NO148488C - Analogifremgangsmaate til fremstilling av terapeutisk aktive acyl-benzimidazol-2-derivater - Google Patents

Analogifremgangsmaate til fremstilling av terapeutisk aktive acyl-benzimidazol-2-derivater

Info

Publication number: NO148488C
Authority: NO; Norway
Prior art keywords: benzimidazole; derivatives; preparation; therapeutic active; active acyl
Prior art date: 1976-08-27

Application number

NO772962A

Other languages

English (en)

Other versions

NO148488B (no

NO772962L (no

Inventor

Ernst Habicht

Pier Giorgio Ferrini

Alfred Sallmann

Original Assignee

Ciba Geigy Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1976-08-27

Filing date

1977-08-26

Publication date

1983-10-19

1977-08-26 Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag

1978-02-28 Publication of NO772962L publication Critical patent/NO772962L/no

1983-07-11 Publication of NO148488B publication Critical patent/NO148488B/no

1983-10-19 Publication of NO148488C publication Critical patent/NO148488C/no

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
- C07D235/12—Radicals substituted by oxygen atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, ***e
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/14—Decongestants or antiallergics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
- C07C205/45—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by at least one doubly—bound oxygen atom, not being part of a —CHO group
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/45—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by condensation
- C07C45/46—Friedel-Crafts reactions
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
- C07C49/76—Ketones containing a keto group bound to a six-membered aromatic ring
- C07C49/80—Ketones containing a keto group bound to a six-membered aromatic ring containing halogen
- C07C49/807—Ketones containing a keto group bound to a six-membered aromatic ring containing halogen all halogen atoms bound to the ring
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
- C07C49/76—Ketones containing a keto group bound to a six-membered aromatic ring
- C07C49/80—Ketones containing a keto group bound to a six-membered aromatic ring containing halogen
- C07C49/813—Ketones containing a keto group bound to a six-membered aromatic ring containing halogen polycyclic

NO772962A 1976-08-27 1977-08-26 Analogifremgangsmaate til fremstilling av terapeutisk aktive acyl-benzimidazol-2-derivater NO148488C (no)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
LU75684A LU75684A1 (no)	1976-08-27	1976-08-27

Publications (3)

Publication Number	Publication Date
NO772962L NO772962L (no)	1978-02-28
NO148488B NO148488B (no)	1983-07-11
NO148488C true NO148488C (no)	1983-10-19

Family

ID=19728336

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO772962A NO148488C (no)	1976-08-27	1977-08-26	Analogifremgangsmaate til fremstilling av terapeutisk aktive acyl-benzimidazol-2-derivater

Country Status (32)

Country	Link
US (3)	US4141982A (no)
JP (1)	JPS5328172A (no)
AR (6)	AR224610A1 (no)
AT (1)	AT359060B (no)
AU (1)	AU517209B2 (no)
BE (1)	BE858157A (no)
CA (1)	CA1098526A (no)
CH (8)	CH631973A5 (no)
DD (1)	DD132735A5 (no)
DE (1)	DE2737462A1 (no)
DK (1)	DK381277A (no)
ES (7)	ES461906A1 (no)
FI (1)	FI68230C (no)
FR (1)	FR2362841A1 (no)
GB (2)	GB1595914A (no)
GR (1)	GR72908B (no)
HK (1)	HK93784A (no)
HU (2)	HU186765B (no)
IE (1)	IE45665B1 (no)
IL (1)	IL52820A (no)
LU (1)	LU75684A1 (no)
MY (1)	MY8500936A (no)
NL (1)	NL7709471A (no)
NO (1)	NO148488C (no)
NZ (1)	NZ185035A (no)
OA (1)	OA05753A (no)
PL (4)	PL105527B1 (no)
PT (1)	PT66947B (no)
SE (1)	SE434397B (no)
SG (1)	SG70784G (no)
SU (7)	SU882410A3 (no)
ZA (1)	ZA775182B (no)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4312873A (en) *	1978-09-29	1982-01-26	Syntex (U.S.A.) Inc.	5(6)-Benzene ring substituted benzimidazole-2-carbamate derivatives having anthelmintic activity
US4322431A (en) *	1979-02-09	1982-03-30	Ciba-Geigy Corporation	Pharmaceutical preparations containing benzimidazole 2-derivatives
US4492708A (en) *	1982-09-27	1985-01-08	Eli Lilly And Company	Antiviral benzimidazoles
DE3772966D1 (de) *	1987-02-03	1991-10-17	Grace W R & Co	Biozide.
JPH04197628A (ja) *	1990-11-28	1992-07-17	Sekisui Chem Co Ltd	壁パネルの製造方法
US5216003A (en) *	1992-01-02	1993-06-01	G. D. Searle & Co.	Diacid-containing benzimidazole compounds for treatment of neurotoxic injury
FR2751649B1 (fr) *	1996-07-26	1998-08-28	Adir	Nouveaux derives de benzimidazole, de benzoxazole et de benzothiazole, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
US9663703B2 (en)	2014-04-25	2017-05-30	James George Clements	Method and compositions for enhanced oil recovery
CN109467512B (zh) *	2018-12-18	2021-06-08	苏州开元民生科技股份有限公司	一种3,4-二氨基-二苯甲酮的合成方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB766749A (en)	1954-01-11	1957-01-23	Aschaffenburger Zellstoffwerke	Benzimidazole cobalamines and process for their preparation and separation
US3318889A (en) *	1963-10-14	1967-05-09	S B Penick & Company	2-benzimidazole carbamates
DE1923481A1 (de) *	1969-05-08	1970-11-12	Hoechst Ag	Verfahren zur Herstellung von Amiden und Estern der 1-Hydroxy-benzimidazol-2-carbonsaeure
NL7013343A (no) *	1969-09-26	1971-03-30
BE759237A (fr) *	1969-11-21	1971-05-01	Montedison Spa	Procede de preparation d'amides a partir de composes heterocycliques azotes
BE792402A (fr) *	1971-12-07	1973-06-07	Ciba Geigy	Composes heterocycliques azotes et medicaments anthelminthiqueset antimicrobiens qui en contiennent
US4026936A (en) *	1975-08-07	1977-05-31	Hoffmann-La Roche Inc.	Anthelmintic pyridine and thiazole substituted benzimidazole carbamates

