PL207570A1 - Sposob wytwarzania nowych pochodnych 3-(1-pirazolilo)-pirydazyny - Google Patents

Sposob wytwarzania nowych pochodnych 3-(1-pirazolilo)-pirydazyny

Info

Publication number
PL207570A1
PL207570A1 PL20757078A PL20757078A PL207570A1 PL 207570 A1 PL207570 A1 PL 207570A1 PL 20757078 A PL20757078 A PL 20757078A PL 20757078 A PL20757078 A PL 20757078A PL 207570 A1 PL207570 A1 PL 207570A1
Authority
PL
Poland
Prior art keywords
pirazolyl
pyridazine
new derivatives
making new
making
Prior art date
Application number
PL20757078A
Other languages
English (en)
Other versions
PL111252B1 (en
Original Assignee
Richter Gedeon Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Richter Gedeon Vegyeszet filed Critical Richter Gedeon Vegyeszet
Publication of PL207570A1 publication Critical patent/PL207570A1/pl
Publication of PL111252B1 publication Critical patent/PL111252B1/pl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
PL1978207570A 1977-06-13 1978-06-12 Process for preparing novel derivatives of 3-/1-pyrazolylo/-pyridazine PL111252B1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU77GO1373A HU175471B (hu) 1977-06-13 1977-06-13 Sposob poluchenija novykh proizvodnykh 3-skobka-1-pirazolil-skobka zakryta-piridazina

Publications (2)

Publication Number Publication Date
PL207570A1 true PL207570A1 (pl) 1979-05-21
PL111252B1 PL111252B1 (en) 1980-08-30

Family

ID=10996834

Family Applications (1)

Application Number Title Priority Date Filing Date
PL1978207570A PL111252B1 (en) 1977-06-13 1978-06-12 Process for preparing novel derivatives of 3-/1-pyrazolylo/-pyridazine

Country Status (25)

Country Link
US (1) US4251658A (pl)
JP (1) JPS5416487A (pl)
AT (1) AT357548B (pl)
AU (1) AU521394B2 (pl)
BE (1) BE867967A (pl)
BG (1) BG28709A3 (pl)
CA (1) CA1095912A (pl)
CH (1) CH638202A5 (pl)
CS (1) CS204029B2 (pl)
DD (1) DD140043A5 (pl)
DE (1) DE2825906A1 (pl)
DK (1) DK263078A (pl)
ES (1) ES470750A1 (pl)
FI (1) FI64156C (pl)
FR (1) FR2394542A1 (pl)
GB (1) GB1603958A (pl)
HU (1) HU175471B (pl)
IL (1) IL54816A (pl)
IT (1) IT1098216B (pl)
NL (1) NL7806380A (pl)
NO (1) NO149210C (pl)
PL (1) PL111252B1 (pl)
SE (1) SE437517B (pl)
SU (2) SU797577A3 (pl)
YU (1) YU140078A (pl)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU176100B (en) * 1977-10-25 1980-12-28 Gyogyszerkutato Intezet Process for preparing new 3-/1-pyrazolyl/-pyridazine derivatives
DE2935359A1 (de) * 1979-09-01 1981-03-26 Basf Ag, 67063 Ludwigshafen 6-imidazolyl-3-hydrazino-pyridazine
DE3130251A1 (de) * 1981-07-31 1983-02-17 A. Nattermann & Cie GmbH, 5000 Köln 6-(4-((omega)-(1-imidazolyl)-alkyl)-phenyl)-3-oxo -2,3,4,5-tetrahydro-pyridazine und deren saeureadditionssalze, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische praeparate
US4353905A (en) * 1981-09-17 1982-10-12 Warner-Lambert Company Substituted 4,5-dihydro-6-[4-(1H-imidazol-1-yl)phenyl]-3(2H)-pyridazinones and 6-[4-(1H-imidazol-1-yl)phenyl]-3(2H)-pyridazinones
US4590194A (en) * 1981-10-05 1986-05-20 Sterling Drug Inc. 3-[methyl or dimethyl)amino]-6-(pyridinyl)pyridazines and their cardiotonic use
US4503056A (en) * 1982-03-02 1985-03-05 Abbott Laboratories 1-(Pyridazinyl)pyrazoline derivatives
DE3825867A1 (de) * 1988-03-04 1989-09-14 Bayer Ag Heterocyclisch substituierte sulfonylaminoazole und ihre verwendung als herbizide
US5536701A (en) * 1994-10-11 1996-07-16 Monsanto Company 3-pyrazolyloxypyridazines, herbicidal compositions and uses thereof
EP1565150A1 (fr) * 2002-11-20 2005-08-24 L'oreal Utilisation d'un compose pyrazolcarboxamide pour stimuler la pousse des fibres keratiniques et/ou freiner leur chute
FR2847160A1 (fr) * 2002-11-20 2004-05-21 Oreal Composition capillaire contenant un compose pyrasol-carboxamide, son utilisation pour stimuler la pousse des cheveux et/ou freiner leur chute
RU2442775C2 (ru) * 2005-07-04 2012-02-20 Хай Пойнт Фармасьютикалс, ЛЛС Антагонисты гистаминовых н3-рецепторов
CN103110635A (zh) 2005-07-04 2013-05-22 海波因特制药有限责任公司 组胺h3受体拮抗剂
EP2038256A1 (en) * 2006-05-23 2009-03-25 TransTech Pharma, Inc 6- (4-cyclopropylpiperazin-1-yl) -2 ' -methyl- [3, 4 ']-bipyridine and its use as a medicament
EA016026B1 (ru) * 2006-05-29 2012-01-30 ХАЙ ПОЙНТ ФАРМАСЬЮТИКАЛЗ, ЭлЭлСи 3-(1,3-бензодиоксол-5-ил)-6-(4-циклопропилпиперазин-1-ил)пиридазин, его соли и сольваты и его применение в качестве антагониста н3 рецептора гистамина
EP2014656A3 (en) * 2007-06-11 2011-08-24 High Point Pharmaceuticals, LLC New heteocyclic h3 antagonists
AR081331A1 (es) 2010-04-23 2012-08-08 Cytokinetics Inc Amino- pirimidinas composiciones de las mismas y metodos para el uso de los mismos
EP2560488B1 (en) 2010-04-23 2015-10-28 Cytokinetics, Inc. Certain amino-pyridines and amino-triazines, compositions thereof, and methods for their use
AR081626A1 (es) * 2010-04-23 2012-10-10 Cytokinetics Inc Compuestos amino-piridazinicos, composiciones farmaceuticas que los contienen y uso de los mismos para tratar trastornos musculares cardiacos y esqueleticos

