SE0202241D0 - Novel Compounds - Google Patents
Novel CompoundsInfo
- Publication number
- SE0202241D0 SE0202241D0 SE0202241A SE0202241A SE0202241D0 SE 0202241 D0 SE0202241 D0 SE 0202241D0 SE 0202241 A SE0202241 A SE 0202241A SE 0202241 A SE0202241 A SE 0202241A SE 0202241 D0 SE0202241 D0 SE 0202241D0
- Authority
- SE
- Sweden
- Prior art keywords
- novel compounds
- relates
- present
- pharmaceutical compounds
- respiratory disorders
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
- A61K31/405—Indole-alkanecarboxylic acids; Derivatives thereof, e.g. tryptophan, indomethacin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/14—Antitussive agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/16—Central respiratory analeptics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
Priority Applications (27)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SE0202241A SE0202241D0 (sv) | 2002-07-17 | 2002-07-17 | Novel Compounds |
SE0203713A SE0203713D0 (sv) | 2002-07-17 | 2002-12-13 | Novel compounds |
TW092118486A TW200404778A (en) | 2002-07-17 | 2003-07-07 | Novel compounds |
US10/521,325 US7723373B2 (en) | 2002-07-17 | 2003-07-15 | Indole-3-sulphur derivatives |
EP03764279A EP1551802B1 (en) | 2002-07-17 | 2003-07-15 | Indole-3-sulphur derivatives |
JP2004521364A JP4791729B2 (ja) | 2002-07-17 | 2003-07-15 | インドール−3−硫黄誘導体 |
DK03764279.0T DK1551802T3 (da) | 2002-07-17 | 2003-07-15 | Indol-3-svovlderivater |
PCT/SE2003/001216 WO2004007451A1 (en) | 2002-07-17 | 2003-07-15 | Indole-3-sulphur derivatives |
PT03764279T PT1551802E (pt) | 2002-07-17 | 2003-07-15 | Derivados de indole-3-enxofre |
NZ537606A NZ537606A (en) | 2002-07-17 | 2003-07-15 | Indole-2-sulphur derivatives and their use to treat prostaglandin D2 mediated diseases |
CA002492445A CA2492445A1 (en) | 2002-07-17 | 2003-07-15 | Indole-3-sulphur derivatives |
AU2003251260A AU2003251260B2 (en) | 2002-07-17 | 2003-07-15 | Indole-3-sulphur derivatives |
BR0312729-0A BR0312729A (pt) | 2002-07-17 | 2003-07-15 | Novos derivados de indol-3-enxofre |
AT03764279T ATE450506T1 (de) | 2002-07-17 | 2003-07-15 | Indol-3-schwefelderivate |
ES03764279T ES2335491T3 (es) | 2002-07-17 | 2003-07-15 | Derivados de indol-3-azufre. |
SI200331737T SI1551802T1 (sl) | 2002-07-17 | 2003-07-15 | Indol žveplovi derivati |
DE60330372T DE60330372D1 (de) | 2002-07-17 | 2003-07-15 | Indol-3-schwefelderivate |
MXPA05000646A MXPA05000646A (es) | 2002-07-17 | 2003-07-15 | Derivados de indol-3-azufre. |
CNB038199718A CN1279023C (zh) | 2002-07-17 | 2003-07-15 | 吲哚-3-硫衍生物 |
AR20030102585A AR040498A1 (es) | 2002-07-17 | 2003-07-17 | Indoles sustituidos utiles para el tratamiento de enfermedades respiratorias |
IL16612105A IL166121A0 (en) | 2002-07-17 | 2005-01-03 | Indole-3-sulphur derivatives |
ZA200500170A ZA200500170B (en) | 2002-07-17 | 2005-01-07 | Indole-3-sulphur derivatives. |
NO20050828A NO20050828L (no) | 2002-07-17 | 2005-02-16 | lndol-3-svovelderivater |
