NO325187B1 - Hydrobromidsalt og hemisuksinatsalt av et isotiazol-4-karboksamid samt anvendelse og fremstilling derav, og farmasoytisk preparat - Google Patents

Hydrobromidsalt og hemisuksinatsalt av et isotiazol-4-karboksamid samt anvendelse og fremstilling derav, og farmasoytisk preparat Download PDF

Info

Publication number: NO325187B1
Authority: NO; Norway
Prior art keywords: salt; isothiazole; ureido; benzyloxy; difluoro
Prior art date: 2000-11-28

Application number

NO20032388A

Other languages

English (en)

Norwegian (no)

Other versions

NO20032388L (no

NO20032388D0 (no

Inventor

Thomas G Gant

Glenn Robert Williams

Original Assignee

Pfizer Prod Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-11-28

Filing date

2003-05-27

Publication date

2008-02-11

2003-05-27 Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc

2003-05-27 Publication of NO20032388D0 publication Critical patent/NO20032388D0/no

2003-07-18 Publication of NO20032388L publication Critical patent/NO20032388L/no

2008-02-11 Publication of NO325187B1 publication Critical patent/NO325187B1/no

Links

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- C07D275/03—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C—CHEMISTRY; METALLURGY
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- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Thiazole And Isothizaole Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

NO20032388A 2000-11-28 2003-05-27 Hydrobromidsalt og hemisuksinatsalt av et isotiazol-4-karboksamid samt anvendelse og fremstilling derav, og farmasoytisk preparat NO325187B1 (no)

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US25351300P	2000-11-28	2000-11-28
PCT/IB2001/002193 WO2002044158A1 (en)	2000-11-28	2001-11-19	Salts of a isothiazole-4-carboxamide and their use as anti-hyperproliferation agents

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NO20032388D0 NO20032388D0 (no)	2003-05-27
NO20032388L NO20032388L (no)	2003-07-18
NO325187B1 true NO325187B1 (no)	2008-02-11

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EP (1)	EP1337521B1 (pt)
JP (2)	JP2004514714A (pt)
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EP1158985B1 (en)	1999-01-13	2011-12-28	Bayer HealthCare LLC	OMEGA-CARBOXY ARYL SUBSTITUTED DIPHENYL UREAS AS p38 KINASE INHIBITORS
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US20030216396A1 (en)	2002-02-11	2003-11-20	Bayer Corporation	Pyridine, quinoline, and isoquinoline N-oxides as kinase inhibitors
PT1478358E (pt)	2002-02-11	2013-09-11	Bayer Healthcare Llc	Tosilato de sorafenib para o tratamento de doenças caracterizadas por angiogénese anormal
JP4511352B2 (ja) *	2002-07-25	2010-07-28	ファイザー・インク	抗癌薬として有用なイソチアゾール誘導体
CN1681495B (zh) *	2002-08-19	2010-05-12	辉瑞产品公司	用于治疗过度增生性疾病的组合物
JP2007511203A (ja)	2003-05-20	2007-05-10	バイエル、ファーマシューテイカルズ、コーポレイション	キナーゼ阻害活性を有するジアリール尿素
DE602004010407T2 (de)	2003-07-23	2008-10-16	Bayer Pharmaceuticals Corp., West Haven	Fluorsubstituierter omega-carboxyaryldiphenylharnstoff zur behandlung und prävention von krankheiten und leiden
AU2004287416C1 (en) *	2003-10-27	2010-09-09	Merck Sharp & Dohme Corp.	CCR-2 antagonist salt
WO2005061519A1 (en)	2003-12-19	2005-07-07	Takeda San Diego, Inc.	Kinase inhibitors
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ATE517885T1 (de)	2004-04-30	2011-08-15	Bayer Healthcare Llc	Substituierte pyrazolyl-harnstoff-derivate zur behandlung von krebs
TW200538104A (en) *	2004-05-17	2005-12-01	Pfizer Prod Inc	Phenyl derivatives for the treatment of abnormal cell growth
EP1778669A2 (en)	2004-08-18	2007-05-02	Takeda San Diego, Inc.	Kinase inhibitors
DE602005023333D1 (de)	2004-10-15	2010-10-14	Takeda Pharmaceutical	Kinaseinhibitoren
US8119655B2 (en)	2005-10-07	2012-02-21	Takeda Pharmaceutical Company Limited	Kinase inhibitors
PL2044043T5 (pl)	2006-06-16	2022-05-02	H. Lundbeck A/S	Bromowodorek 1-[2-(2,4-dimetylofenylosulfanylo)fenylo]piperazyny jako związek o połączonym działaniu wychwytu zwrotnego serotoniny i działaniu na 5-ht3 i 5-ht1a do leczenia upośledzenia funckji poznawczych
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GEP20135728B (en)	2006-10-09	2013-01-25	Takeda Pharmaceuticals Co	Kinase inhibitors
MX2010001636A (es)	2007-08-14	2010-03-15	Hoffmann La Roche	Derivados de pirazolo[3,4-d]-pirimidina como agentes antiproliferativos.
WO2011073521A1 (en)	2009-12-15	2011-06-23	Petri Salven	Methods for enriching adult-derived endothelial progenitor cells and uses thereof
JP2013538191A (ja)	2010-07-23	2013-10-10	トラスティーズオブボストンユニバーシティ	病的血管新生および腫瘍細胞侵襲性の阻害のための治療法としてならびに分子イメージングおよび標的化送達のための抗ＤＥｓｕｐＲ阻害剤
BR112015021334B1 (pt) *	2013-03-14	2020-04-07	Panoptica Inc	formulação ocular tópica em suspenão e uso da mesma para tratamento e/ou melhora de uma doença do segmento posterior do olho
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2001
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2003
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Also Published As

