MX2009012079A - Compuestos heterociclicos condensados como inhibidores de proteina cinasas. - Google Patents
Compuestos heterociclicos condensados como inhibidores de proteina cinasas.Info
- Publication number
- MX2009012079A MX2009012079A MX2009012079A MX2009012079A MX2009012079A MX 2009012079 A MX2009012079 A MX 2009012079A MX 2009012079 A MX2009012079 A MX 2009012079A MX 2009012079 A MX2009012079 A MX 2009012079A MX 2009012079 A MX2009012079 A MX 2009012079A
- Authority
- MX
- Mexico
- Prior art keywords
- inhibitors
- heterocyclic compounds
- protein kinases
- condensed heterocyclic
- compounds
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Abstract
Se describen compuestos que tienen la Fórmula (I) que inhiben las Aurora-cinasas, composiciones que contienen los compuestos y métodos para tratar enfermedades utilizando los compuestos.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US91683807P | 2007-05-09 | 2007-05-09 | |
US91684607P | 2007-05-09 | 2007-05-09 | |
PCT/US2008/063197 WO2008141145A1 (en) | 2007-05-09 | 2008-05-09 | Condensed heterocyclic compounds as inhibitors of protein kinases |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2009012079A true MX2009012079A (es) | 2009-11-19 |
Family
ID=39650562
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2009012079A MX2009012079A (es) | 2007-05-09 | 2008-05-09 | Compuestos heterociclicos condensados como inhibidores de proteina cinasas. |
Country Status (8)
Country | Link |
---|---|
EP (1) | EP2150553B1 (es) |
JP (1) | JP5412424B2 (es) |
CN (1) | CN101730700A (es) |
AT (1) | ATE527264T1 (es) |
CA (1) | CA2685351A1 (es) |
ES (1) | ES2372559T3 (es) |
MX (1) | MX2009012079A (es) |
WO (1) | WO2008141145A1 (es) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8624027B2 (en) * | 2005-05-12 | 2014-01-07 | Abbvie Inc. | Combination therapy for treating cancer and diagnostic assays for use therein |
US8124759B2 (en) | 2007-05-09 | 2012-02-28 | Abbott Laboratories | Inhibitors of protein kinases |
CN102532042A (zh) * | 2010-12-30 | 2012-07-04 | 上海医药工业研究院 | 一种芳基脲类化合物、其中间体及其应用 |
BR112015006828A8 (pt) | 2012-09-26 | 2019-09-17 | Univ California | composto, ou um sal farmaceuticamente aceitável do mesmo; composição farmacêutica; uso do composto; e método para modular a atividade de uma proteína ire1 |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP4916883B2 (ja) * | 2003-10-15 | 2012-04-18 | オーエスアイ・ファーマスーティカルズ・インコーポレーテッド | イミダゾピラジンチロシンキナーゼ阻害剤 |
WO2005097800A1 (en) * | 2004-04-02 | 2005-10-20 | Osi Pharmaceuticals, Inc. | 6,6-bicyclic ring substituted heterobicyclic protein kinase inhibitors |
ATE533770T1 (de) * | 2005-10-06 | 2011-12-15 | Schering Corp | Pyrazolopyrimidine als proteinkinaseinhibitoren |
JP5335432B2 (ja) * | 2005-11-17 | 2013-11-06 | オーエスアイ・フアーマシユーテイカルズ・エル・エル・シー | 縮合2環系mTOR阻害剤 |
AR057960A1 (es) * | 2005-12-02 | 2007-12-26 | Osi Pharm Inc | Inhibidores de proteina quinasa biciclicos |
US7659274B2 (en) * | 2006-01-25 | 2010-02-09 | Osi Pharmaceuticals, Inc. | Unsaturated mTOR inhibitors |
JP5372737B2 (ja) * | 2006-03-13 | 2013-12-18 | オーエスアイ・フアーマシユーテイカルズ・エル・エル・シー | Egfrキナーゼ阻害剤およびegfrキナーゼ阻害剤の効果に対し腫瘍細胞を感作する薬剤を用いる併用治療 |
-
2008
- 2008-05-09 MX MX2009012079A patent/MX2009012079A/es active IP Right Grant
- 2008-05-09 WO PCT/US2008/063197 patent/WO2008141145A1/en active Application Filing
- 2008-05-09 AT AT08780617T patent/ATE527264T1/de not_active IP Right Cessation
- 2008-05-09 EP EP08780617A patent/EP2150553B1/en active Active
- 2008-05-09 JP JP2010507687A patent/JP5412424B2/ja not_active Expired - Fee Related
- 2008-05-09 ES ES08780617T patent/ES2372559T3/es active Active
- 2008-05-09 CN CN200880023583A patent/CN101730700A/zh active Pending
- 2008-05-09 CA CA002685351A patent/CA2685351A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
EP2150553B1 (en) | 2011-10-05 |
WO2008141145A1 (en) | 2008-11-20 |
JP2010526833A (ja) | 2010-08-05 |
JP5412424B2 (ja) | 2014-02-12 |
CN101730700A (zh) | 2010-06-09 |
CA2685351A1 (en) | 2008-11-20 |
ES2372559T3 (es) | 2012-01-23 |
EP2150553A1 (en) | 2010-02-10 |
ATE527264T1 (de) | 2011-10-15 |
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Legal Events
Date | Code | Title | Description |
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HH | Correction or change in general | ||
FG | Grant or registration | ||
GB | Transfer or rights |