CY20101100086T CY1109760T1 (el) | 2002-07-17 | 2010-01-28 | Παραγωγα ινδολης-3-θειου |
US12/758,348 US20100197756A1 (en) | 2002-07-17 | 2010-04-12 | Indole-3-Sulphur Derivatives |
JP2010166138A JP2010280680A (ja) | 2002-07-17 | 2010-07-23 | インドール−3−硫黄誘導体 |
JP2011043693A JP2011116770A (ja) | 2002-07-17 | 2011-03-01 | インドール−3−硫黄誘導体 |
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SE0202241A SE0202241D0 (sv) | 2002-07-17 | 2002-07-17 | Novel Compounds |
SE0203713A SE0203713D0 (sv) | 2002-07-17 | 2002-12-13 | Novel compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
SE0202241D0 true SE0202241D0 (sv) | 2002-07-17 |
Family
ID=30117585
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SE0202241A SE0202241D0 (sv) | 2002-07-17 | 2002-07-17 | Novel Compounds |
SE0203713A SE0203713D0 (sv) | 2002-07-17 | 2002-12-13 | Novel compounds |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SE0203713A SE0203713D0 (sv) | 2002-07-17 | 2002-12-13 | Novel compounds |
Country Status (23)
Country | Link |
---|---|
US (2) | US7723373B2 (sv) |
EP (1) | EP1551802B1 (sv) |
JP (3) | JP4791729B2 (sv) |
CN (1) | CN1279023C (sv) |
AR (1) | AR040498A1 (sv) |
AT (1) | ATE450506T1 (sv) |
AU (1) | AU2003251260B2 (sv) |
BR (1) | BR0312729A (sv) |
CA (1) | CA2492445A1 (sv) |
CY (1) | CY1109760T1 (sv) |
DE (1) | DE60330372D1 (sv) |
DK (1) | DK1551802T3 (sv) |
ES (1) | ES2335491T3 (sv) |
IL (1) | IL166121A0 (sv) |
MX (1) | MXPA05000646A (sv) |
NO (1) | NO20050828L (sv) |
NZ (1) | NZ537606A (sv) |
PT (1) | PT1551802E (sv) |
SE (2) | SE0202241D0 (sv) |
SI (1) | SI1551802T1 (sv) |
TW (1) | TW200404778A (sv) |
WO (1) | WO2004007451A1 (sv) |
ZA (1) | ZA200500170B (sv) |
Families Citing this family (80)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SE0201635D0 (sv) | 2002-05-30 | 2002-05-30 | Astrazeneca Ab | Novel compounds |
TW200307542A (en) | 2002-05-30 | 2003-12-16 | Astrazeneca Ab | Novel compounds |
SE0202241D0 (sv) * | 2002-07-17 | 2002-07-17 | Astrazeneca Ab | Novel Compounds |
SE0301010D0 (sv) | 2003-04-07 | 2003-04-07 | Astrazeneca Ab | Novel compounds |
SE0301569D0 (sv) * | 2003-05-27 | 2003-05-27 | Astrazeneca Ab | Novel compounds |
EP1648867B1 (en) | 2003-07-17 | 2013-09-04 | Plexxikon Inc. | Ppar active compounds |
US7348338B2 (en) | 2003-07-17 | 2008-03-25 | Plexxikon, Inc. | PPAR active compounds |
SE0302232D0 (sv) * | 2003-08-18 | 2003-08-18 | Astrazeneca Ab | Novel Compounds |
SA04250253B1 (ar) | 2003-08-21 | 2009-11-10 | استرازينيكا ايه بي | احماض فينوكسي اسيتيك مستبدلة باعتبارها مركبات صيدلانية لعلاج الامراض التنفسية مثل الربو ومرض الانسداد الرئوي المزمن |
JP2007508363A (ja) * | 2003-10-14 | 2007-04-05 | オキサジェン リミテッド | Crth2アンタゴニスト活性を有する化合物 |
SE0303180D0 (sv) * | 2003-11-26 | 2003-11-26 | Astrazeneca Ab | Novel compounds |
DE602005006539D1 (de) | 2004-03-11 | 2008-06-19 | Actelion Pharmaceuticals Ltd | Tetrahydropyridoindolderivate |
