ECSP14013217A - 4-imidazopiridazin-1-il-benzamidas y 4-imidazotriazin-1-il-benzamidas como inhibidores de btk. - Google Patents

4-imidazopiridazin-1-il-benzamidas y 4-imidazotriazin-1-il-benzamidas como inhibidores de btk.

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Publication number
ECSP14013217A
ECSP14013217A ECSP14013217A ECSP14013217A EC SP14013217 A ECSP14013217 A EC SP14013217A EC SP14013217 A ECSP14013217 A EC SP14013217A EC SP14013217 A ECSP14013217 A EC SP14013217A
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EC
Ecuador
Prior art keywords
benzamidas
imidazotriazin
imidazopiridazin
formula
btk inhibitors
Prior art date
Application number
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English (en)
Inventor
Tjeerd A Barf
Christiaan Gerardus Johannes Maria Jans
De Adrianus Petrus Antonius Man
Arthur A Oubrie
Hans C A Raaijmakers
Johannes Bernardus Maria Rewinkel
Jan-Gerard Sterrenburg
Jacobus C H M Wijkmans
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Msd Oss Bv
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Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=47557677&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ECSP14013217(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Msd Oss Bv filed Critical Msd Oss Bv
Publication of ECSP14013217A publication Critical patent/ECSP14013217A/es

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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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Abstract

La presente invención se refiere a compuestos de anillos de piridina fusionados de 5-6 miembros según la fórmula I Fórmula Io una sal farmacéuticamente aceptable de los mismos o a composiciones farmacéuticas que comprenden estos compuestos y a su uso en terapia. En particular, la presente invención se refiere al uso de compuestos de anillos de piridina fusionados de 5-6 miembros según la fórmula I en el tratamiento de trastornos mediados por tirosina cinasa de Bruton (Btk).
ECSP14013217 2011-07-19 2014-02-19 4-imidazopiridazin-1-il-benzamidas y 4-imidazotriazin-1-il-benzamidas como inhibidores de btk. ECSP14013217A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201161509397P 2011-07-19 2011-07-19
EP11174578 2011-07-19

Publications (1)

Publication Number Publication Date
ECSP14013217A true ECSP14013217A (es) 2015-03-31

Family

ID=47557677

Family Applications (1)

Application Number Title Priority Date Filing Date
ECSP14013217 ECSP14013217A (es) 2011-07-19 2014-02-19 4-imidazopiridazin-1-il-benzamidas y 4-imidazotriazin-1-il-benzamidas como inhibidores de btk.

Country Status (35)

Country Link
US (7) US9290504B2 (es)
EP (4) EP4249076A3 (es)
JP (6) JP5826931B2 (es)
KR (2) KR101802689B1 (es)
CN (2) CN106243113B (es)
AU (4) AU2012285987C1 (es)
BR (1) BR112014001255B1 (es)
CA (1) CA2841886C (es)
CL (1) CL2014000130A1 (es)
CO (1) CO6940411A2 (es)
CR (1) CR20140030A (es)
DK (2) DK3689878T3 (es)
DO (1) DOP2014000008A (es)
EA (2) EA037644B1 (es)
EC (1) ECSP14013217A (es)
ES (3) ES2708224T3 (es)
GT (1) GT201400009A (es)
HR (2) HRP20212021T1 (es)
HU (3) HUE056249T2 (es)
IL (3) IL230511B (es)
IN (1) IN2014CN00408A (es)
LT (1) LT2734522T (es)
MA (1) MA35348B1 (es)
MX (1) MX342983B (es)
MY (1) MY192354A (es)
PE (1) PE20141681A1 (es)
PH (1) PH12017500166A1 (es)
PL (2) PL3689878T3 (es)
PT (1) PT3689878T (es)
RS (2) RS58177B1 (es)
SG (1) SG10201605913VA (es)
SI (2) SI2734522T1 (es)
TN (1) TN2014000027A1 (es)
UA (1) UA115312C2 (es)
WO (1) WO2013010868A1 (es)

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