SE0201635D0 - Novel compounds - Google Patents
Novel compoundsInfo
- Publication number
- SE0201635D0 SE0201635D0 SE0201635A SE0201635A SE0201635D0 SE 0201635 D0 SE0201635 D0 SE 0201635D0 SE 0201635 A SE0201635 A SE 0201635A SE 0201635 A SE0201635 A SE 0201635A SE 0201635 D0 SE0201635 D0 SE 0201635D0
- Authority
- SE
- Sweden
- Prior art keywords
- novel compounds
- useful
- formula
- relates
- present
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
Priority Applications (25)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SE0201635A SE0201635D0 (sv) | 2002-05-30 | 2002-05-30 | Novel compounds |
TW092114174A TW200407305A (en) | 2002-05-30 | 2003-05-26 | Novel compounds |
JP2004509654A JP4485354B2 (ja) | 2002-05-30 | 2003-05-27 | 新規な置換インドール類 |
KR10-2004-7019452A KR20050010507A (ko) | 2002-05-30 | 2003-05-27 | 신규 치환 인돌 |
MXPA04011876A MXPA04011876A (es) | 2002-05-30 | 2003-05-27 | Nuevos indoles sustituidos. |
ES03725970T ES2360936T3 (es) | 2002-05-30 | 2003-05-27 | Indoles sustituidos. |
US10/516,557 US7166607B2 (en) | 2002-05-30 | 2003-05-27 | Substituted indoles |
BR0311494-5A BR0311494A (pt) | 2002-05-30 | 2003-05-27 | Novos indóis substituìdos |
AU2003228201A AU2003228201A1 (en) | 2002-05-30 | 2003-05-27 | Novel substituted indoles |
PL03375111A PL375111A1 (en) | 2002-05-30 | 2003-05-27 | Novel substituted indoles |
RU2004135064/04A RU2288914C2 (ru) | 2002-05-30 | 2003-05-27 | Новые замещенные индолы |
CA002487675A CA2487675A1 (en) | 2002-05-30 | 2003-05-27 | Novel substituted indoles |
AT03725970T ATE501118T1 (de) | 2002-05-30 | 2003-05-27 | Substituierte indole |
DE60336314T DE60336314D1 (de) | 2002-05-30 | 2003-05-27 | Substituierte indole |
PCT/SE2003/000856 WO2003101961A1 (en) | 2002-05-30 | 2003-05-27 | Novel substituted indoles |
CNB038183447A CN100404505C (zh) | 2002-05-30 | 2003-05-27 | 新的取代吲哚 |
EP03725970A EP1513812B1 (en) | 2002-05-30 | 2003-05-27 | Substituted indoles |
UA20041109794A UA79464C2 (en) | 2002-05-30 | 2003-05-27 | Substituted indoles, methods for their production and method for treating disorders mediated by prostaglandin d2 |
NZ536883A NZ536883A (en) | 2002-05-30 | 2003-05-27 | Novel substituted indoles |
MYPI20031973A MY133624A (en) | 2002-05-30 | 2003-05-28 | Thio-substituted indole acetic acid derivatives for the treatment of respiratory disease |
ARP030101932A AR039934A1 (es) | 2002-05-30 | 2003-05-30 | Indoles sustituidos para el tratamiento de desordenes respiratorios |
CO04120052A CO5631431A2 (es) | 2002-05-30 | 2004-11-29 | Indoles sustituidos novedosos |
ZA200409641A ZA200409641B (en) | 2002-05-30 | 2004-11-29 | Novel substituted indoles. |
IS7607A IS7607A (is) | 2002-05-30 | 2004-12-21 | Ný útskipt indól |
NO20045589A NO20045589L (no) | 2002-05-30 | 2004-12-22 | Nye forbindelser |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SE0201635A SE0201635D0 (sv) | 2002-05-30 | 2002-05-30 | Novel compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
