MX2010009207A - Compuestos y composiciones heterociclicos como inhibidores de c-kit y pdgfr cinasa. - Google Patents

Compuestos y composiciones heterociclicos como inhibidores de c-kit y pdgfr cinasa.

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Publication number
MX2010009207A
MX2010009207A MX2010009207A MX2010009207A MX2010009207A MX 2010009207 A MX2010009207 A MX 2010009207A MX 2010009207 A MX2010009207 A MX 2010009207A MX 2010009207 A MX2010009207 A MX 2010009207A MX 2010009207 A MX2010009207 A MX 2010009207A
Authority
MX
Mexico
Prior art keywords
kit
compositions
kinase inhibitors
heterocyclic compounds
pdgfr kinase
Prior art date
Application number
MX2010009207A
Other languages
English (en)
Inventor
Molteni Valentina
Nabakka Juliet
Li Xiaolin
Liu Xiaodong
Chianelli Donatella
Yeh Vince
Original Assignee
Irm Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40577860&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX2010009207(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Irm Llc filed Critical Irm Llc
Publication of MX2010009207A publication Critical patent/MX2010009207A/es

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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Abstract

La presente invención proporciona una nueva clase de compuestos de la fórmula I: (I) composiciones farmacéuticas que comprenden tales compuestos para el tratamiento o prevención de enfermedades o trastornos asociados con la actividad anormal o desregulada de cinasas, particularmente enfermedades o trastornos que involucran la activación anormal de las c-kit, PDGFRa y PDGFRß cinasas.
MX2010009207A 2008-02-22 2009-02-20 Compuestos y composiciones heterociclicos como inhibidores de c-kit y pdgfr cinasa. MX2010009207A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US3091208P 2008-02-22 2008-02-22
PCT/US2009/034778 WO2009105712A1 (en) 2008-02-22 2009-02-20 Heterocyclic compounds and compositions as c-kit and pdgfr kinase inhibitors

Publications (1)

Publication Number Publication Date
MX2010009207A true MX2010009207A (es) 2011-03-03

Family

ID=40577860

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2010009207A MX2010009207A (es) 2008-02-22 2009-02-20 Compuestos y composiciones heterociclicos como inhibidores de c-kit y pdgfr cinasa.

Country Status (17)

Country Link
US (1) US8278452B2 (es)
EP (1) EP2252612B1 (es)
JP (1) JP5230755B2 (es)
KR (1) KR101216323B1 (es)
CN (1) CN102083828B (es)
AR (1) AR070469A1 (es)
AT (1) ATE551342T1 (es)
AU (1) AU2009217356B2 (es)
BR (1) BRPI0908849A2 (es)
CA (1) CA2714700C (es)
CL (1) CL2009000400A1 (es)
EA (1) EA018551B1 (es)
ES (1) ES2383331T3 (es)
MX (1) MX2010009207A (es)
PE (1) PE20091492A1 (es)
TW (1) TW200940538A (es)
WO (1) WO2009105712A1 (es)

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