DE69530989D1 - Neue pyrimidinderivate und verfahren zu ihrer herstellung - Google Patents

Neue pyrimidinderivate und verfahren zu ihrer herstellung

Info

Publication number
DE69530989D1
DE69530989D1 DE69530989T DE69530989T DE69530989D1 DE 69530989 D1 DE69530989 D1 DE 69530989D1 DE 69530989 T DE69530989 T DE 69530989T DE 69530989 T DE69530989 T DE 69530989T DE 69530989 D1 DE69530989 D1 DE 69530989D1
Authority
DE
Germany
Prior art keywords
new
production
pyrimid
derivatives
pyrimid derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE69530989T
Other languages
English (en)
Other versions
DE69530989T2 (de
Inventor
Wook Lee
Seok Chae
Seop Kim
Kyu Kim
Sung Lim
Kyu Shon
Shik Choi
Ho Lee
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Yuhan Corp
Original Assignee
Yuhan Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from KR1019940019998A external-priority patent/KR0157076B1/ko
Priority claimed from KR1019940019997A external-priority patent/KR0157075B1/ko
Application filed by Yuhan Corp filed Critical Yuhan Corp
Publication of DE69530989D1 publication Critical patent/DE69530989D1/de
Application granted granted Critical
Publication of DE69530989T2 publication Critical patent/DE69530989T2/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
DE69530989T 1994-08-13 1995-08-10 Neue pyrimidinderivate und verfahren zu ihrer herstellung Expired - Lifetime DE69530989T2 (de)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
KR1999794 1994-08-13
KR1019940019998A KR0157076B1 (ko) 1994-08-13 1994-08-13 신규의 피리미딘 유도체 및 그의 제조방법
KR1999894 1994-08-13
KR1019940019997A KR0157075B1 (ko) 1994-08-13 1994-08-13 신규의 피리미딘 유도체 및 그의 제조방법
PCT/KR1995/000105 WO1996005177A1 (en) 1994-08-13 1995-08-10 Novel pyrimidine derivatives and processes for the preparation thereof

Publications (2)

Publication Number Publication Date
DE69530989D1 true DE69530989D1 (de) 2003-07-10
DE69530989T2 DE69530989T2 (de) 2004-05-19

Family

ID=26630534

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69530989T Expired - Lifetime DE69530989T2 (de) 1994-08-13 1995-08-10 Neue pyrimidinderivate und verfahren zu ihrer herstellung

Country Status (11)

Country Link
US (1) US5750531A (de)
EP (1) EP0775120B1 (de)
JP (1) JP2896532B2 (de)
CN (1) CN1102144C (de)
AU (1) AU688087B2 (de)
CA (1) CA2197298C (de)
DE (1) DE69530989T2 (de)
ES (1) ES2201112T3 (de)
HK (1) HK1001618A1 (de)
RU (1) RU2129549C1 (de)
WO (1) WO1996005177A1 (de)

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* Cited by examiner, † Cited by third party
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US7365047B1 (en) 1999-09-28 2008-04-29 The Regents Of The University Of California Use of pentagastrin to inhibit gastric acid secretion or as a diuretic
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CN105669642B (zh) 2014-11-19 2020-06-09 江苏天士力帝益药业有限公司 一种盐酸洛氟普啶的制备方法
CN107405359B (zh) 2015-11-25 2021-04-20 艾克萨姆治疗公司 包含美洛昔康的药物组合物
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Family Cites Families (5)

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DE9190155U1 (de) * 1990-11-06 1993-10-07 Pfizer Chinazolinderivate zur Steigerung der Antitumoraktivität
JPH04305526A (ja) * 1991-03-28 1992-10-28 Morishita Roussel Kk 薬剤組成物
JPH05262747A (ja) * 1991-10-17 1993-10-12 Morishita Roussel Kk 潰瘍性大腸炎治療剤
KR0144833B1 (ko) * 1992-12-28 1998-07-15 김태훈 신규의 퀴나졸린 유도체 및 그의 제조방법
JPH0753527A (ja) * 1993-08-09 1995-02-28 Toa Boshoku Kk 置換ピリミジン誘導体、その製造方法、及び鎮痛・抗炎症剤

Also Published As

Publication number Publication date
EP0775120B1 (de) 2003-06-04
HK1001618A1 (en) 1998-07-03
CA2197298A1 (en) 1996-02-22
CN1155281A (zh) 1997-07-23
JP2896532B2 (ja) 1999-05-31
EP0775120A1 (de) 1997-05-28
CN1102144C (zh) 2003-02-26
RU2129549C1 (ru) 1999-04-27
US5750531A (en) 1998-05-12
AU688087B2 (en) 1998-03-05
JPH09509188A (ja) 1997-09-16
CA2197298C (en) 1999-10-19
AU3122595A (en) 1996-03-07
WO1996005177A1 (en) 1996-02-22
DE69530989T2 (de) 2004-05-19
ES2201112T3 (es) 2004-03-16

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