Publication number	Publication date
EA200300424A1 (ru)	2003-10-30
CA2430065A1 (en)	2002-06-06
TNSN01167A1 (fr)	2005-11-10
HUP0302553A2 (hu)	2003-11-28
BR0115621A (pt)	2003-09-02
DE60123461D1 (de)	2006-11-09
JP4971946B2 (ja)	2012-07-11
US6831091B2 (en)	2004-12-14
AU2002214204B2 (en)	2007-05-24
SI1337521T1 (sl)	2006-12-31
GEP20053652B (en)	2005-11-10
EE200300247A (et)	2003-10-15
PA8533801A1 (es)	2002-10-31
OA12532A (en)	2006-06-02
ECSP034628A (es)	2003-07-25
AP2001002358A0 (en)	2001-12-31
CA2430065C (en)	2008-05-20
ES2271086T3 (es)	2007-04-16
US20020151573A1 (en)	2002-10-17
ATE340786T1 (de)	2006-10-15
IS6788A (is)	2003-04-14
CR6963A (es)	2003-11-25
CZ20031315A3 (cs)	2004-04-14
GT200100237A (es)	2002-07-03
MA26960A1 (fr)	2004-12-20
EP1337521A1 (en)	2003-08-27
KR20050116401A (ko)	2005-12-12
BG107752A (bg)	2004-01-30
CN1476439A (zh)	2004-02-18
SK5862003A3 (en)	2004-05-04
TWI287542B (en)	2007-10-01
EP1337521B1 (en)	2006-09-27
UY27039A1 (es)	2002-07-31
JP2008056692A (ja)	2008-03-13
KR20030059275A (ko)	2003-07-07
ZA200303341B (en)	2004-04-30
WO2002044158A1 (en)	2002-06-06
PL362079A1 (en)	2004-10-18
DK1337521T3 (da)	2007-01-29
PE20020591A1 (es)	2002-07-06
NO20032388L (no)	2003-07-18
NZ525788A (en)	2004-11-26
JP2004514714A (ja)	2004-05-20
HK1059085A1 (en)	2004-06-18
NO20032388D0 (no)	2003-05-27
AU1420402A (en)	2002-06-11
EA005859B1 (ru)	2005-06-30
IL155371A0 (en)	2003-11-23
HUP0302553A3 (en)	2009-03-30
MY136686A (en)	2008-11-28
HN2001000268A (es)	2002-01-30
HRP20030408A2 (en)	2003-08-31
UA74221C2 (uk)	2005-11-15
CY1106240T1 (el)	2011-06-08
MXPA03004714A (es)	2003-08-19
SV2002000748A (es)	2002-12-02
YU36403A (sh)	2006-08-17
CN1231474C (zh)	2005-12-14
PT1337521E (pt)	2006-12-29
DE60123461T2 (de)	2007-02-15
DOP2001000288A (es)	2002-12-15
AR031512A1 (es)	2003-09-24

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