SG10201401061XA - Pyridopyrazine Derivatives And Use Thereof As Modulators Of The Signal Transduction Paths - Google Patents

Pyridopyrazine Derivatives And Use Thereof As Modulators Of The Signal Transduction Paths

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Publication number
SG10201401061XA
SG10201401061XA SG10201401061XA SG10201401061XA SG10201401061XA SG 10201401061X A SG10201401061X A SG 10201401061XA SG 10201401061X A SG10201401061X A SG 10201401061XA SG 10201401061X A SG10201401061X A SG 10201401061XA SG 10201401061X A SG10201401061X A SG 10201401061XA
Authority
SG
Singapore
Prior art keywords
modulators
signal transduction
transduction paths
pyridopyrazine derivatives
pyridopyrazine
Prior art date
Application number
SG10201401061XA
Other languages
English (en)
Inventor
Irene Seipelt
Eckhard Claus
Eckhard Günther
Tilmann Schuster
Michael Czech
Emmanuel Polymeropoulos
Original Assignee
Terna Zentaris Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Terna Zentaris Gmbh filed Critical Terna Zentaris Gmbh
Publication of SG10201401061XA publication Critical patent/SG10201401061XA/en

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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/02—Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
SG10201401061XA 2005-11-11 2006-11-10 Pyridopyrazine Derivatives And Use Thereof As Modulators Of The Signal Transduction Paths SG10201401061XA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US73570705P 2005-11-11 2005-11-11
EP05024692A EP1790342A1 (de) 2005-11-11 2005-11-11 Pyridopyrazin-Derivate und deren Verwendung als Modulatoren der Signaltransduktionswege

Publications (1)

Publication Number Publication Date
SG10201401061XA true SG10201401061XA (en) 2014-07-30

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Family Applications (1)

Application Number Title Priority Date Filing Date
SG10201401061XA SG10201401061XA (en) 2005-11-11 2006-11-10 Pyridopyrazine Derivatives And Use Thereof As Modulators Of The Signal Transduction Paths

Country Status (21)

Country Link
US (1) US8937068B2 (zh)
EP (2) EP1790342A1 (zh)
JP (1) JP5448450B2 (zh)
KR (1) KR101473662B1 (zh)
CN (1) CN101330918B (zh)
AR (1) AR056216A1 (zh)
AU (1) AU2006334721B2 (zh)
BR (1) BRPI0618451A2 (zh)
CA (1) CA2628186A1 (zh)
ES (1) ES2543962T3 (zh)
HK (1) HK1125823A1 (zh)
IL (1) IL191160A (zh)
NO (1) NO20082509L (zh)
NZ (1) NZ595879A (zh)
PL (1) PL1962854T3 (zh)
RU (1) RU2487713C2 (zh)
SG (1) SG10201401061XA (zh)
TW (1) TWI423973B (zh)
UA (1) UA95464C2 (zh)
WO (1) WO2007079999A2 (zh)
ZA (1) ZA200803867B (zh)

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UA95464C2 (en) 2011-08-10
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WO2007079999A2 (de) 2007-07-19
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EP1790342A1 (de) 2007-05-30
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US20070123494A1 (en) 2007-05-31
AU2006334721A1 (en) 2007-07-19
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