GB0412914D0 (en) * | 2004-06-10 | 2004-07-14 | Oxagen Ltd | Compounds |
MY144903A (en) | 2004-06-17 | 2011-11-30 | Novartis Ag | Pyrrolopyridine derivatives and their use as crth2 antagonists |
GB0415320D0 (en) | 2004-07-08 | 2004-08-11 | Astrazeneca Ab | Novel compounds |
GB0418830D0 (en) | 2004-08-24 | 2004-09-22 | Astrazeneca Ab | Novel compounds |
US8273740B2 (en) * | 2004-08-26 | 2012-09-25 | Actelion Pharmaceuticals, Ltd. | 2-sulfanyl-benzoimidazol-1-yi-acetic acid derivatives as CRTH2 antagonists |
CA2581338A1 (en) | 2004-09-21 | 2006-03-30 | Athersys, Inc. | Indole acetic acids exhibiting crth2 receptor antagonism and uses thereof |
ES2314739T3 (es) * | 2004-10-27 | 2009-03-16 | Janssen Pharmaceutica Nv | Derivados de indol como moduladores de receptores de progesterona. |
ATE517085T1 (de) | 2004-11-23 | 2011-08-15 | Astrazeneca Ab | Zur behandlung von atemwegserkrankungen geeignete phenoxyessigsäurederivate |
JP2008521829A (ja) | 2004-11-30 | 2008-06-26 | プレキシコン,インコーポレーテッド | Ppar活性化合物 |
CA2589896A1 (en) * | 2004-11-30 | 2006-06-08 | Plexxikon, Inc. | Indole derivatives for use as ppar active compounds |
NZ556657A (en) | 2004-12-27 | 2010-10-29 | Actelion Pharmaceuticals Ltd | 2,3,4,9-tetrahydro-1H-carbazole derivatives as CRTH2 receptor antagonists |
GB0500604D0 (en) | 2005-01-13 | 2005-02-16 | Astrazeneca Ab | Novel process |
RU2416601C2 (ru) * | 2005-02-25 | 2011-04-20 | Оно Фармасьютикал Ко., Лтд. | Соединение индола и его применение |
GB0505048D0 (en) | 2005-03-11 | 2005-04-20 | Oxagen Ltd | Compounds with PGD antagonist activity |
JP5064219B2 (ja) | 2005-07-22 | 2012-10-31 | 塩野義製薬株式会社 | Pgd2受容体アンタゴニスト活性を有するアザインドール酸誘導体 |
JP5072594B2 (ja) | 2005-07-22 | 2012-11-14 | 塩野義製薬株式会社 | Pgd2受容体アンタゴニスト活性を有するインドール誘導体 |
US20070027105A1 (en) | 2005-07-26 | 2007-02-01 | Alza Corporation | Peroxide removal from drug delivery vehicle |
CA2621406A1 (en) * | 2005-09-07 | 2007-03-15 | Plexxikon, Inc. | Pparactive compounds |
JP2009509932A (ja) * | 2005-09-07 | 2009-03-12 | プレキシコン,インコーポレーテッド | Ppar活性化合物 |
TW200745003A (en) | 2005-10-06 | 2007-12-16 | Astrazeneca Ab | Novel compounds |
WO2007039736A1 (en) | 2005-10-06 | 2007-04-12 | Astrazeneca Ab | Novel compounds |
GB0525143D0 (en) | 2005-12-09 | 2006-01-18 | Novartis Ag | Organic compounds |
GB0526257D0 (en) * | 2005-12-22 | 2006-02-01 | Novartis Ag | Organic compounds |
JP2009538289A (ja) | 2006-05-26 | 2009-11-05 | アストラゼネカ・アクチエボラーグ | ビアリールまたはヘテロアリール置換インドール |
SI2037967T1 (sl) | 2006-06-16 | 2017-04-26 | The Trustees Of The University Of Pennsylvania | Antagonisti receptorja za prostaglandin d2 za zdravljenje androgene alopecije |
JP5270542B2 (ja) | 2006-07-22 | 2013-08-21 | オキサジェン リミテッド | Crth2アンタゴニスト活性を有する化合物 |
EP2316824A1 (en) | 2006-08-07 | 2011-05-04 | Actelion Pharmaceuticals Ltd. | (3-Amino-1,2,3,4-tetrahydro-9H-carbazoI-9-yl)-acetic acid derivates |