SE0201635D0 true SE0201635D0 (sv) | 2002-05-30 |
Family
ID=20288018
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SE0201635A SE0201635D0 (sv) | 2002-05-30 | 2002-05-30 | Novel compounds |
Country Status (25)
Country | Link |
---|---|
US (1) | US7166607B2 (sv) |
EP (1) | EP1513812B1 (sv) |
JP (1) | JP4485354B2 (sv) |
KR (1) | KR20050010507A (sv) |
CN (1) | CN100404505C (sv) |
AR (1) | AR039934A1 (sv) |
AT (1) | ATE501118T1 (sv) |
AU (1) | AU2003228201A1 (sv) |
BR (1) | BR0311494A (sv) |
CA (1) | CA2487675A1 (sv) |
CO (1) | CO5631431A2 (sv) |
DE (1) | DE60336314D1 (sv) |
ES (1) | ES2360936T3 (sv) |
IS (1) | IS7607A (sv) |
MX (1) | MXPA04011876A (sv) |
MY (1) | MY133624A (sv) |
NO (1) | NO20045589L (sv) |
NZ (1) | NZ536883A (sv) |
PL (1) | PL375111A1 (sv) |
RU (1) | RU2288914C2 (sv) |
SE (1) | SE0201635D0 (sv) |
TW (1) | TW200407305A (sv) |
UA (1) | UA79464C2 (sv) |
WO (1) | WO2003101961A1 (sv) |
ZA (1) | ZA200409641B (sv) |
Families Citing this family (97)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TW200307542A (en) | 2002-05-30 | 2003-12-16 | Astrazeneca Ab | Novel compounds |
SE0201635D0 (sv) | 2002-05-30 | 2002-05-30 | Astrazeneca Ab | Novel compounds |
SE0202241D0 (sv) * | 2002-07-17 | 2002-07-17 | Astrazeneca Ab | Novel Compounds |
KR20050111314A (ko) | 2002-12-20 | 2005-11-24 | 암젠 인코포레이션 | 천식 및 알레르기성 염증 조절제들 |
SE0301010D0 (sv) | 2003-04-07 | 2003-04-07 | Astrazeneca Ab | Novel compounds |
SE0301569D0 (sv) * | 2003-05-27 | 2003-05-27 | Astrazeneca Ab | Novel compounds |
SE0302232D0 (sv) * | 2003-08-18 | 2003-08-18 | Astrazeneca Ab | Novel Compounds |
SA04250253B1 (ar) | 2003-08-21 | 2009-11-10 | استرازينيكا ايه بي | احماض فينوكسي اسيتيك مستبدلة باعتبارها مركبات صيدلانية لعلاج الامراض التنفسية مثل الربو ومرض الانسداد الرئوي المزمن |
JP2007508363A (ja) * | 2003-10-14 | 2007-04-05 | オキサジェン リミテッド | Crth2アンタゴニスト活性を有する化合物 |
GB0324763D0 (en) | 2003-10-23 | 2003-11-26 | Oxagen Ltd | Use of compounds in therapy |
SE0303180D0 (sv) * | 2003-11-26 | 2003-11-26 | Astrazeneca Ab | Novel compounds |
DE602005006539D1 (de) | 2004-03-11 | 2008-06-19 | Actelion Pharmaceuticals Ltd | Tetrahydropyridoindolderivate |
US7417063B2 (en) | 2004-04-13 | 2008-08-26 | Bristol-Myers Squibb Company | Bicyclic heterocycles useful as serine protease inhibitors |
AU2005247110B2 (en) | 2004-05-29 | 2010-08-26 | 7Tm Pharma A/S | CRTH2 receptor ligands for medicinal uses |
GB0412914D0 (en) * | 2004-06-10 | 2004-07-14 | Oxagen Ltd | Compounds |
MY144903A (en) * | 2004-06-17 | 2011-11-30 | Novartis Ag | Pyrrolopyridine derivatives and their use as crth2 antagonists |
GB0415320D0 (en) | 2004-07-08 | 2004-08-11 | Astrazeneca Ab | Novel compounds |
GB0418830D0 (en) | 2004-08-24 | 2004-09-22 | Astrazeneca Ab | Novel compounds |
