DZ2300A1 - Dérivés 6,5-hétérobicycliques substitués, procédé pour leur préparation et compositions pharmaceutiques les contenant. - Google Patents

Dérivés 6,5-hétérobicycliques substitués, procédé pour leur préparation et compositions pharmaceutiques les contenant.

Info

Publication number
DZ2300A1
DZ2300A1 DZ970150A DZ970150A DZ2300A1 DZ 2300 A1 DZ2300 A1 DZ 2300A1 DZ 970150 A DZ970150 A DZ 970150A DZ 970150 A DZ970150 A DZ 970150A DZ 2300 A1 DZ2300 A1 DZ 2300A1
Authority
DZ
Algeria
Prior art keywords
substituted
preparation
pharmaceutical compositions
compositions containing
heterobicyclic derivatives
Prior art date
Application number
DZ970150A
Other languages
English (en)
Inventor
Liang Chen Yuhpyng
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=21823717&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DZ2300(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of DZ2300A1 publication Critical patent/DZ2300A1/fr

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
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    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P1/12Antidiarrhoeals
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    • A61P1/14Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • AHUMAN NECESSITIES
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    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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    • A61P25/36Opioid-abuse
    • AHUMAN NECESSITIES
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    • AHUMAN NECESSITIES
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    • A61P5/38Drugs for disorders of the endocrine system of the suprarenal hormones
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    • A61P7/12Antidiuretics, e.g. drugs for diabetes insipidus
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    • A61P9/06Antiarrhythmics
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    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
DZ970150A 1996-08-28 1997-08-27 Dérivés 6,5-hétérobicycliques substitués, procédé pour leur préparation et compositions pharmaceutiques les contenant. DZ2300A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US2503996P 1996-08-28 1996-08-28

Publications (1)

Publication Number Publication Date
DZ2300A1 true DZ2300A1 (fr) 2002-12-25

Family

ID=21823717

Family Applications (1)

Application Number Title Priority Date Filing Date
DZ970150A DZ2300A1 (fr) 1996-08-28 1997-08-27 Dérivés 6,5-hétérobicycliques substitués, procédé pour leur préparation et compositions pharmaceutiques les contenant.

Country Status (36)

Country Link
EP (1) EP0923582B1 (fr)
JP (2) JP3621706B2 (fr)
KR (1) KR20000035934A (fr)
CN (1) CN1227554A (fr)
AP (1) AP762A (fr)
AR (1) AR015103A1 (fr)
AT (1) ATE340176T1 (fr)
AU (1) AU735401B2 (fr)
BG (1) BG103189A (fr)
BR (1) BR9711970A (fr)
CA (1) CA2263566C (fr)
CO (1) CO4600634A1 (fr)
CZ (1) CZ68199A3 (fr)
DE (1) DE69736711T2 (fr)
DZ (1) DZ2300A1 (fr)
EA (1) EA002769B1 (fr)
ES (1) ES2273369T3 (fr)
GT (1) GT199700095A (fr)
HR (1) HRP970454B1 (fr)
HU (1) HUP9903965A3 (fr)
ID (1) ID18249A (fr)
IL (1) IL127566A0 (fr)
IS (1) IS4963A (fr)
MA (1) MA26438A1 (fr)
NO (1) NO313636B1 (fr)
NZ (1) NZ333302A (fr)
OA (1) OA10977A (fr)
PA (1) PA8436201A1 (fr)
PE (1) PE108898A1 (fr)
PL (1) PL332040A1 (fr)
SK (1) SK23399A3 (fr)
TN (1) TNSN97145A1 (fr)
TR (1) TR199900389T2 (fr)
TW (1) TW575573B (fr)
WO (1) WO1998008847A1 (fr)
ZA (1) ZA977687B (fr)

