UA100983C2 - Бифенилоксипропановая кислота как модулятор crth2 и интермедиаты - Google Patents

Бифенилоксипропановая кислота как модулятор crth2 и интермедиаты

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Publication number
UA100983C2
UA100983C2 UAA200913443A UAA200913443A UA100983C2 UA 100983 C2 UA100983 C2 UA 100983C2 UA A200913443 A UAA200913443 A UA A200913443A UA A200913443 A UAA200913443 A UA A200913443A UA 100983 C2 UA100983 C2 UA 100983C2
Authority
UA
Ukraine
Prior art keywords
biphenyloxypropanoic
intermediates
acid
crth2
modulator
Prior art date
Application number
UAA200913443A
Other languages
English (en)
Ukrainian (uk)
Inventor
Роджер Віктор Боннерт
Тімоті Джон Лукер
Аніл Патель
Аарон Ріґбі
Original Assignee
Астразенека Аб
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39942682&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UA100983(C2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Астразенека Аб filed Critical Астразенека Аб
Publication of UA100983C2 publication Critical patent/UA100983C2/ru

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    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
    • C07D295/182—Radicals derived from carboxylic acids
    • C07D295/192—Radicals derived from carboxylic acids from aromatic carboxylic acids
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
    • C07D295/182—Radicals derived from carboxylic acids

Abstract

Изобретение касается амидных соединений, полезных в качестве фармацевтических препаратов для лечения респираторных расстройств, например астмы, ринита и COPD.
UAA200913443A 2007-07-05 2008-01-07 Бифенилоксипропановая кислота как модулятор crth2 и интермедиаты UA100983C2 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US94801207P 2007-07-05 2007-07-05
PCT/GB2008/050525 WO2009004379A1 (en) 2007-07-05 2008-07-01 Novel compounds 951: a biphenyloxypropanoic acid as crth2 modulator and intermediates

Publications (1)

Publication Number Publication Date
UA100983C2 true UA100983C2 (ru) 2013-02-25

Family

ID=39942682

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA200913443A UA100983C2 (ru) 2007-07-05 2008-01-07 Бифенилоксипропановая кислота как модулятор crth2 и интермедиаты

Country Status (30)

Country Link
US (1) US8507544B2 (ru)
EP (1) EP2173730B1 (ru)
JP (1) JP5368438B2 (ru)
KR (1) KR20100039326A (ru)
CN (1) CN101796042B (ru)
AR (1) AR067461A1 (ru)
AU (1) AU2008272690B2 (ru)
BR (1) BRPI0813992A2 (ru)
CA (1) CA2691615A1 (ru)
CL (1) CL2008001982A1 (ru)
CO (1) CO6270211A2 (ru)
CY (1) CY1114804T1 (ru)
DK (1) DK2173730T3 (ru)
EC (1) ECSP109848A (ru)
ES (1) ES2442523T3 (ru)
HK (1) HK1143140A1 (ru)
HR (1) HRP20140004T1 (ru)
MY (1) MY153957A (ru)
NZ (1) NZ582192A (ru)
PE (2) PE20090475A1 (ru)
PL (1) PL2173730T3 (ru)
PT (1) PT2173730E (ru)
RS (1) RS53129B (ru)
SA (1) SA08290406B1 (ru)
SI (1) SI2173730T1 (ru)
TW (1) TWI453017B (ru)
UA (1) UA100983C2 (ru)
UY (1) UY31208A1 (ru)
WO (1) WO2009004379A1 (ru)
ZA (1) ZA200909226B (ru)

Families Citing this family (28)

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SE0301010D0 (sv) * 2003-04-07 2003-04-07 Astrazeneca Ab Novel compounds
SE0301009D0 (sv) * 2003-04-07 2003-04-07 Astrazeneca Ab Novel compounds
SA04250253B1 (ar) * 2003-08-21 2009-11-10 استرازينيكا ايه بي احماض فينوكسي اسيتيك مستبدلة باعتبارها مركبات صيدلانية لعلاج الامراض التنفسية مثل الربو ومرض الانسداد الرئوي المزمن
GB0415320D0 (en) * 2004-07-08 2004-08-11 Astrazeneca Ab Novel compounds
GB0418830D0 (en) * 2004-08-24 2004-09-22 Astrazeneca Ab Novel compounds
GB0422057D0 (en) * 2004-10-05 2004-11-03 Astrazeneca Ab Novel compounds
SI1817282T1 (sl) 2004-11-23 2011-10-28 Astrazeneca Ab Derivati fenoksiocetne kisline, uporabni za zdravljenje respiratornih bolezni
JP5155171B2 (ja) 2005-10-06 2013-02-27 アストラゼネカ・アクチエボラーグ 新規化合物
TW200745003A (en) 2005-10-06 2007-12-16 Astrazeneca Ab Novel compounds
WO2007052023A2 (en) * 2005-11-05 2007-05-10 Astrazeneca Ab Novel compounds
ES2380683T3 (es) * 2005-12-15 2012-05-17 Astrazeneca Ab Difenil-éteres, -amidas, -sulfuros y - metanos sustituidos para el tratamiento de la enfermedad respiratoria
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