1976
- 1976-08-27 LU LU75684A patent/LU75684A1/xx unknown
1977
- 1977-08-01 HU HU811133A patent/HU186765B/hu unknown
- 1977-08-01 HU HU77CI1761A patent/HU180700B/hu unknown
- 1977-08-18 US US05/825,630 patent/US4141982A/en not_active Expired - Lifetime
- 1977-08-19 DE DE19772737462 patent/DE2737462A1/de not_active Ceased
- 1977-08-22 PT PT66947A patent/PT66947B/pt unknown
- 1977-08-23 DD DD7700200697A patent/DD132735A5/xx unknown
- 1977-08-24 OA OA56266A patent/OA05753A/xx unknown
- 1977-08-25 PL PL1977200449A patent/PL105527B1/pl not_active IP Right Cessation
- 1977-08-25 CH CH1040177A patent/CH631973A5/de not_active IP Right Cessation
- 1977-08-25 FI FI772521A patent/FI68230C/fi not_active IP Right Cessation
- 1977-08-25 CA CA285,456A patent/CA1098526A/en not_active Expired
- 1977-08-25 PL PL1977206452A patent/PL108853B1/pl unknown
- 1977-08-25 GB GB17219/80A patent/GB1595914A/en not_active Expired
- 1977-08-25 GB GB35710/77A patent/GB1595913A/en not_active Expired
- 1977-08-25 IL IL52820A patent/IL52820A/xx unknown
- 1977-08-25 PL PL1977211468A patent/PL110215B1/pl unknown
- 1977-08-25 FR FR7725938A patent/FR2362841A1/fr active Granted
- 1977-08-25 PL PL1977213906A patent/PL112665B1/pl unknown
- 1977-08-26 ZA ZA00775182A patent/ZA775182B/xx unknown
- 1977-08-26 ES ES461906A patent/ES461906A1/es not_active Expired
- 1977-08-26 AT AT620677A patent/AT359060B/de not_active IP Right Cessation
- 1977-08-26 NO NO772962A patent/NO148488C/no unknown
- 1977-08-26 DK DK381277A patent/DK381277A/da not_active Application Discontinuation
- 1977-08-26 NZ NZ185035A patent/NZ185035A/xx unknown
- 1977-08-26 GR GR54237A patent/GR72908B/el unknown
- 1977-08-26 IE IE1779/77A patent/IE45665B1/en unknown
- 1977-08-26 AU AU28255/77A patent/AU517209B2/en not_active Expired
- 1977-08-26 SU SU772513755A patent/SU882410A3/ru active
- 1977-08-26 NL NL7709471A patent/NL7709471A/xx not_active Application Discontinuation
- 1977-08-26 SE SE7709615A patent/SE434397B/xx not_active IP Right Cessation
- 1977-08-26 BE BE180470A patent/BE858157A/xx not_active IP Right Cessation
- 1977-08-27 JP JP10312777A patent/JPS5328172A/ja active Granted
- 1977-08-29 AR AR268986A patent/AR224610A1/es active
1978
- 1978-06-26 SU SU782627856A patent/SU745365A3/ru active
- 1978-07-13 ES ES471688A patent/ES471688A1/es not_active Expired
- 1978-07-13 ES ES471687A patent/ES471687A1/es not_active Expired
- 1978-07-13 ES ES471686A patent/ES471686A1/es not_active Expired
- 1978-07-13 ES ES471690A patent/ES471690A1/es not_active Expired
- 1978-07-13 ES ES471689A patent/ES471689A1/es not_active Expired
- 1978-11-16 SU SU782685604A patent/SU923368A3/ru active
- 1978-11-16 SU SU782685606A patent/SU831074A3/ru active
- 1978-11-16 SU SU782685605A patent/SU843744A3/ru active
- 1978-11-20 US US05/962,426 patent/US4213993A/en not_active Expired - Lifetime
1979
- 1979-01-15 SU SU792708672A patent/SU888819A3/ru active
- 1979-01-15 SU SU792707652A patent/SU784766A3/ru active
- 1979-01-18 AR AR275220A patent/AR231536A1/es active
- 1979-01-18 AR AR275221A patent/AR225889A1/es active
- 1979-01-18 AR AR275222A patent/AR227621A1/es active
- 1979-01-18 AR AR275219A patent/AR222318A1/es active
- 1979-01-18 AR AR275218A patent/AR230990A1/es active
- 1979-04-02 ES ES79479189A patent/ES8106706A1/es not_active Expired
- 1979-12-28 US US06/107,980 patent/US4344957A/en not_active Expired - Lifetime
1981
- 1981-09-30 CH CH630581A patent/CH631974A5/de not_active IP Right Cessation
- 1981-10-01 CH CH630481A patent/CH632749A5/de not_active IP Right Cessation
- 1981-10-13 CH CH653681A patent/CH632253A5/de not_active IP Right Cessation
- 1981-10-13 CH CH653881A patent/CH631975A5/de not_active IP Right Cessation
1982
- 1982-03-23 CH CH177582A patent/CH634305A5/de not_active IP Right Cessation
- 1982-07-27 CH CH455582A patent/CH637120A5/de not_active IP Right Cessation
- 1982-07-27 CH CH455682A patent/CH637121A5/de not_active IP Right Cessation
1984
- 1984-10-05 SG SG707/84A patent/SG70784G/en unknown
- 1984-11-29 HK HK937/84A patent/HK93784A/xx unknown
1985
- 1985-12-30 MY MY936/85A patent/MY8500936A/xx unknown