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1595920B2 (de) * 1964-11-04 1978-08-10 Merck Patent Gmbh, 6100 Darmstadt 4-(co-Piperazinoalkyl)-pyrazole, ihre Salze und Verfahren zu ihrer Herstellung
JPS5831347B2 (ja) * 1975-09-05 1983-07-05 中外製薬株式会社 ピラゾリルピリダジンユウドウタイノ セイホウ

Also Published As

Publication number Publication date
FR2394542B1 (pl) 1980-12-05
IT7824490A0 (it) 1978-06-13
CA1095912A (en) 1981-02-17
CS204029B2 (en) 1981-03-31
BE867967A (fr) 1978-12-11
NO149210C (no) 1984-03-07
AT357548B (de) 1980-07-10
DD140043A5 (de) 1980-02-06
IL54816A0 (en) 1978-07-31
BG28709A3 (en) 1980-06-16
US4251658A (en) 1981-02-17
SE7806576L (sv) 1978-12-14
NO149210B (no) 1983-11-28
PL111252B1 (en) 1980-08-30
CH638202A5 (de) 1983-09-15
SU797577A3 (ru) 1981-01-15
FI64156C (fi) 1983-10-10
YU140078A (en) 1983-01-21
HU175471B (hu) 1980-08-28
FR2394542A1 (fr) 1979-01-12
AU521394B2 (en) 1982-04-01
NL7806380A (nl) 1978-12-15
FI781856A (fi) 1978-12-14
ATA414478A (de) 1979-12-15
SU860703A1 (ru) 1981-08-30
DK263078A (da) 1978-12-14
FI64156B (fi) 1983-06-30
DE2825906A1 (de) 1979-01-18
NO782043L (no) 1978-12-14
ES470750A1 (es) 1979-01-16
JPS5416487A (en) 1979-02-07
GB1603958A (en) 1981-12-02
JPS569506B2 (pl) 1981-03-02
IT1098216B (it) 1985-09-07
SE437517B (sv) 1985-03-04
AU3683678A (en) 1979-12-06
IL54816A (en) 1981-09-13

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