PE20090159A1 (es) * | 2007-03-08 | 2009-02-21 | Plexxikon Inc | COMPUESTOS DERIVADOS DE ACIDO INDOL-PROPIONICO COMO MODULADORES PPARs |
UA100983C2 (ru) | 2007-07-05 | 2013-02-25 | Астразенека Аб | Бифенилоксипропановая кислота как модулятор crth2 и интермедиаты |
GB0722055D0 (en) * | 2007-11-09 | 2007-12-19 | Argenta Discovery Ltd | Compounds |
EP2229358B1 (en) | 2007-12-14 | 2011-03-23 | Pulmagen Therapeutics (Asthma) Limited | Indoles and their therapeutic use |
DK2250161T3 (da) * | 2008-01-18 | 2014-01-27 | Atopix Therapeutics Ltd | Forbindelser med CRTH2-antagonistaktivitet |
US7750027B2 (en) | 2008-01-18 | 2010-07-06 | Oxagen Limited | Compounds having CRTH2 antagonist activity |
WO2009093029A1 (en) | 2008-01-22 | 2009-07-30 | Oxagen Limited | Compounds having crth2 antagonist activity |
US20100022613A1 (en) | 2008-01-22 | 2010-01-28 | Oxagen Limited | Compounds Having CRTH2 Antagonist Activity |
TWI469965B (zh) | 2008-12-22 | 2015-01-21 | Ono Pharmaceutical Co | 乙炔基吲哚化合物 |
AU2010270050B9 (en) * | 2009-07-06 | 2013-06-27 | Astrazeneca Ab | Intermediates and processes for the preparation of 4- (acetylamino) ) -3- [ (4-chloro-phenyl) thio] -2-methyl-1H-indole-1-acetic acid |
WO2011055270A1 (en) | 2009-11-04 | 2011-05-12 | Wyeth Llc | Indole based receptor crth2 antagonists |
TW201130810A (en) | 2009-12-23 | 2011-09-16 | Ironwood Pharmaceuticals Inc | CRTH2 modulators |
US20130178475A1 (en) | 2010-03-17 | 2013-07-11 | Ironwood Pharmaceuticals, Inc. | sGC STIMULATORS |
CN102791689B (zh) | 2010-03-22 | 2014-10-29 | 埃科特莱茵药品有限公司 | 3-(杂芳基-氨基)-1,2,3,4-四氢-9h-咔唑衍生物及其作为***素d2受体调节剂的用途 |
EP2583964B1 (en) | 2010-06-21 | 2016-03-23 | ONO Pharmaceutical Co., Ltd. | New crystalline forms of 4,4'-[4-fluoro-7-({4-[4-(3-fluoro-2-methylphenyl)butoxy]phenyl}ethynyl)-2-methyl-1h-indole-1,3-diyl]dibutanoic acid |
CN107021951B (zh) | 2010-06-30 | 2020-10-20 | 赛克里翁治疗有限公司 | sGC刺激物 |
WO2012009134A1 (en) | 2010-07-12 | 2012-01-19 | Ironwood Pharmaceuticals, Inc. | Crth2 modulators |
US20130216552A1 (en) | 2010-07-12 | 2013-08-22 | Ironwood Pharmaceuticals, Inc. | Crth2 modulators |
AU2011326241B2 (en) | 2010-11-09 | 2016-11-17 | Ironwood Pharmaceuticals, Inc. | sGC stimulators |
JP5964945B2 (ja) | 2011-04-14 | 2016-08-03 | アクテリオン ファーマシューティカルズ リミテッドActelion Pharmaceuticals Ltd | 7−(ヘテロアリ−ル−アミノ)−6,7,8,9−テトラヒドロピリド[1,2−a]インド−ル酢酸誘導体及びプロスタグランジンD2受容体調節剤としてのそれらの使用 |
JP6054600B2 (ja) * | 2011-08-11 | 2016-12-27 | 富士通コンポーネント株式会社 | コネクタ |
BR112014014558A8 (pt) | 2011-12-16 | 2017-07-04 | Atopix Therapeutics Ltd | composição farmacêutica, uso de um antagonista de crth2 e de um inibidor de bomba de prótons, e, kit para o tratamento de esofagite eosinofílica |
CN106117194A (zh) | 2011-12-27 | 2016-11-16 | 铁木医药有限公司 | 可用作sgc刺激剂的2‑苄基、3‑(嘧啶‑2‑基)取代的吡唑类 |
CN108938441A (zh) | 2012-03-21 | 2018-12-07 | 宾夕法尼亚大学理事会 | 用于调节毛发生长的组合物和方法 |
WO2014047111A1 (en) | 2012-09-18 | 2014-03-27 | Ironwood Pharmaceuticals, Inc. | Sgc stimulators |