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US6124289A (en) * 1996-07-24 2000-09-26 Dupont Pharmaceuticals Co. Azolo triazines and pyrimidines
US6313124B1 (en) 1997-07-23 2001-11-06 Dupont Pharmaceuticals Company Tetrazine bicyclic compounds
US7094782B1 (en) 1996-07-24 2006-08-22 Bristol-Myers Squibb Company Azolo triazines and pyrimidines
US6060478A (en) * 1996-07-24 2000-05-09 Dupont Pharmaceuticals Azolo triazines and pyrimidines
US6191131B1 (en) 1997-07-23 2001-02-20 Dupont Pharmaceuticals Company Azolo triazines and pyrimidines
EP0970082A2 (fr) 1997-02-18 2000-01-12 Neurocrine Biosciences, Inc. Antagonistes crf biazacycliques
US6211195B1 (en) 1997-04-22 2001-04-03 Neurocrine Biosciences, Inc. CRF antagonistic thiophenopyridines
PL337888A1 (en) 1997-07-03 2000-09-11 Du Pont Pharm Co Imidazoprimidines and imidazopyridines for use in treating neurological disorders
DE69926665T2 (de) * 1998-01-28 2006-06-08 Bristol-Myers Squibb Pharma Co. Azolo-Pyrimidine
US6187777B1 (en) 1998-02-06 2001-02-13 Amgen Inc. Compounds and methods which modulate feeding behavior and related diseases
US6472402B1 (en) 1998-04-02 2002-10-29 Neurogen Corporation Aminoalkyl substituted 5,6,7,8-Tetrahydro-9H-Pyridino [2,3-B]indole derivatives
WO1999051597A1 (fr) 1998-04-02 1999-10-14 Neurogen Corporation Derives de 5,6,7,8-tetrahydro-9h pyrimidino[2,3-b]indole et de 5,6,7,8-tetrahydro-9h-pyrimidino[4,5-b]indole a substitution aminoalkyl: des ligands specifiques du crf1
AU3213699A (en) * 1998-04-03 1999-10-25 Du Pont Pharmaceuticals Company Thiazolo(4,5-d)pyrimidines and pyridines as corticotropin releasing factor (CRF)antagonists
CA2334671A1 (fr) 1998-06-09 1999-12-16 Neurogen Corporation Derives de pyrido[2, 3-b]indolizine et analogues aza associes; ligands crf1 specifiques
US6509338B1 (en) 1998-06-22 2003-01-21 Bristol-Myers Squibb Company Pyrazolo[1,5-A]triazine corticotropin releasing factor antagonists
CA2339188A1 (fr) 1998-08-21 2000-03-02 Dupont Pharmaceuticals Company Isoxazolo¬4,5-d|pyrimidines comme antagonistes du crf
US6531475B1 (en) * 1998-11-12 2003-03-11 Neurocrine Biosciences, Inc. CRF receptor antagonists and methods relating thereto
ES2196898T3 (es) 1998-11-12 2003-12-16 Neurocrine Biosciences Inc Antagonistas de receptores de crf y metodos relacionados.
JP2002529465A (ja) 1998-11-12 2002-09-10 ニューロクライン バイオサイエンシーズ, インコーポレイテッド Crfレセプターアンタゴニストおよびcrfレセプターアンタゴニストに関する方法
EP1149835A4 (fr) * 1999-01-29 2002-08-21 Sumitomo Chemical Co Agents inhibiteurs d'accumulation de graisse
EP1040831A3 (fr) * 1999-04-02 2003-05-02 Pfizer Products Inc. Utilisation d'antagonistes du facteur de libération de la corticotropine pour la prévention de la mort subite
WO2000059907A2 (fr) 1999-04-06 2000-10-12 Du Pont Pharmaceuticals Company Pyrazolotriazines antagonistes de corticoliberine (crf)
WO2000059908A2 (fr) 1999-04-06 2000-10-12 Du Pont Pharmaceuticals Company Pyrazolopyrimidines antagonistes de corticoliberine (crf)
US6982265B1 (en) 1999-05-21 2006-01-03 Bristol Myers Squibb Company Pyrrolotriazine inhibitors of kinases
EP1669071B1 (fr) * 1999-05-21 2009-07-22 Bristol-Myers Squibb Company Pyrrolotriazines comme inhibiteurs des kinases.
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