US8273740B2 (en) * | 2004-08-26 | 2012-09-25 | Actelion Pharmaceuticals, Ltd. | 2-sulfanyl-benzoimidazol-1-yi-acetic acid derivatives as CRTH2 antagonists |
CA2581338A1 (en) | 2004-09-21 | 2006-03-30 | Athersys, Inc. | Indole acetic acids exhibiting crth2 receptor antagonism and uses thereof |
ES2314739T3 (es) * | 2004-10-27 | 2009-03-16 | Janssen Pharmaceutica Nv | Derivados de indol como moduladores de receptores de progesterona. |
ATE517085T1 (de) | 2004-11-23 | 2011-08-15 | Astrazeneca Ab | Zur behandlung von atemwegserkrankungen geeignete phenoxyessigsäurederivate |
NZ556657A (en) | 2004-12-27 | 2010-10-29 | Actelion Pharmaceuticals Ltd | 2,3,4,9-tetrahydro-1H-carbazole derivatives as CRTH2 receptor antagonists |
GB0500604D0 (en) | 2005-01-13 | 2005-02-16 | Astrazeneca Ab | Novel process |
JP5064219B2 (ja) | 2005-07-22 | 2012-10-31 | 塩野義製薬株式会社 | Pgd2受容体アンタゴニスト活性を有するアザインドール酸誘導体 |
JP5072594B2 (ja) * | 2005-07-22 | 2012-11-14 | 塩野義製薬株式会社 | Pgd2受容体アンタゴニスト活性を有するインドール誘導体 |
US20070027105A1 (en) | 2005-07-26 | 2007-02-01 | Alza Corporation | Peroxide removal from drug delivery vehicle |
WO2007039736A1 (en) | 2005-10-06 | 2007-04-12 | Astrazeneca Ab | Novel compounds |
TW200745003A (en) | 2005-10-06 | 2007-12-16 | Astrazeneca Ab | Novel compounds |
GB0521275D0 (en) * | 2005-10-19 | 2005-11-30 | Argenta Discovery Ltd | 3-Aminoindole compounds |
GB0524428D0 (en) | 2005-11-30 | 2006-01-11 | 7Tm Pharma As | Medicinal use of receptor ligands |
GB0525143D0 (en) * | 2005-12-09 | 2006-01-18 | Novartis Ag | Organic compounds |
JP2009538289A (ja) | 2006-05-26 | 2009-11-05 | アストラゼネカ・アクチエボラーグ | ビアリールまたはヘテロアリール置換インドール |
SI2037967T1 (sl) | 2006-06-16 | 2017-04-26 | The Trustees Of The University Of Pennsylvania | Antagonisti receptorja za prostaglandin d2 za zdravljenje androgene alopecije |
JP5270542B2 (ja) | 2006-07-22 | 2013-08-21 | オキサジェン リミテッド | Crth2アンタゴニスト活性を有する化合物 |
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EA035752B1 (ru) | 2015-09-15 | 2020-08-05 | Идорсиа Фармасьютиклз Лтд | КРИСТАЛЛИЧЕСКАЯ ФОРМА (S)-2-(8-((5-ХЛОРПИРИМИДИН-2-ИЛ)(МЕТИЛ)-АМИНО)-2-ФТОР-6,7,8,9-ТЕТРАГИДРО-5Н-ПИРИДО[3,2-b]ИНДОЛ-5-ИЛ)УКСУСНОЙ КИСЛОТЫ И СОДЕРЖАЩИЕ ЕЁ ФАРМАЦЕВТИЧЕСКИЕ КОМПОЗИЦИИ |
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TW200307542A (en) | 2002-05-30 | 2003-12-16 | Astrazeneca Ab | Novel compounds |
SE0201635D0 (sv) | 2002-05-30 | 2002-05-30 | Astrazeneca Ab | Novel compounds |
SE0202241D0 (sv) | 2002-07-17 | 2002-07-17 | Astrazeneca Ab | Novel Compounds |
SE0301569D0 (sv) | 2003-05-27 | 2003-05-27 | Astrazeneca Ab | Novel compounds |
SE0302232D0 (sv) | 2003-08-18 | 2003-08-18 | Astrazeneca Ab | Novel Compounds |
SE0303180D0 (sv) | 2003-11-26 | 2003-11-26 | Astrazeneca Ab | Novel compounds |
-
2002
- 2002-05-30 SE SE0201635A patent/SE0201635D0/sv unknown
-
2003
- 2003-05-26 TW TW092114174A patent/TW200407305A/zh unknown