WO2014047325A1 (en) | 2012-09-19 | 2014-03-27 | Ironwood Pharmaceuticals, Inc. | Sgc stimulators |
RS63108B1 (sr) | 2013-03-15 | 2022-04-29 | Cyclerion Therapeutics Inc | Sgc stimulatori |
CN106304835A (zh) | 2013-12-11 | 2017-01-04 | 铁木医药有限公司 | sGC刺激剂 |
US20160324856A1 (en) | 2014-01-13 | 2016-11-10 | Ironwood Pharmaceuticals, Inc. | Use of sgc stimulators for the treatment of neuromuscular disorders |
MX368179B (es) | 2014-03-17 | 2019-09-23 | Idorsia Pharmaceuticals Ltd | Derivados del acido acetico azaindol y su uso como moduladores de receptor de prostaglandina d2. |
EP3119780B1 (en) | 2014-03-18 | 2018-08-29 | Idorsia Pharmaceuticals Ltd | Azaindole acetic acid derivatives and their use as prostaglandin d2 receptor modulators |
GB201407807D0 (en) | 2014-05-02 | 2014-06-18 | Atopix Therapeutics Ltd | Polymorphic form |
GB201407820D0 (en) | 2014-05-02 | 2014-06-18 | Atopix Therapeutics Ltd | Polymorphic form |
JP6624616B2 (ja) | 2014-09-17 | 2019-12-25 | サイクレリオン・セラピューティクス,インコーポレーテッド | sGC刺激剤 |
WO2016044445A2 (en) | 2014-09-17 | 2016-03-24 | Ironwood Pharmaceuticals, Inc. | sGC STIMULATORS |
US10844064B2 (en) | 2014-09-17 | 2020-11-24 | Cyclerion Therapeutics, Inc. | sGC stimulators |
CN108472510A (zh) | 2015-07-30 | 2018-08-31 | 宾夕法尼亚大学理事会 | 用于检测pgd2对毛发生长抑制的易感性的人dp-2基因的单核苷酸多态性等位基因 |
EA035752B1 (ru) | 2015-09-15 | 2020-08-05 | Идорсиа Фармасьютиклз Лтд | КРИСТАЛЛИЧЕСКАЯ ФОРМА (S)-2-(8-((5-ХЛОРПИРИМИДИН-2-ИЛ)(МЕТИЛ)-АМИНО)-2-ФТОР-6,7,8,9-ТЕТРАГИДРО-5Н-ПИРИДО[3,2-b]ИНДОЛ-5-ИЛ)УКСУСНОЙ КИСЛОТЫ И СОДЕРЖАЩИЕ ЕЁ ФАРМАЦЕВТИЧЕСКИЕ КОМПОЗИЦИИ |
JP2019524710A (ja) | 2016-07-07 | 2019-09-05 | アイアンウッド ファーマシューティカルズ インコーポレイテッド | Sgc刺激剤の固体形態 |
CA3029374A1 (en) | 2016-07-07 | 2018-01-11 | Ironwood Pharmaceuticals, Inc. | Phosphorus prodrugs of sgc stimulators |
CN115666621A (zh) | 2020-01-13 | 2023-01-31 | 度勒科特公司 | 具有减少的杂质的持续释放药物递送***及相关方法 |
Family Cites Families (41)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US741360A (en) * | 1899-11-13 | 1903-10-13 | William M Moseley | Toy. |
BE790679A (fr) | 1971-11-03 | 1973-04-27 | Ici Ltd | Derives de l'indole |
JPH0615542B2 (ja) | 1986-07-22 | 1994-03-02 | 吉富製薬株式会社 | ピラゾロピリジン化合物 |
NZ222878A (en) * | 1986-12-17 | 1991-02-26 | Merck Frosst Canada Inc | 3-hetero-substituted-n-benzyl-indole derivatives, and pharmaceutical compositions |
US5095031A (en) * | 1990-08-20 | 1992-03-10 | Abbott Laboratories | Indole derivatives which inhibit leukotriene biosynthesis |
WO1993005020A1 (en) | 1991-09-06 | 1993-03-18 | Merck & Co., Inc. | Indoles as inhibitors of hiv reverse transcriptase |
CA2079374C (en) * | 1991-09-30 | 2003-08-05 | Merck Frosst Canada Incorporated | (bicyclic-azaarylmethoxy)indoles as inhibitors of leukotriene biosynthesis |
FR2692574B1 (fr) | 1992-06-23 | 1995-06-23 | Sanofi Elf | Derives hydroxy-4 benzenethio, leur preparation ainsi que leur utilisation pour la preparation de derives aminoalkoxybenzenesulfonyles. |
