1991-07-17 1996-09-30 Pfizer Sposób wytwarzania nowych pochodnych 2-(4-hydroksypiperydyno)-1-alkanolowych PL PL PL
US6255322B1 (en) 1992-06-19 2001-07-03 Pfizer Inc. 2-(4-hydroxypiperidino)-1-alkanol derivatives as antiischemic agents
WO1994022826A1 (en) * 1993-04-07 1994-10-13 Otsuka Pharmaceutical Co., Ltd. Peripheral vasodilating agent containing n-acylated 4-amino piperidine derivatives as active ingredients
DK0709384T3 (da) * 1994-10-31 1999-08-23 Merck Patent Gmbh Benzylpiperidinderivater med høj affinitet til aminosyrereceptorers bindingssteder
ZA9610736B (en) * 1995-12-22 1997-06-27 Warner Lambert Co 2-Substituted piperidine analogs and their use as subtypeselective nmda receptor antagonists
ZA9610738B (en) 1995-12-22 1997-06-24 Warner Lambert Co Subtype selective nmda receptor ligands and the use thereof
ZA9610745B (en) * 1995-12-22 1997-06-24 Warner Lambert Co 4-Subsituted piperidine analogs and their use as subtype selective nmda receptor antagonists
ZA9610741B (en) * 1995-12-22 1997-06-24 Warner Lambert Co 4-Substituted piperidine analogs and their use as subtype selective nmda receptor antagonists
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FR2823749B1 (fr) * 2001-04-20 2004-02-20 Sanofi Synthelabo Phenyl- et pyridyl-piperidines, procede pour leur preparation et compositions pharmaceutiques les contenant
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DE10210779A1 (de) * 2002-03-12 2003-10-09 Merck Patent Gmbh Cyclische Amide
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MXPA04007776A (es) 2002-03-13 2004-10-15 Janssen Pharmaceutica Nv Derivados de sulfonilamino como nuevos inhibidores de histona deacetilasa.
ATE398105T1 (de) * 2002-03-13 2008-07-15 Janssen Pharmaceutica Nv Carbonylamino- derivativate als neue inhibitoren von histone deacetylase
MY142362A (en) * 2004-01-29 2010-11-30 Otsuka Pharma Co Ltd Pharmaceutical composition for promoting angiogenesis
SG156687A1 (en) * 2004-07-28 2009-11-26 Janssen Pharmaceutica Nv Substituted indolyl alkyl amino derivatives as novel inhibitors of histone deacetylase
ME01058B (me) * 2004-07-28 2012-10-20 Janssen Pharmaceutica Nv Supstituisani derivati propenil piperazina kao novi inhibitori histonske deacetilaze
DE602005014646D1 (de) * 2004-07-28 2009-07-09 Janssen Pharmaceutica Nv Substituierte propenylpiperazinderivate als neue inhibitoren von histondeacetylase
TWI320783B (en) 2005-04-14 2010-02-21 Otsuka Pharma Co Ltd Heterocyclic compound
EP1885710B1 (en) 2005-05-18 2015-08-19 Janssen Pharmaceutica N.V. Substituted aminopropenyl piperidine or morpholine derivatives as novel inhibitors of histone deacetylase
JP5225104B2 (ja) * 2006-01-19 2013-07-03 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ 新しい、ヒストンデアセチラーゼのインヒビターとしてのアミノフェニル誘導体
US8101616B2 (en) * 2006-01-19 2012-01-24 Janssen Pharmaceutica N.V. Pyridine and pyrimidine derivatives as inhibitors of histone deacetylase
CN101370803B (zh) * 2006-01-19 2012-12-12 詹森药业有限公司 作为组蛋白脱乙酰酶抑制剂的取代的吲哚基-烷基-氨基衍生物
JP5247470B2 (ja) 2006-01-19 2013-07-24 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ ヒストンデアセチラーゼのインヒビターとしてのピリジン及びピリミジン誘導体
US7935706B2 (en) * 2006-02-23 2011-05-03 Shionogi & Co., Ltd. Nitrogen-containing heterocycle derivatives substituted with cyclic group
WO2009034029A2 (de) * 2007-09-07 2009-03-19 Boehringer Ingelheim International Gmbh 1-substituierte 4 -heterocyclylpiperidine als cgrp antagonisten
AU2010217772B2 (en) * 2009-02-26 2014-10-23 Reviva Pharmaceuticals, Inc. Compositions, synthesis, and methods of utilizing arylpiperazine derivatives
CA2872883A1 (en) * 2012-05-09 2013-11-14 Sunovion Pharmaceuticals Inc. Heteroaryl compounds and methods of use thereof
CN106608875A (zh) 2015-10-26 2017-05-03 江苏恩华药业股份有限公司 一种稠和杂环类衍生物合成及其应用
CN108031471A (zh) * 2017-10-27 2018-05-15 苏州盖德精细材料有限公司 一种静电纺丝制备的负载型纳米纤维催化剂及其在3,5-二羟基甲苯制备中的应用
CN114409680B (zh) * 2018-01-19 2023-11-21 上海怡立舍生物技术有限公司 Ppar激动剂及其应用
CN116554127A (zh) * 2022-01-28 2023-08-08 成都麻沸散医药科技有限公司 哌嗪取代苯酚类衍生物及其用途

