HK1172549A1 - Dpp iv inhibitor formulations iv - Google Patents

Dpp iv inhibitor formulations iv

Info

Publication number
HK1172549A1
HK1172549A1 HK12113310.2A HK12113310A HK1172549A1 HK 1172549 A1 HK1172549 A1 HK 1172549A1 HK 12113310 A HK12113310 A HK 12113310A HK 1172549 A1 HK1172549 A1 HK 1172549A1
Authority
HK
Hong Kong
Prior art keywords
dpp
inhibitor formulations
formulations
inhibitor
Prior art date
Application number
HK12113310.2A
Other languages
English (en)
Chinese (zh)
Inventor
安賈．科爾勞希
帕特里克．羅默
格爾德．塞費爾特
Original Assignee
勃林格殷格翰國際有限公司
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36972901&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1172549(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by 勃林格殷格翰國際有限公司 filed Critical 勃林格殷格翰國際有限公司
Publication of HK1172549A1 publication Critical patent/HK1172549A1/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/38—Cellulose; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
    • A—HUMAN NECESSITIES
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52—Purines, e.g. adenine
    • A61K31/522—Purines, e.g. adenine having oxo groups directly attached to the heterocyclic ring, e.g. hypoxanthine, guanine, acyclovir
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    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A—HUMAN NECESSITIES
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    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/34—Macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyesters, polyamino acids, polysiloxanes, polyphosphazines, copolymers of polyalkylene glycol or poloxamers
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    • A—HUMAN NECESSITIES
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    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/2853—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers, poly(lactide-co-glycolide)
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
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    • A61K9/2893—Tablet coating processes
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K9/00—Medicinal preparations characterised by special physical form
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K9/4891—Coated capsules; Multilayered drug free capsule shells
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    • A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
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    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
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    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
HK12113310.2A 2006-05-04 2009-11-13 Dpp iv inhibitor formulations iv HK1172549A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP06009201A EP1852108A1 (en) 2006-05-04 2006-05-04 DPP IV inhibitor formulations

Publications (1)

Publication Number Publication Date
HK1172549A1 true HK1172549A1 (en) 2013-04-26

Family

ID=36972901

Family Applications (2)

Application Number Title Priority Date Filing Date
HK09110601.1A HK1130442A1 (en) 2006-05-04 2009-11-13 Dpp iv inhibitor formulations
HK12113310.2A HK1172549A1 (en) 2006-05-04 2009-11-13 Dpp iv inhibitor formulations iv

Family Applications Before (1)

Application Number Title Priority Date Filing Date
HK09110601.1A HK1130442A1 (en) 2006-05-04 2009-11-13 Dpp iv inhibitor formulations

Country Status (37)

Country Link
US (8) US20080107731A1 (es)
EP (5) EP1852108A1 (es)
JP (7) JP5478244B2 (es)
KR (5) KR101855323B1 (es)
CN (2) CN102526737B (es)
AR (2) AR060755A1 (es)
AT (1) ATE480228T1 (es)
AU (1) AU2007247193B2 (es)
BR (2) BRPI0711179B1 (es)
CA (1) CA2649922C (es)
CL (2) CL2012002521A1 (es)
CY (2) CY1111354T1 (es)
DE (1) DE602007009091D1 (es)
DK (3) DK2277509T5 (es)
EA (2) EA016559B1 (es)
EC (1) ECSP088800A (es)
ES (3) ES2527409T4 (es)
HK (2) HK1130442A1 (es)
HR (2) HRP20100507T1 (es)
HU (1) HUE025210T2 (es)
IL (2) IL195030A (es)
ME (2) ME01170B (es)
MX (2) MX358617B (es)
MY (2) MY146969A (es)
NO (1) NO343067B1 (es)
NZ (3) NZ613426A (es)
PE (2) PE20080698A1 (es)
PL (3) PL2283819T3 (es)
PT (2) PT2283819E (es)
RS (2) RS51466B (es)
SG (1) SG171649A1 (es)
SI (2) SI2023902T1 (es)
TW (2) TWI520753B (es)
UA (1) UA94942C2 (es)
UY (1) UY30319A1 (es)
WO (1) WO2007128724A1 (es)
ZA (1) ZA200808361B (es)

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