BRPI0011674B8 - cristal de (r)-2-[[[3-metil-4-(2,2,2-trifluoroetóxi)-2-piridinil]metil] sulfinil]-1h-benzimidazol, composição farmacêutica, e, uso do referido cristal - Google Patents
cristal de (r)-2-[[[3-metil-4-(2,2,2-trifluoroetóxi)-2-piridinil]metil] sulfinil]-1h-benzimidazol, composição farmacêutica, e, uso do referido cristalInfo
- Publication number
- BRPI0011674B8 BRPI0011674B8 BRPI0011674A BR0011674A BRPI0011674B8 BR PI0011674 B8 BRPI0011674 B8 BR PI0011674B8 BR PI0011674 A BRPI0011674 A BR PI0011674A BR 0011674 A BR0011674 A BR 0011674A BR PI0011674 B8 BRPI0011674 B8 BR PI0011674B8
- Authority
- BR
- Brazil
- Prior art keywords
- crystal
- methyl
- trifluoroethoxy
- sulfinyl
- pyridinyl
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
Abstract
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP17150999 | 1999-06-17 | ||
PCT/JP2000/003880 WO2000078745A2 (en) | 1999-06-17 | 2000-06-15 | Crystalline form of (r)-2-[[[3-methyl- 4- (2,2,2,- trifluoroethoxy) -2- pyridinyl] methyl] sulfinyl] -1h-benzimidazole |
Publications (3)
Publication Number | Publication Date |
---|---|
BR0011674A BR0011674A (pt) | 2002-03-19 |
BRPI0011674B1 BRPI0011674B1 (pt) | 2017-05-30 |
BRPI0011674B8 true BRPI0011674B8 (pt) | 2021-05-25 |
Family
ID=15924444
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0011674A BRPI0011674B8 (pt) | 1999-06-17 | 2000-06-15 | cristal de (r)-2-[[[3-metil-4-(2,2,2-trifluoroetóxi)-2-piridinil]metil] sulfinil]-1h-benzimidazol, composição farmacêutica, e, uso do referido cristal |
Country Status (27)
Country | Link |
---|---|
US (11) | US6462058B1 (pt) |
EP (3) | EP2343289A1 (pt) |
KR (3) | KR100514204B1 (pt) |
CN (1) | CN1150186C (pt) |
AR (5) | AR031069A1 (pt) |
AT (1) | ATE391126T1 (pt) |
AU (1) | AU778820B2 (pt) |
BE (1) | BE2014C017I2 (pt) |
BR (1) | BRPI0011674B8 (pt) |
CA (1) | CA2375201C (pt) |
CY (2) | CY1110384T1 (pt) |
DE (1) | DE60038481T2 (pt) |
DK (2) | DK1129088T3 (pt) |
ES (2) | ES2300265T3 (pt) |
HK (2) | HK1038227A1 (pt) |
HU (1) | HU229067B1 (pt) |
IL (2) | IL145996A0 (pt) |
MX (1) | MXPA01012642A (pt) |
MY (1) | MY125399A (pt) |
NO (1) | NO321168B1 (pt) |
NZ (1) | NZ515702A (pt) |
PL (1) | PL201068B1 (pt) |
PT (2) | PT1977751E (pt) |
SI (1) | SI1129088T1 (pt) |
TW (2) | TWI289557B (pt) |
WO (2) | WO2004083200A1 (pt) |
ZA (1) | ZA200108331B (pt) |
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