- 2003-05-27 AU AU2003228201A patent/AU2003228201A1/en not_active Abandoned
- 2003-05-27 US US10/516,557 patent/US7166607B2/en not_active Expired - Fee Related
- 2003-05-27 PL PL03375111A patent/PL375111A1/xx not_active Application Discontinuation
- 2003-05-27 WO PCT/SE2003/000856 patent/WO2003101961A1/en active Application Filing
- 2003-05-27 EP EP03725970A patent/EP1513812B1/en not_active Expired - Lifetime
- 2003-05-27 ES ES03725970T patent/ES2360936T3/es not_active Expired - Lifetime
- 2003-05-27 AT AT03725970T patent/ATE501118T1/de not_active IP Right Cessation
- 2003-05-27 JP JP2004509654A patent/JP4485354B2/ja not_active Expired - Fee Related
- 2003-05-27 DE DE60336314T patent/DE60336314D1/de not_active Expired - Lifetime
- 2003-05-27 BR BR0311494-5A patent/BR0311494A/pt not_active IP Right Cessation
- 2003-05-27 NZ NZ536883A patent/NZ536883A/en unknown
- 2003-05-27 MX MXPA04011876A patent/MXPA04011876A/es active IP Right Grant
- 2003-05-27 CN CNB038183447A patent/CN100404505C/zh not_active Expired - Fee Related
- 2003-05-27 KR KR10-2004-7019452A patent/KR20050010507A/ko not_active Application Discontinuation
- 2003-05-27 UA UA20041109794A patent/UA79464C2/uk unknown
- 2003-05-27 CA CA002487675A patent/CA2487675A1/en not_active Abandoned
- 2003-05-27 RU RU2004135064/04A patent/RU2288914C2/ru not_active IP Right Cessation
- 2003-05-28 MY MYPI20031973A patent/MY133624A/en unknown
- 2003-05-30 AR ARP030101932A patent/AR039934A1/es not_active Application Discontinuation
-
2004
- 2004-11-29 CO CO04120052A patent/CO5631431A2/es not_active Application Discontinuation
- 2004-11-29 ZA ZA200409641A patent/ZA200409641B/xx unknown
- 2004-12-21 IS IS7607A patent/IS7607A/is unknown
- 2004-12-22 NO NO20045589A patent/NO20045589L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
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CN1671659A (zh) | 2005-09-21 |
CO5631431A2 (es) | 2006-04-28 |
TW200407305A (en) | 2004-05-16 |
ES2360936T3 (es) | 2011-06-10 |
DE60336314D1 (de) | 2011-04-21 |
RU2004135064A (ru) | 2005-08-10 |
WO2003101961A1 (en) | 2003-12-11 |
MXPA04011876A (es) | 2005-03-31 |
NO20045589L (no) | 2005-02-02 |
IS7607A (is) | 2004-12-21 |
AR039934A1 (es) | 2005-03-09 |
EP1513812B1 (en) | 2011-03-09 |
ZA200409641B (en) | 2006-02-22 |
PL375111A1 (en) | 2005-11-28 |
CN100404505C (zh) | 2008-07-23 |
UA79464C2 (en) | 2007-06-25 |
RU2288914C2 (ru) | 2006-12-10 |
ATE501118T1 (de) | 2011-03-15 |
MY133624A (en) | 2007-11-30 |
BR0311494A (pt) | 2005-03-29 |
KR20050010507A (ko) | 2005-01-27 |
AU2003228201A1 (en) | 2003-12-19 |
EP1513812A1 (en) | 2005-03-16 |
CA2487675A1 (en) | 2003-12-11 |
JP4485354B2 (ja) | 2010-06-23 |
US20050165055A1 (en) | 2005-07-28 |
JP2005538955A (ja) | 2005-12-22 |
NZ536883A (en) | 2006-08-31 |
US7166607B2 (en) | 2007-01-23 |
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