MA26438A1 - Derives 6,5-heterobicycliques substitues, procede pour leur preparation et compositions pharmaceutiques les contenant. - Google Patents
Derives 6,5-heterobicycliques substitues, procede pour leur preparation et compositions pharmaceutiques les contenant.Info
- Publication number
- MA26438A1 MA26438A1 MA24779A MA24779A MA26438A1 MA 26438 A1 MA26438 A1 MA 26438A1 MA 24779 A MA24779 A MA 24779A MA 24779 A MA24779 A MA 24779A MA 26438 A1 MA26438 A1 MA 26438A1
- Authority
- MA
- Morocco
- Prior art keywords
- substituted
- preparation
- pharmaceutical compositions
- compositions containing
- heterobicyclic derivatives
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/12—Antidiarrhoeals
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
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- A—HUMAN NECESSITIES
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- A61P11/06—Antiasthmatics
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- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
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- A61P15/06—Antiabortive agents; Labour repressants
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- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US2503996P | 1996-08-28 | 1996-08-28 |
Publications (1)
Publication Number | Publication Date |
---|---|
MA26438A1 true MA26438A1 (fr) | 2004-12-20 |
Family
ID=21823717
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MA24779A MA26438A1 (fr) | 1996-08-28 | 1997-08-27 | Derives 6,5-heterobicycliques substitues, procede pour leur preparation et compositions pharmaceutiques les contenant. |
Country Status (36)
Country | Link |
---|---|
EP (1) | EP0923582B1 (fr) |
JP (2) | JP3621706B2 (fr) |
KR (1) | KR20000035934A (fr) |
CN (1) | CN1227554A (fr) |
AP (1) | AP762A (fr) |
AR (1) | AR015103A1 (fr) |
AT (1) | ATE340176T1 (fr) |
AU (1) | AU735401B2 (fr) |
BG (1) | BG103189A (fr) |
BR (1) | BR9711970A (fr) |
CA (1) | CA2263566C (fr) |
CO (1) | CO4600634A1 (fr) |
CZ (1) | CZ68199A3 (fr) |
DE (1) | DE69736711T2 (fr) |
DZ (1) | DZ2300A1 (fr) |
EA (1) | EA002769B1 (fr) |
ES (1) | ES2273369T3 (fr) |
GT (1) | GT199700095A (fr) |
HR (1) | HRP970454B1 (fr) |
HU (1) | HUP9903965A3 (fr) |
ID (1) | ID18249A (fr) |
IL (1) | IL127566A0 (fr) |
IS (1) | IS4963A (fr) |
MA (1) | MA26438A1 (fr) |
NO (1) | NO313636B1 (fr) |
NZ (1) | NZ333302A (fr) |
OA (1) | OA10977A (fr) |
PA (1) | PA8436201A1 (fr) |
PE (1) | PE108898A1 (fr) |
PL (1) | PL332040A1 (fr) |
SK (1) | SK23399A3 (fr) |
TN (1) | TNSN97145A1 (fr) |
TR (1) | TR199900389T2 (fr) |
TW (1) | TW575573B (fr) |
WO (1) | WO1998008847A1 (fr) |
ZA (1) | ZA977687B (fr) |
Families Citing this family (147)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2194756A1 (fr) | 1995-05-12 | 1996-11-14 | Jun Yuan | Derives nouveaux de deazapurine; une nouvelle classe de ligands specifiques de crf1 |
US6313124B1 (en) | 1997-07-23 | 2001-11-06 | Dupont Pharmaceuticals Company | Tetrazine bicyclic compounds |
US6060478A (en) * | 1996-07-24 | 2000-05-09 | Dupont Pharmaceuticals | Azolo triazines and pyrimidines |