Also Published As

Publication number	Publication date
HK93784A (en)	1984-12-07
JPS5328172A (en)	1978-03-16
IL52820A (en)	1981-02-27
AT359060B (de)	1980-10-27
PL200449A1 (pl)	1978-05-22
AR230990A1 (es)	1984-08-31
ES471687A1 (es)	1979-10-16
BE858157A (fr)	1978-02-27
AR222318A1 (es)	1981-05-15
CA1098526A (en)	1981-03-31
DD132735A5 (de)	1978-10-25
CH631974A5 (de)	1982-09-15
FI68230B (fi)	1985-04-30
HU186765B (en)	1985-09-30
LU75684A1 (no)	1978-04-13
PL105527B1 (pl)	1979-10-31
US4213993A (en)	1980-07-22
HU180700B (en)	1983-04-29
ES471688A1 (es)	1979-10-16
PT66947A (en)	1977-09-01
PL112665B1 (en)	1980-10-31
CH634305A5 (de)	1983-01-31
ES461906A1 (es)	1978-12-01
MY8500936A (en)	1985-12-31
ZA775182B (en)	1978-07-26
SE7709615L (sv)	1978-02-28
NZ185035A (en)	1981-05-29
FI772521A (fi)	1978-02-28
SU784766A3 (ru)	1980-11-30
US4344957A (en)	1982-08-17
NL7709471A (nl)	1978-03-01
FR2362841A1 (fr)	1978-03-24
AU517209B2 (en)	1981-07-16
IE45665L (en)	1978-02-27
GR72908B (no)	1984-01-04
NO148488B (no)	1983-07-11
IE45665B1 (en)	1982-10-20
AR231536A1 (es)	1984-12-28
NO772962L (no)	1978-02-28
CH632749A5 (de)	1982-10-29
CH631973A5 (de)	1982-09-15
ES479189A0 (es)	1981-09-01
ES471686A1 (es)	1979-10-16
SE434397B (sv)	1984-07-23
IL52820A0 (en)	1977-10-31
ES471689A1 (es)	1979-10-16
PL110215B1 (en)	1980-07-31
ATA620677A (de)	1980-03-15
ES471690A1 (es)	1979-10-16
GB1595914A (en)	1981-08-19
CH632253A5 (de)	1982-09-30
SU882410A3 (ru)	1981-11-15
SU888819A3 (ru)	1981-12-07
SG70784G (en)	1985-03-15
FR2362841B1 (no)	1981-11-20
ES8106706A1 (es)	1981-09-01
CH637120A5 (de)	1983-07-15
CH637121A5 (de)	1983-07-15
SU745365A3 (ru)	1980-06-30
DK381277A (da)	1978-02-28
AR227621A1 (es)	1982-11-30
PT66947B (en)	1979-02-07
GB1595913A (en)	1981-08-19
CH631975A5 (de)	1982-09-15
SU843744A3 (ru)	1981-06-30
US4141982A (en)	1979-02-27
AR225889A1 (es)	1982-05-14
SU831074A3 (ru)	1981-05-15
AU2825577A (en)	1979-03-01
OA05753A (fr)	1981-05-31
DE2737462A1 (de)	1978-03-02
PL108853B1 (en)	1980-05-31
JPS6231706B2 (no)	1987-07-09
AR224610A1 (es)	1981-12-30
SU923368A3 (ru)	1982-04-23
FI68230C (fi)	1985-08-12