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US3910924A (en) * 1972-04-13 1975-10-07 Otsuka Pharma Co Ltd 3,4-Dihydrocarbostyril derivatives and a process for preparing the same
JPS5239035B2 (ru) * 1972-12-14 1977-10-03
US4068076A (en) * 1972-12-29 1978-01-10 Otsuka Pharmaceutical Co., Ltd. 5-(1-Hydroxy-2-(heterocyclic amino))ethyl-8-hydroxy-3,4-dihydrocarbostyril derivatives
US4022784A (en) * 1974-01-31 1977-05-10 Otsuka Pharmaceutical Company Limited 5-[1-Hydroxy-2-(substituted-amino)]alkyl-8-substituted-carbostyril and -3,4-dihydrocarbostyril derivatives
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DE2827566A1 (de) * 1978-06-23 1980-01-10 Boehringer Mannheim Gmbh 1,2-dihydro-chinolin-2-on-derivate und verfahren zu ihrer herstellung
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PH17194A (en) * 1980-03-06 1984-06-19 Otsuka Pharma Co Ltd Novel carbostyril derivatives,and pharmaceutical composition containing the same
FI77852C (fi) * 1981-02-17 1989-05-10 Otsuka Pharma Co Ltd Foerfarande foer framstaellning av nya, saosom hjaertmediciner anvaendbara substituerade amid- och (maettad heterocykel)karbonylkarbostyrilderivat.
AU532361B2 (en) * 1981-09-01 1983-09-29 Otsuka Pharmaceutical Co., Ltd. Carbostyril derivatives

Also Published As

Publication number Publication date
AT381307B (de) 1986-09-25
FR2477542B1 (ru) 1983-09-09
GB2071094B (en) 1984-09-26
MX6980E (es) 1987-01-19
US4567187A (en) 1986-01-28
SU1367857A3 (ru) 1988-01-15
ES500137A0 (es) 1982-11-01
FR2477542A1 (fr) 1981-09-11
DE3107601C2 (ru) 1989-07-20
IT8167311A0 (it) 1981-03-05
FI76323B (fi) 1988-06-30
AU6797381A (en) 1981-09-10
CA1155119A (en) 1983-10-11
ES509659A0 (es) 1983-05-01
NO810765L (no) 1981-09-07
NL184364C (nl) 1989-07-03
FI810669L (fi) 1981-09-07
ES509658A0 (es) 1983-04-01
PT72622B (en) 1982-06-15
ES518667A0 (es) 1984-06-16
SE447255B (sv) 1986-11-03
US4619932A (en) 1986-10-28
IT1144315B (it) 1986-10-29
NL184364B (nl) 1989-02-01
ES8301962A1 (es) 1982-11-01
AU523005B2 (en) 1982-07-08
ES8305356A1 (es) 1983-04-01
ATA98481A (de) 1986-02-15
FI76323C (fi) 1988-10-10
DE3152880C2 (ru) 1990-03-22
US4455422A (en) 1984-06-19
SE8101409L (sv) 1981-09-07
BE887800A (fr) 1981-09-07
DK99781A (da) 1981-09-07
GB2071094A (en) 1981-09-16
DE3107601A1 (de) 1982-02-04
NL8101099A (nl) 1981-10-01
DK155282C (da) 1989-08-07
RU1779249C (ru) 1992-11-30
CH647775A5 (de) 1985-02-15
ES8306141A1 (es) 1983-05-01
US4460593A (en) 1984-07-17
PT72622A (en) 1981-04-01
NO159531B (no) 1988-10-03
DK155282B (da) 1989-03-20
ES8405782A1 (es) 1984-06-16
NO159531C (no) 1989-01-11

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