HUT74614A (en) | 1993-02-24 | 1997-01-28 | Merck & Co Inc | Nindol derivates suitable for treatment of infection by hiv and pharmaceutical compositions containing them |
US5486525A (en) | 1993-12-16 | 1996-01-23 | Abbott Laboratories | Platelet activating factor antagonists: imidazopyridine indoles |
US5482960A (en) * | 1994-11-14 | 1996-01-09 | Warner-Lambert Company | Nonpeptide endothelin antagonists |
US5567711A (en) | 1995-04-19 | 1996-10-22 | Abbott Laboratories | Indole-3-carbonyl and indole-3-sulfonyl derivatives as platelet activating factor antagonists |
TW472045B (en) * | 1996-09-25 | 2002-01-11 | Astra Ab | Protein kinase C inhibitor compounds, method for their preparation, pharmaceutical composition thereof and intermediate used for their preparation |
AR017256A1 (es) | 1997-08-21 | 2001-09-05 | American Home Prod | Compuestos de indol sustituidos, metodo para la sintesis en fase solida de los mismos, conjuntos de combinacion para ser empleados en dicho metodo, uso delos compuestos para preparar un medicamento y composiciones farmaceuticas que los comprenden |
ES2198033T3 (es) | 1997-12-19 | 2004-01-16 | Eli Lilly And Company | Compuestos de imidazolina hipoglucemicos. |
US6916841B2 (en) * | 1998-02-25 | 2005-07-12 | Genetics Institute, Llc | Inhibitors of phospholipase enzymes |
AU5886500A (en) | 1999-06-23 | 2001-01-09 | Sepracor, Inc. | Indolyl-benzimidazole antibacterials, and methods of use thereof |
WO2001032621A1 (fr) | 1999-10-29 | 2001-05-10 | Wakunaga Pharmaceutical Co., Ltd. | Nouveaux derives d'indole, et medicaments contenant lesdits derives comme principe actif |
CN1615873A (zh) | 1999-12-24 | 2005-05-18 | 阿文蒂斯药物有限公司 | 氮杂吲哚类化合物 |
WO2001092224A1 (en) | 2000-05-31 | 2001-12-06 | Astrazeneca Ab | Indole derivatives with vascular damaging activity |
WO2002000216A1 (en) * | 2000-06-28 | 2002-01-03 | Teva Pharmaceutical Industries Ltd. | Carvedilol |
US6878522B2 (en) * | 2000-07-07 | 2005-04-12 | Baiyong Li | Methods for the identification of compounds useful for the treatment of disease states mediated by prostaglandin D2 |
JP4141954B2 (ja) * | 2001-09-27 | 2008-08-27 | エフ.ホフマン−ラ ロシュ アーゲー | Coxiiインヒビターとしてのインドール誘導体 |
TWI317634B (en) * | 2001-12-13 | 2009-12-01 | Nat Health Research Institutes | Aroyl indoles compounds |
AU2003218962B2 (en) | 2002-02-01 | 2008-09-25 | F. Hoffmann-La Roche Ag | Substituted indoles as alpha-1 agonists |
SE0200356D0 (sv) | 2002-02-05 | 2002-02-05 | Astrazeneca Ab | Novel use |
SE0200411D0 (sv) | 2002-02-05 | 2002-02-05 | Astrazeneca Ab | Novel use |
EP1505061A4 (en) | 2002-05-16 | 2007-08-22 | Shionogi & Co | CONNECTION WITH PGD-2 RECEPTOR ANTAGONISM |
TW200307542A (en) | 2002-05-30 | 2003-12-16 | Astrazeneca Ab | Novel compounds |
SE0201635D0 (sv) | 2002-05-30 | 2002-05-30 | Astrazeneca Ab | Novel compounds |
SE0202241D0 (sv) | 2002-07-17 | 2002-07-17 | Astrazeneca Ab | Novel Compounds |
