SG11201408052WA - IMIDAZO[1,2-b]PYRIDAZINE DERIVATIVES AS KINASE INHIBITORS - Google Patents

IMIDAZO[1,2-b]PYRIDAZINE DERIVATIVES AS KINASE INHIBITORS

Info

Publication number
SG11201408052WA
SG11201408052WA SG11201408052WA SG11201408052WA SG11201408052WA SG 11201408052W A SG11201408052W A SG 11201408052WA SG 11201408052W A SG11201408052W A SG 11201408052WA SG 11201408052W A SG11201408052W A SG 11201408052WA SG 11201408052W A SG11201408052W A SG 11201408052WA
Authority
SG
Singapore
Prior art keywords
imidazo
compound
kinase inhibitors
pyridazine derivatives
acceptable salt
Prior art date
Application number
SG11201408052WA
Other languages
English (en)
Inventor
Yasuyuki Takeda
Kenji Yoshikawa
Yoshiko Kagoshima
Yuko Yamamoto
Ryoichi Tanaka
Yuichi Tominaga
Masaki Kiga
Yoshito Hamada
Original Assignee
Daiichi Sankyo Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Daiichi Sankyo Co Ltd filed Critical Daiichi Sankyo Co Ltd
Publication of SG11201408052WA publication Critical patent/SG11201408052WA/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50—Pyridazines; Hydrogenated pyridazines
    • A61K31/5025—Pyridazines; Hydrogenated pyridazines ortho- or peri-condensed with heterocyclic ring systems
SG11201408052WA 2012-06-04 2013-06-03 IMIDAZO[1,2-b]PYRIDAZINE DERIVATIVES AS KINASE INHIBITORS SG11201408052WA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2012127079 2012-06-04
PCT/JP2013/065328 WO2013183578A1 (ja) 2012-06-04 2013-06-03 キナーゼ阻害剤としてのイミダゾ[１，２－ｂ]ピリダジン誘導体

Publications (1)

Publication Number Publication Date
SG11201408052WA true SG11201408052WA (en) 2015-01-29

Family

ID=49711970

Family Applications (1)

Application Number Title Priority Date Filing Date
SG11201408052WA SG11201408052WA (en) 2012-06-04 2013-06-03 IMIDAZO[1,2-b]PYRIDAZINE DERIVATIVES AS KINASE INHIBITORS

Country Status (32)

Country Link
US (2) US9187489B2 (ru)
EP (1) EP2857404B1 (ru)
JP (1) JP5814467B2 (ru)
KR (1) KR101781255B1 (ru)
CN (1) CN104520300B (ru)
AU (1) AU2013272701B2 (ru)
BR (1) BR112014029851B1 (ru)
CA (1) CA2874819C (ru)
CO (1) CO7160119A2 (ru)
CY (1) CY1119607T1 (ru)
DK (1) DK2857404T3 (ru)
ES (1) ES2648228T3 (ru)
HK (1) HK1207374A1 (ru)
HR (1) HRP20171724T1 (ru)
HU (1) HUE037221T2 (ru)
IL (1) IL236075A (ru)
IN (1) IN2014MN02497A (ru)
LT (1) LT2857404T (ru)
MX (1) MX357021B (ru)
MY (1) MY170326A (ru)
NO (1) NO2857404T3 (ru)
NZ (1) NZ702574A (ru)
PH (1) PH12014502721A1 (ru)
PL (1) PL2857404T3 (ru)
PT (1) PT2857404T (ru)
RS (1) RS56625B1 (ru)
RU (1) RU2635917C2 (ru)
SG (1) SG11201408052WA (ru)
SI (1) SI2857404T1 (ru)
TW (1) TWI585088B (ru)
WO (1) WO2013183578A1 (ru)
ZA (1) ZA201408843B (ru)

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Also Published As

Publication number Publication date
KR101781255B1 (ko) 2017-09-22
NO2857404T3 (ru) 2018-01-20
IL236075A (en) 2017-10-31
RU2014153627A (ru) 2016-08-10
IN2014MN02497A (ru) 2015-07-17
PL2857404T3 (pl) 2018-04-30
HUE037221T2 (hu) 2018-08-28
WO2013183578A1 (ja) 2013-12-12
MY170326A (en) 2019-07-17
PT2857404T (pt) 2017-11-23
IL236075A0 (en) 2015-02-01
HK1207374A1 (en) 2016-01-29
NZ702574A (en) 2016-07-29
HRP20171724T1 (hr) 2018-01-12
US20160046639A1 (en) 2016-02-18
EP2857404A1 (en) 2015-04-08
MX357021B (es) 2018-06-25
EP2857404B1 (en) 2017-08-23
TWI585088B (zh) 2017-06-01
EP2857404A4 (en) 2016-01-20
AU2013272701A2 (en) 2015-01-22
CA2874819A1 (en) 2013-12-12
JP5814467B2 (ja) 2015-11-17
ZA201408843B (en) 2016-01-27
MX2014014803A (es) 2015-02-12
BR112014029851B1 (pt) 2023-01-03
AU2013272701A1 (en) 2015-01-15
BR112014029851A2 (pt) 2017-06-27
AU2013272701B2 (en) 2017-12-21
DK2857404T3 (en) 2017-12-04
US9187489B2 (en) 2015-11-17
TW201400486A (zh) 2014-01-01
CN104520300A (zh) 2015-04-15
RS56625B1 (sr) 2018-03-30
US9751887B2 (en) 2017-09-05
SI2857404T1 (sl) 2017-11-30
CA2874819C (en) 2017-06-20
KR20150014942A (ko) 2015-02-09
CY1119607T1 (el) 2018-04-04
CN104520300B (zh) 2016-12-21
PH12014502721B1 (en) 2015-02-02
ES2648228T3 (es) 2017-12-29
JPWO2013183578A1 (ja) 2016-01-28
US20150051190A1 (en) 2015-02-19
PH12014502721A1 (en) 2015-02-02
RU2635917C2 (ru) 2017-11-17
CO7160119A2 (es) 2015-01-15
LT2857404T (lt) 2017-11-10

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