US6191131B1 (en) | 1997-07-23 | 2001-02-20 | Dupont Pharmaceuticals Company | Azolo triazines and pyrimidines |
US6124289A (en) * | 1996-07-24 | 2000-09-26 | Dupont Pharmaceuticals Co. | Azolo triazines and pyrimidines |
US7094782B1 (en) | 1996-07-24 | 2006-08-22 | Bristol-Myers Squibb Company | Azolo triazines and pyrimidines |
EP0970082A2 (fr) | 1997-02-18 | 2000-01-12 | Neurocrine Biosciences, Inc. | Antagonistes crf biazacycliques |
JP2002501493A (ja) * | 1997-04-22 | 2002-01-15 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | Crfアンタゴニストのチオフェノピリジン類 |
BR9810508A (pt) * | 1997-07-03 | 2000-09-05 | Du Pont Pharm Co | Composto, composição farmacêutica e método de tratamento de uma desordem |
NZ524842A (en) * | 1998-01-28 | 2003-10-31 | Bristol Myers Squibb Pharma Co | Azolo triazines and pyrimidines |
US6187777B1 (en) | 1998-02-06 | 2001-02-13 | Amgen Inc. | Compounds and methods which modulate feeding behavior and related diseases |
US6472402B1 (en) | 1998-04-02 | 2002-10-29 | Neurogen Corporation | Aminoalkyl substituted 5,6,7,8-Tetrahydro-9H-Pyridino [2,3-B]indole derivatives |
AU3375999A (en) | 1998-04-02 | 1999-10-25 | Neurogen Corporation | Aminoalkyl substituted 5,6,7,8-tetrahydro-9h pyrimidino(2,3-b)indole and 5,6,7,8-tetrahydro-9h-pyrimidino(4,5-b)indole derivatives: crf1 specific ligands |
AU3213699A (en) * | 1998-04-03 | 1999-10-25 | Du Pont Pharmaceuticals Company | Thiazolo(4,5-d)pyrimidines and pyridines as corticotropin releasing factor (CRF)antagonists |
AU4556999A (en) | 1998-06-09 | 1999-12-30 | Neurogen Corporation | Pyrido[2,3-b]indolizine derivatives and aza analogues thereof; crf1 specific ligands |
US6509338B1 (en) | 1998-06-22 | 2003-01-21 | Bristol-Myers Squibb Company | Pyrazolo[1,5-A]triazine corticotropin releasing factor antagonists |
AU5777299A (en) | 1998-08-21 | 2000-03-14 | Du Pont Pharmaceuticals Company | Isoxazolo(4,5-d)pyrimidines as CRF antagonists |
US6531475B1 (en) * | 1998-11-12 | 2003-03-11 | Neurocrine Biosciences, Inc. | CRF receptor antagonists and methods relating thereto |
BR9915129A (pt) * | 1998-11-12 | 2001-08-07 | Neurocrine Biosciences Inc | Antagonistas do receptor de crf e processos relacionados aos mesmos |
DK1129091T3 (da) | 1998-11-12 | 2002-11-04 | Neurocrine Biosciences Inc | Antagonister for CRF-receptorer og fremgangsmåder med relation dertil |
CA2359041A1 (fr) * | 1999-01-29 | 2000-08-03 | Sumitomo Chemical Co., Ltd. | Agents inhibiteurs d'accumulation de graisse |
EP1040831A3 (fr) * | 1999-04-02 | 2003-05-02 | Pfizer Products Inc. | Utilisation d'antagonistes du facteur de libération de la corticotropine pour la prévention de la mort subite |
WO2000059908A2 (fr) | 1999-04-06 | 2000-10-12 | Du Pont Pharmaceuticals Company | Pyrazolopyrimidines antagonistes de corticoliberine (crf) |
WO2000059907A2 (fr) | 1999-04-06 | 2000-10-12 | Du Pont Pharmaceuticals Company | Pyrazolotriazines antagonistes de corticoliberine (crf) |
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2004
- 2004-09-21 JP JP2004273978A patent/JP2005047930A/ja not_active Withdrawn
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