SE0202463D0 (sv) | 2002-08-14 | 2002-08-14 | Astrazeneca Ab | Novel compounds |
SE0301569D0 (sv) | 2003-05-27 | 2003-05-27 | Astrazeneca Ab | Novel compounds |
SE0302232D0 (sv) | 2003-08-18 | 2003-08-18 | Astrazeneca Ab | Novel Compounds |
JP2007508363A (ja) | 2003-10-14 | 2007-04-05 | オキサジェン リミテッド | Crth2アンタゴニスト活性を有する化合物 |
SE0303180D0 (sv) * | 2003-11-26 | 2003-11-26 | Astrazeneca Ab | Novel compounds |
GB0500604D0 (en) | 2005-01-13 | 2005-02-16 | Astrazeneca Ab | Novel process |
GB2422831A (en) | 2005-02-04 | 2006-08-09 | Oxagen Ltd | Pyrrolopyridines and their use in the treatment of diseases mediated by PGD2 at the CRTH2 receptor |
JP2009538289A (ja) | 2006-05-26 | 2009-11-05 | アストラゼネカ・アクチエボラーグ | ビアリールまたはヘテロアリール置換インドール |
US20090318526A1 (en) | 2006-06-08 | 2009-12-24 | Uno Jacob Weber | Use of cannabinoid receptor agonists as hypothermia inducing drugs for the treatment of ischemia |
JP5237938B2 (ja) | 2006-06-28 | 2013-07-17 | サノフイ | 新規なcxcr2阻害剤 |
-
2002
- 2002-07-17 SE SE0202241A patent/SE0202241D0/sv unknown
- 2002-12-13 SE SE0203713A patent/SE0203713D0/sv unknown
-
2003
- 2003-07-07 TW TW092118486A patent/TW200404778A/zh unknown
- 2003-07-15 ES ES03764279T patent/ES2335491T3/es not_active Expired - Lifetime
- 2003-07-15 WO PCT/SE2003/001216 patent/WO2004007451A1/en active Application Filing
- 2003-07-15 BR BR0312729-0A patent/BR0312729A/pt not_active IP Right Cessation
- 2003-07-15 AU AU2003251260A patent/AU2003251260B2/en not_active Expired - Fee Related
- 2003-07-15 JP JP2004521364A patent/JP4791729B2/ja not_active Expired - Fee Related
- 2003-07-15 PT PT03764279T patent/PT1551802E/pt unknown
- 2003-07-15 CN CNB038199718A patent/CN1279023C/zh not_active Expired - Fee Related
- 2003-07-15 NZ NZ537606A patent/NZ537606A/en unknown
- 2003-07-15 US US10/521,325 patent/US7723373B2/en not_active Expired - Fee Related
- 2003-07-15 CA CA002492445A patent/CA2492445A1/en not_active Abandoned
- 2003-07-15 SI SI200331737T patent/SI1551802T1/sl unknown
- 2003-07-15 EP EP03764279A patent/EP1551802B1/en not_active Expired - Lifetime
- 2003-07-15 DE DE60330372T patent/DE60330372D1/de not_active Expired - Lifetime
- 2003-07-15 DK DK03764279.0T patent/DK1551802T3/da active
- 2003-07-15 MX MXPA05000646A patent/MXPA05000646A/es unknown
- 2003-07-15 AT AT03764279T patent/ATE450506T1/de active
- 2003-07-17 AR AR20030102585A patent/AR040498A1/es not_active Application Discontinuation
-
2005
- 2005-01-03 IL IL16612105A patent/IL166121A0/xx unknown
- 2005-01-07 ZA ZA200500170A patent/ZA200500170B/xx unknown
- 2005-02-16 NO NO20050828A patent/NO20050828L/no not_active Application Discontinuation
-
2010
- 2010-01-28 CY CY20101100086T patent/CY1109760T1/el unknown
- 2010-04-12 US US12/758,348 patent/US20100197756A1/en not_active Abandoned
- 2010-07-23 JP JP2010166138A patent/JP2010280680A/ja not_active Withdrawn
-
2011
- 2011-03-01 JP JP2011043693A patent/JP2011116770A/ja not_active Withdrawn