Publication	Publication Date	Title
NO147243C (no)	1983-03-02	Analogifremgangsmaate for fremstilling av terapeutisk aktive ftalanderivater
NO149586C (no)	1984-05-16	Analogifremgangsmaate for fremstilling av terapeutisk aktive polypeptider
NO151321C (no)	1985-03-20	Analogifremgangsmaate for fremstilling av terapeutisk aktive karbostyrilderivater
NO151463C (no)	1985-04-17	Analogifremgangsmaate for fremstilling av terapeutisk aktive kinazolinderivater
NO148148C (no)	1983-08-17	Fremgangsmaate til fremstilling av terapeutisk aktive 4-hydroksy-2-pyrrolidinonderivater
NO151411C (no)	1985-04-10	Analogifremgangsmaate for fremstilling av terapeutisk aktive 1-aryloksy-2-hydroksy-3-alkylenaminopropan-derivater
NO148453C (no)	1983-10-12	Analogifremgangsmaate for fremstilling av terapeutisk aktive spirohydantoinderivater
NO800881L (no)	1980-09-29	Analogifremgangsmaate for fremstilling av terapeutisk aktive kinolonderivater
NO144848C (no)	1981-11-25	Analogifremgangsmaate til fremstilling av terapeutisk virksomme 4-hydroksyfenylalkanolamin-derivater
NO148777C (no)	1984-01-25	Analogifremgangsmaate for fremstilling av terapeutisk aktive antrakinon-derivater
NO150044C (no)	1984-08-22	Analogifremgangsmaate for fremstilling av terapeutisk aktive tetrazol-derivater
NO145198C (no)	1982-02-03	Analogifremgangsmaate til fremstilling av terapeutisk aktivt 1,2-benzisotia-zolinon-3
NO149313C (no)	1984-03-28	Analogifremgangsmaate for fremstilling av terapeutisk aktive pyridobenzodiazepiner
NO145951C (no)	1982-06-30	Analogifremgangsmaate for fremstilling av terapeutisk aktive imidazolinderivater
NO149037C (no)	1984-02-01	Analogifremgangsmaate for fremstilling av terapeutisk aktive pyridobenzodiazepiner
NO148291C (no)	1983-09-14	Analogifremgangsmaate til fremstilling av terapeutisk aktive basisk substituerte teofyllinderivater
NO148488C (no)	1983-10-19	Analogifremgangsmaate til fremstilling av terapeutisk aktive acyl-benzimidazol-2-derivater
NO145163C (no)	1982-01-27	Analogifremgangsmaate til fremstilling av terapeutisk aktive antitumorglykosider
NO151660C (no)	1985-05-15	Analogifremgangsmaate til fremstilling av terapeutisk aktive imidazolderivater.
NO143903C (no)	1981-05-06	Analogifremgangsmaate for fremstilling av terapeutisk aktive 5-fluorpyrimidin-4-on-derivater
NO780644L (no)	1978-08-25	Fremgangsmaate til fremstilling av terapeutisk virksomme 9-hydroksyetoksymetylguanin-derivater
NO152172C (no)	1985-08-14	Analogifremgangsmaate for fremstilling av terapeutisk aktive spiro-kinolyl-hydantoin-derivater
NO146600C (no)	1982-11-03	Analogifremgangsmaate til fremstilling av terapeutisk aktive imidazolderivater
NO147273C (no)	1983-03-09	Analogifremgangsmaate til fremstilling av terapeutisk aktive cykloheksadien-derivater
NO152556C (no)	1985-10-16	Analogifremgangsmaate for fremstilling av terapeutisk aktive antracen-biskarbonylhydrazoner