DE602007011773D1 - Substituierte pyrazolopyrimidine, ein verfahren zu ihrer herstellung und ihre verwendung als medizin - Google Patents

Substituierte pyrazolopyrimidine, ein verfahren zu ihrer herstellung und ihre verwendung als medizin

Info

Publication number
DE602007011773D1
DE602007011773D1 DE602007011773T DE602007011773T DE602007011773D1 DE 602007011773 D1 DE602007011773 D1 DE 602007011773D1 DE 602007011773 T DE602007011773 T DE 602007011773T DE 602007011773 T DE602007011773 T DE 602007011773T DE 602007011773 D1 DE602007011773 D1 DE 602007011773D1
Authority
DE
Germany
Prior art keywords
medicine
preparation
substituted pyrazolopyrimidines
pyrazolopyrimidines
substituted
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
DE602007011773T
Other languages
English (en)
Inventor
Wojciech Danysz
Andrzej Dekundy
Mirko Hechenberger
Markus Henrich
Claudia Jatzke
Jens Nagel
Christopher Graham Raphael Parsons
Tanja Weil
Juris Fotins
Aleksandra Gutcaits
Ivars Kalvinsh
Ronalds Zemribo
Valerjans Kauss
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merz Pharma GmbH and Co KGaA
Original Assignee
Merz Pharma GmbH and Co KGaA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merz Pharma GmbH and Co KGaA filed Critical Merz Pharma GmbH and Co KGaA
Publication of DE602007011773D1 publication Critical patent/DE602007011773D1/de
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
DE602007011773T 2006-08-04 2007-08-03 Substituierte pyrazolopyrimidine, ein verfahren zu ihrer herstellung und ihre verwendung als medizin Active DE602007011773D1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US83582006P 2006-08-04 2006-08-04
US87754406P 2006-12-28 2006-12-28
PCT/EP2007/058060 WO2008015269A1 (en) 2006-08-04 2007-08-03 Substituted pyrazolopyrimidines, a process for their preparation and their use as medicine

Publications (1)

Publication Number Publication Date
DE602007011773D1 true DE602007011773D1 (de) 2011-02-17

Family

ID=38710494

Family Applications (2)

Application Number Title Priority Date Filing Date
DE602007011773T Active DE602007011773D1 (de) 2006-08-04 2007-08-03 Substituierte pyrazolopyrimidine, ein verfahren zu ihrer herstellung und ihre verwendung als medizin
DE602007010640T Active DE602007010640D1 (de) 2006-08-04 2007-08-03 Pyrazolopyrimidine, ein verfahren zu ihrer herstellung und ihre verwendung als medizin

Family Applications After (1)

Application Number Title Priority Date Filing Date
DE602007010640T Active DE602007010640D1 (de) 2006-08-04 2007-08-03 Pyrazolopyrimidine, ein verfahren zu ihrer herstellung und ihre verwendung als medizin

Country Status (21)

Country Link
US (4) US20080032998A1 (de)
EP (3) EP2054416B8 (de)
JP (2) JP2010500288A (de)
KR (1) KR20090047450A (de)
AR (3) AR062210A1 (de)
AT (2) ATE488520T1 (de)
AU (2) AU2007280428B2 (de)
BR (2) BRPI0714766A2 (de)
CA (2) CA2659871A1 (de)
CY (1) CY1112003T1 (de)
DE (2) DE602007011773D1 (de)
DK (1) DK2054416T3 (de)
HR (1) HRP20110128T1 (de)
IL (2) IL196007A0 (de)
MX (2) MX2009000919A (de)
PL (1) PL2054416T3 (de)
PT (1) PT2054416E (de)
RU (2) RU2009107688A (de)
TW (3) TW200823215A (de)
WO (3) WO2008015270A1 (de)
ZA (1) ZA200810605B (de)

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RU2496494C2 (ru) * 2008-06-30 2013-10-27 Новартис Аг КОМБИНАЦИИ, СОДЕРЖАЩИЕ МОДУЛЯТОРЫ mGluR, ДЛЯ ЛЕЧЕНИЯ БОЛЕЗНИ ПАРКИНСОНА
KR20120098745A (ko) 2009-11-25 2012-09-05 메르츠 파마 게엠베하 운트 코. 카가아 치환된 피라졸로피리미딘의 결정질 형태
EP2648723A4 (de) 2010-12-08 2014-04-02 Univ Vanderbilt Bicyclische pyrazolverbindungen als allosterische mglur5-rezeptormodulatoren
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EP2970297A1 (de) 2013-03-14 2016-01-20 Bristol-Myers Squibb Company Hemmer der neubildung menschlicher immundefektviren
US9975879B2 (en) 2013-06-04 2018-05-22 Temple University Of The Commonwealth System Of Higher Education Beta lactams as modulators of glutamate uptake and methods for use thereof
EP3065724A4 (de) 2013-11-05 2017-05-03 Temple University Of The Commonwealth System Of Higher Education Polykationische amphiphile als antimikrobiotika
US10398142B2 (en) 2013-11-05 2019-09-03 Temple University Of The Commonwealth System Of Higher Education Polycationic amphiphiles as antimicrobial agents
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