PL205135A1 - Sposob wytwarzania pochodnych 3-(tiometylo)-cefalosporyn - Google Patents

Sposob wytwarzania pochodnych 3-(tiometylo)-cefalosporyn

Info

Publication number
PL205135A1
PL205135A1 PL20513578A PL20513578A PL205135A1 PL 205135 A1 PL205135 A1 PL 205135A1 PL 20513578 A PL20513578 A PL 20513578A PL 20513578 A PL20513578 A PL 20513578A PL 205135 A1 PL205135 A1 PL 205135A1
Authority
PL
Poland
Prior art keywords
cephalosporine
thiomethyl
derivatives
production
Prior art date
Application number
PL20513578A
Other languages
English (en)
Other versions
PL122152B1 (en
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/862,871 external-priority patent/US4144391A/en
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of PL205135A1 publication Critical patent/PL205135A1/pl
Publication of PL122152B1 publication Critical patent/PL122152B1/pl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/207-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/247-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/36Methylene radicals, substituted by sulfur atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PL1978205135A 1977-03-07 1978-03-07 Process for preparing derivatives of 3-/thiomethyl/ cephalosporinsnov PL122152B1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US77501877A 1977-03-07 1977-03-07
US05/862,871 US4144391A (en) 1977-03-07 1977-12-27 Cephalosporin displacement reaction

Publications (2)

Publication Number Publication Date
PL205135A1 true PL205135A1 (pl) 1979-06-04
PL122152B1 PL122152B1 (en) 1982-06-30

Family

ID=27118982

Family Applications (1)

Application Number Title Priority Date Filing Date
PL1978205135A PL122152B1 (en) 1977-03-07 1978-03-07 Process for preparing derivatives of 3-/thiomethyl/ cephalosporinsnov

Country Status (30)

Country Link
JP (1) JPS53130689A (pl)
AT (1) AT366696B (pl)
AU (1) AU515428B2 (pl)
BG (1) BG31379A3 (pl)
CA (1) CA1083141A (pl)
CH (1) CH637964A5 (pl)
CS (1) CS205115B2 (pl)
CY (1) CY1196A (pl)
DD (1) DD137356A5 (pl)
DE (1) DE2809058A1 (pl)
DK (1) DK97378A (pl)
EG (1) EG13454A (pl)
ES (1) ES467637A1 (pl)
FI (1) FI69309C (pl)
FR (1) FR2383189A1 (pl)
GB (1) GB1597036A (pl)
GR (1) GR68893B (pl)
HK (1) HK49083A (pl)
HU (1) HU179967B (pl)
IE (1) IE46437B1 (pl)
IL (1) IL54181A (pl)
IT (1) IT1093504B (pl)
MX (1) MX5142E (pl)
NL (1) NL190703C (pl)
NZ (1) NZ186610A (pl)
PH (1) PH14596A (pl)
PL (1) PL122152B1 (pl)
PT (1) PT67732A (pl)
SE (1) SE437991B (pl)
YU (1) YU51478A (pl)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5543043A (en) * 1978-09-22 1980-03-26 Sankyo Co Ltd Preparation of 3-substituted thiomethylcephalosporin derivative
US4576937A (en) * 1984-02-29 1986-03-18 Smithkline Beckman Corporation 7-D-Mandelamido-3(1-sulfomethyltetrazol-5-yl)thiomethyl-3-cephem-4-carboxylic acid monosodium salt
GB8519606D0 (en) * 1985-08-05 1985-09-11 Fujisawa Pharmaceutical Co 3 7-d substituted-3-cephem compounds
JP2503500B2 (ja) * 1986-04-14 1996-06-05 萬有製薬株式会社 新規セフアロスポリン誘導体及びその製造法
JPS62281881A (ja) * 1986-09-08 1987-12-07 Sankyo Co Ltd 3−置換チオメチルセフアロスポリン誘導体の製法
EP2539348A4 (en) * 2010-02-26 2013-07-24 Gary Igor Dmitrienko CEPHALOSPORIN DERIVATIVES AS BETA LACTAMASE HEMMER AND COMPOSITIONS THEREFOR AND METHOD FOR THEIR USE
GB201818410D0 (en) * 2018-11-12 2018-12-26 Imperial Innovations Ltd Compounds

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3641021A (en) * 1969-04-18 1972-02-08 Lilly Co Eli 3 7-(ring-substituted) cephalosporin compounds
JPS5116436B1 (pl) * 1971-05-31 1976-05-24
JPS5143785A (en) * 1974-10-11 1976-04-14 Yamanouchi Pharma Co Ltd Shinsefuarosuhorinkanrenkagobutsuno goseiho
JPS612674B2 (pl) * 1974-06-20 1986-01-27 Meiji Seika Co
CA1100129A (en) * 1974-08-02 1981-04-28 William H.W. Lunn Cephalosporin compounds
FI761035A (pl) * 1975-04-21 1976-10-22 Erba Carlo Spa

Also Published As

Publication number Publication date
MX5142E (es) 1983-03-30
GR68893B (pl) 1982-03-15
HU179967B (en) 1983-01-28
NL7802376A (nl) 1978-09-11
GB1597036A (en) 1981-09-03
NZ186610A (en) 1979-11-01
SE7802530L (sv) 1978-09-08
NL190703B (nl) 1994-02-01
CA1083141A (en) 1980-08-05
FI69309B (fi) 1985-09-30
IE46437B1 (en) 1983-06-15
JPH025758B2 (pl) 1990-02-05
HK49083A (en) 1983-11-04
AT366696B (de) 1982-04-26
DE2809058A1 (de) 1978-09-14
CY1196A (en) 1983-12-31
DD137356A5 (de) 1979-08-29
DK97378A (da) 1978-09-08
NL190703C (nl) 1994-07-01
SE437991B (sv) 1985-03-25
JPS53130689A (en) 1978-11-14
IT1093504B (it) 1985-07-19
IL54181A (en) 1981-03-31
CS205115B2 (en) 1981-04-30
IT7820912A0 (it) 1978-03-06
DE2809058C2 (pl) 1989-02-09
PH14596A (en) 1981-10-02
FR2383189B1 (pl) 1981-06-26
IL54181A0 (en) 1978-06-15
FR2383189A1 (fr) 1978-10-06
YU51478A (en) 1982-10-31
PT67732A (en) 1978-04-01
ATA150778A (de) 1981-09-15
FI69309C (fi) 1986-01-10
BG31379A3 (en) 1981-12-15
ES467637A1 (es) 1980-04-01
EG13454A (en) 1981-12-31
IE780453L (en) 1978-09-07
AU3382878A (en) 1979-09-06
AU515428B2 (en) 1981-04-02
CH637964A5 (en) 1983-08-31
PL122152B1 (en) 1982-06-30
FI780716A (fi) 1978-09-08

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