MXPA05006123A - Analogos de quinazolin-4-ilamina 2-sustituida como moduladores de receptores de capsaicina. - Google Patents

Analogos de quinazolin-4-ilamina 2-sustituida como moduladores de receptores de capsaicina.

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Publication number
MXPA05006123A
MXPA05006123A MXPA05006123A MXPA05006123A MXPA05006123A MX PA05006123 A MXPA05006123 A MX PA05006123A MX PA05006123 A MXPA05006123 A MX PA05006123A MX PA05006123 A MXPA05006123 A MX PA05006123A MX PA05006123 A MXPA05006123 A MX PA05006123A
Authority
MX
Mexico
Prior art keywords
receptor modulators
capsaicin receptor
substituted quinazolin
ylamine analogues
ligands
Prior art date
Application number
MXPA05006123A
Other languages
English (en)
Inventor
Delombaert Stephane
Original Assignee
Neurogen Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Neurogen Corp filed Critical Neurogen Corp
Publication of MXPA05006123A publication Critical patent/MXPA05006123A/es

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    • C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings

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  • Chemical & Material Sciences (AREA)
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  • Pain & Pain Management (AREA)
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  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Virology (AREA)
  • Otolaryngology (AREA)
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  • Pregnancy & Childbirth (AREA)
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  • Ophthalmology & Optometry (AREA)
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Abstract

Se proporcionan ciertos analogos de quinazolin-4-ilamina 2-sustituida. Estos compuestos son ligandos que se pueden utilizar in vitro o in vivo, para modular la actividad de receptores especificos y son particularmente utiles en el tratamiento de condiciones asociadas con la activacion de receptores patologicos en humanos, animales domesticos de compania y ganado. Ser proporcionan composiciones farmaceuticas y metodos para utilizarlas en el tratamiento de estos trastornos, como son los metodos para utilizar estos ligandos para estudios de localizacion de receptores.
MXPA05006123A 2002-12-13 2003-12-12 Analogos de quinazolin-4-ilamina 2-sustituida como moduladores de receptores de capsaicina. MXPA05006123A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US43313902P 2002-12-13 2002-12-13
PCT/US2003/039606 WO2004055003A1 (en) 2002-12-13 2003-12-12 2-substituted quinazolin-4-ylamine analogues as capsaicin receptor modulators

Publications (1)

Publication Number Publication Date
MXPA05006123A true MXPA05006123A (es) 2005-09-30

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MXPA05006123A MXPA05006123A (es) 2002-12-13 2003-12-12 Analogos de quinazolin-4-ilamina 2-sustituida como moduladores de receptores de capsaicina.

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Country Link
US (2) US7432275B2 (es)
EP (2) EP1569925A1 (es)
JP (2) JP2006515847A (es)
KR (1) KR20050084292A (es)
CN (1) CN1726205A (es)
AR (1) AR042461A1 (es)
AU (2) AU2003300898A1 (es)
BR (1) BR0317168A (es)
CA (2) CA2509233A1 (es)
MX (1) MXPA05006123A (es)
PE (1) PE20040935A1 (es)
TW (1) TW200418480A (es)
WO (2) WO2004055003A1 (es)

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