HK1030611A1 - 2-(purin-9-yl)-tetrahydrofuran-3,4-diol derivatives - Google Patents

2-(purin-9-yl)-tetrahydrofuran-3,4-diol derivatives

Info

Publication number
HK1030611A1
HK1030611A1 HK01101621A HK01101621A HK1030611A1 HK 1030611 A1 HK1030611 A1 HK 1030611A1 HK 01101621 A HK01101621 A HK 01101621A HK 01101621 A HK01101621 A HK 01101621A HK 1030611 A1 HK1030611 A1 HK 1030611A1
Authority
HK
Hong Kong
Prior art keywords
purin
tetrahydrofuran
diol derivatives
diol
derivatives
Prior art date
Application number
HK01101621A
Other languages
English (en)
Inventor
Chuen Chan
Richard Peter Charles Cousins
Brian Cox
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9802066.2A external-priority patent/GB9802066D0/en
Priority claimed from GBGB9813528.8A external-priority patent/GB9813528D0/en
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of HK1030611A1 publication Critical patent/HK1030611A1/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16Purine radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A61K31/706Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
    • A61K31/7064Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
    • A61K31/7076Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines containing purines, e.g. adenosine, adenylic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00Processes for the preparation of sugar derivatives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pulmonology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Saccharide Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
HK01101621A 1998-01-31 2001-03-06 2-(purin-9-yl)-tetrahydrofuran-3,4-diol derivatives HK1030611A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB9802066.2A GB9802066D0 (en) 1998-01-31 1998-01-31 Chemical compounds
GBGB9813528.8A GB9813528D0 (en) 1998-06-23 1998-06-23 Chemical compounds
PCT/EP1999/000503 WO1999038877A2 (en) 1998-01-31 1999-01-29 2-(PURIN-9-yl)-TETRAHYDROFURAN-3,4-DIOL DERIVATIVES

Publications (1)

Publication Number Publication Date
HK1030611A1 true HK1030611A1 (en) 2001-05-11

Family

ID=26313042

Family Applications (1)

Application Number Title Priority Date Filing Date
HK01101621A HK1030611A1 (en) 1998-01-31 2001-03-06 2-(purin-9-yl)-tetrahydrofuran-3,4-diol derivatives

Country Status (39)

Country Link
US (1) US6762170B1 (hr)
EP (1) EP1051425B1 (hr)
JP (1) JP2002501928A (hr)
KR (1) KR20010034473A (hr)
CN (1) CN1289338A (hr)
AP (1) AP2000001875A0 (hr)
AR (1) AR014508A1 (hr)
AT (1) ATE226957T1 (hr)
AU (1) AU757183B2 (hr)
BG (1) BG63783B1 (hr)
BR (1) BR9907270A (hr)
CA (1) CA2318278A1 (hr)
CO (1) CO4980872A1 (hr)
DE (1) DE69903708T2 (hr)
DK (1) DK1051425T3 (hr)
EA (1) EA003194B1 (hr)
EE (1) EE200000441A (hr)
ES (1) ES2186330T3 (hr)
GE (1) GEP20022839B (hr)
HK (1) HK1030611A1 (hr)
HR (1) HRP20000511A2 (hr)
HU (1) HUP0101305A3 (hr)
ID (1) ID26326A (hr)
IL (1) IL137042A0 (hr)
IS (1) IS5550A (hr)
MA (1) MA26601A1 (hr)
NO (1) NO20003867L (hr)
NZ (1) NZ505452A (hr)
OA (1) OA11447A (hr)
PE (1) PE20000280A1 (hr)
PL (1) PL342670A1 (hr)
PT (1) PT1051425E (hr)
SI (1) SI1051425T1 (hr)
SK (1) SK11192000A3 (hr)
SV (1) SV1999000009A (hr)
TR (1) TR200002218T2 (hr)
TW (1) TW434250B (hr)
WO (1) WO1999038877A2 (hr)
YU (1) YU44900A (hr)

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Also Published As

Publication number Publication date
WO1999038877A2 (en) 1999-08-05
EP1051425B1 (en) 2002-10-30
EA003194B1 (ru) 2003-02-27
JP2002501928A (ja) 2002-01-22
CN1289338A (zh) 2001-03-28
BR9907270A (pt) 2000-10-24
DE69903708T2 (de) 2003-07-03
SV1999000009A (es) 2000-09-05
AU2719799A (en) 1999-08-16
TW434250B (en) 2001-05-16
NO20003867D0 (no) 2000-07-28
SK11192000A3 (sk) 2001-06-11
BG63783B1 (bg) 2002-12-29
ID26326A (id) 2000-12-14
EE200000441A (et) 2001-12-17
CA2318278A1 (en) 1999-08-05
HUP0101305A3 (en) 2002-08-28
WO1999038877A3 (en) 1999-09-30
NO20003867L (no) 2000-07-28
HRP20000511A2 (en) 2000-12-31
DE69903708D1 (de) 2002-12-05
DK1051425T3 (da) 2003-03-03
AR014508A1 (es) 2001-02-28
AP2000001875A0 (en) 2000-09-30
YU44900A (sh) 2003-01-31
ES2186330T3 (es) 2003-05-01
US6762170B1 (en) 2004-07-13
PE20000280A1 (es) 2000-03-28
CO4980872A1 (es) 2000-11-27
SI1051425T1 (en) 2003-04-30
GEP20022839B (en) 2002-11-25
MA26601A1 (fr) 2004-12-20
PT1051425E (pt) 2003-03-31
KR20010034473A (ko) 2001-04-25
EP1051425A2 (en) 2000-11-15
ATE226957T1 (de) 2002-11-15
IS5550A (is) 2000-06-27
TR200002218T2 (tr) 2000-12-21
BG104729A (en) 2001-04-30
EA200000723A1 (ru) 2001-04-23
OA11447A (en) 2004-04-29
PL342670A1 (en) 2001-07-02
IL137042A0 (en) 2001-06-14
HUP0101305A2 (hu) 2002-04-29
AU757183B2 (en) 2003-02-06
NZ505452A (en) 2003-01-31

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