Also Published As
Publication number | Publication date |
---|---|
JP2010280680A (ja) | 2010-12-16 |
JP2011116770A (ja) | 2011-06-16 |
TW200404778A (en) | 2004-04-01 |
BR0312729A (pt) | 2005-05-10 |
EP1551802B1 (en) | 2009-12-02 |
NO20050828L (no) | 2005-04-05 |
JP4791729B2 (ja) | 2011-10-12 |
SI1551802T1 (sl) | 2010-03-31 |
US20100197756A1 (en) | 2010-08-05 |
MXPA05000646A (es) | 2005-06-02 |
CN1279023C (zh) | 2006-10-11 |
US20060111426A1 (en) | 2006-05-25 |
IL166121A0 (en) | 2006-01-15 |
AR040498A1 (es) | 2005-04-06 |
EP1551802A1 (en) | 2005-07-13 |
ES2335491T3 (es) | 2010-03-29 |
CY1109760T1 (el) | 2014-09-10 |
CA2492445A1 (en) | 2004-01-22 |
JP2005537265A (ja) | 2005-12-08 |
US7723373B2 (en) | 2010-05-25 |
AU2003251260A1 (en) | 2004-02-02 |
NZ537606A (en) | 2006-08-31 |
DE60330372D1 (de) | 2010-01-14 |
WO2004007451A1 (en) | 2004-01-22 |
ZA200500170B (en) | 2006-02-22 |
AU2003251260B2 (en) | 2007-04-26 |
ATE450506T1 (de) | 2009-12-15 |
CN1678579A (zh) | 2005-10-05 |
PT1551802E (pt) | 2010-02-02 |
DK1551802T3 (da) | 2010-03-15 |
SE0203713D0 (sv) | 2002-12-13 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
SE0203713D0 (sv) | Novel compounds | |
TW200407305A (en) | Novel compounds | |
TW200510301A (en) | Novel compounds | |
TW200510303A (en) | Novel compounds | |
SE0303180D0 (sv) | Novel compounds | |
SE0301010D0 (sv) | Novel compounds | |
TW200612892A (en) | Novel compounds | |
SE0301009D0 (sv) | Novel compounds | |
MX2007011847A (es) | Derivados de pirimidindiona como antagonistas del receptor de procineticina 2. | |
EA200900828A1 (ru) | Соединения и композиции в качестве ингибиторов активности каннабиноидного рецептора 1 | |
TW200732296A (en) | Novel compounds | |
NO20052884L (no) | Substituerte indolpyridinforbindelser som anti-infeksjonsmidler. | |
MY153719A (en) | Prokineticin 1 receptor antagonists | |
DE602006010738D1 (de) | Pyrroloä2,3-cüpyridinderivate | |
MX2007011698A (es) | Derivados de oxindol sustituido, medicamentos que contienen dichos derivados y uso de los mismos. | |
ATE467632T1 (de) | Pyrroloä2,3-büpyridinderivate als modulatoren des h3-rezeptors | |
TW200745039A (en) | Isotopically substituted pantoprazole | |
MY141528A (en) | Anilinopyrazole derivatives useful for the treatment of diabetes | |
UA106200C2 (uk) | Заміщені похідні оксіндолу та їхнє застосування для лікування захворювань, залежних від вазопресину | |
DE60316128D1 (de) | N-sulfonylurea-apoptosis-förderer | |
ATE486078T1 (de) | 5,6-disubstituierte oxadiazolopyrazine und thiadiazolopyrazine als liganden des cxc- chemokinrezeptors | |
EA200602081A1 (ru) | Пиридиновые производные алкилоксиндолов в качестве агентов, активных в отношении рецептора 5-нт7 | |
EA200602080A1 (ru) | Пиперазиновые производные алкилоксиндолов | |
UA84701C2 (ru) | Замещенные индолы, способ их получения, их использования | |
SE0301798D0 (sv) | New use IV |