MXPA02007632A - Derivados de 2-benzotiazolil urea y su uso como inhibidores de proteina cinasa. - Google Patents
Derivados de 2-benzotiazolil urea y su uso como inhibidores de proteina cinasa.Info
- Publication number
- MXPA02007632A MXPA02007632A MXPA02007632A MXPA02007632A MXPA02007632A MX PA02007632 A MXPA02007632 A MX PA02007632A MX PA02007632 A MXPA02007632 A MX PA02007632A MX PA02007632 A MXPA02007632 A MX PA02007632A MX PA02007632 A MXPA02007632 A MX PA02007632A
- Authority
- MX
- Mexico
- Prior art keywords
- protein kinase
- kinase inhibitors
- urea derivatives
- inhibitors
- benzothiazolyl urea
- Prior art date
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Abstract
La presente invencion es dirigida a un compuesto de formula (l), mezclas racemicas-diastereomericas del mismo, isomeros opticos del mismo, promedicamentos del mismo, isotopos del mismo o sales farmaceuticamente aceptables de dicho compuesto, isomeros, promedicamentos e isotopos, en donde las variables son definidas en la presente. Los compuestos de esta invencion son utiles como inhibidores de serina/treonina y tirosina cinasas. En particular, compuestos de esta invencion son utiles como inhibidores de tirosina cinasas, que son importantes en enfermedades hiper-proliferativas, especialmente en cancer y en el proceso de angiogenesis. (ver formula).
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
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US18084100P | 2000-02-07 | 2000-02-07 | |
PCT/US2001/003803 WO2001057008A1 (en) | 2000-02-07 | 2001-02-06 | 2-benzothiazolyl urea derivatives and their use as protein kinase inhibitors |
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-
2001
- 2001-02-06 JP JP2001556858A patent/JP2003521543A/ja not_active Withdrawn
- 2001-02-06 BR BR0108085-7A patent/BR0108085A/pt not_active Application Discontinuation
- 2001-02-06 PL PL01357099A patent/PL357099A1/xx not_active Application Discontinuation
- 2001-02-06 IL IL15104501A patent/IL151045A0/xx unknown
- 2001-02-06 HU HU0300359A patent/HUP0300359A2/hu unknown
- 2001-02-06 EP EP01908878A patent/EP1254123A1/en not_active Withdrawn
- 2001-02-06 MX MXPA02007632A patent/MXPA02007632A/es unknown
- 2001-02-06 CA CA002398754A patent/CA2398754A1/en not_active Abandoned
- 2001-02-06 KR KR1020027010188A patent/KR20020084116A/ko not_active Application Discontinuation
- 2001-02-06 SK SK1271-2002A patent/SK12712002A3/sk unknown
- 2001-02-06 AU AU2001236698A patent/AU2001236698A1/en not_active Abandoned
- 2001-02-06 WO PCT/US2001/003803 patent/WO2001057008A1/en not_active Application Discontinuation
- 2001-02-06 US US09/777,554 patent/US7091227B2/en not_active Expired - Lifetime
- 2001-02-06 CN CN01807734A patent/CN1422262A/zh active Pending
- 2001-02-07 AR ARP010100543A patent/AR030189A1/es unknown
-
2002
- 2002-08-05 ZA ZA200206235A patent/ZA200206235B/en unknown
- 2002-08-06 NO NO20023713A patent/NO20023713L/no not_active Application Discontinuation
- 2002-09-04 BG BG107062A patent/BG107062A/bg unknown
Also Published As
Publication number | Publication date |
---|---|
IL151045A0 (en) | 2003-04-10 |
SK12712002A3 (sk) | 2003-02-04 |
CN1422262A (zh) | 2003-06-04 |
WO2001057008A1 (en) | 2001-08-09 |
NO20023713L (no) | 2002-10-04 |
ZA200206235B (en) | 2004-02-13 |
KR20020084116A (ko) | 2002-11-04 |
CA2398754A1 (en) | 2001-08-09 |
EP1254123A1 (en) | 2002-11-06 |
BG107062A (bg) | 2003-04-30 |
BR0108085A (pt) | 2003-03-18 |
US7091227B2 (en) | 2006-08-15 |
AU2001236698A1 (en) | 2001-08-14 |
HUP0300359A2 (hu) | 2003-06-28 |
JP2003521543A (ja) | 2003-07-15 |
NO20023713D0 (no) | 2002-08-06 |
PL357099A1 (en) | 2004-07-12 |
AR030189A1 (es) | 2003-08-13 |
US20030153568A1 (en) | 2003-08-14 |
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