MX9400206A - Derivados de vinil-azaindol, proceso para su preparacion y composiciones farmaceuticas que los contienen. - Google Patents

Derivados de vinil-azaindol, proceso para su preparacion y composiciones farmaceuticas que los contienen.

Info

Publication number
MX9400206A
MX9400206A MX9400206A MX9400206A MX9400206A MX 9400206 A MX9400206 A MX 9400206A MX 9400206 A MX9400206 A MX 9400206A MX 9400206 A MX9400206 A MX 9400206A MX 9400206 A MX9400206 A MX 9400206A
Authority
MX
Mexico
Prior art keywords
azaindol
vinyl
derivatives
contain
preparation
Prior art date
Application number
MX9400206A
Other languages
English (en)
Inventor
Felicita Greco
Franco Buzzetti
Angelo Crugnola
Dario Ballinari
Original Assignee
Erba Carlo Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Carlo Spa filed Critical Erba Carlo Spa
Publication of MX9400206A publication Critical patent/MX9400206A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Abstract

La presente invención se relaciona a nuevos derivados de vinilen-azaindol, a un proceso para su preparación, a composiciones farmacéuticas que los contienen y a su uso como agentes terapéuticos. La presente invención incluye todos los posibles isómeros, esteroisómeros, en particular los isómeros Z-y E- y mezclas de los mismos, así como los metabólicos y precursores metabólicos o bioprecursores (también conocidos como profármacos).
MX9400206A 1992-12-23 1994-01-03 Derivados de vinil-azaindol, proceso para su preparacion y composiciones farmaceuticas que los contienen. MX9400206A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB929226855A GB9226855D0 (en) 1992-12-23 1992-12-23 Vinylene-azaindole derivatives and process for their preparation

Publications (1)

Publication Number Publication Date
MX9400206A true MX9400206A (es) 1994-07-29

Family

ID=10727139

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9400206A MX9400206A (es) 1992-12-23 1994-01-03 Derivados de vinil-azaindol, proceso para su preparacion y composiciones farmaceuticas que los contienen.

Country Status (24)

Country Link
US (1) US5397787A (es)
EP (1) EP0626963B1 (es)
JP (1) JP3507497B2 (es)
KR (1) KR950700296A (es)
CN (1) CN1093707A (es)
AT (1) ATE181074T1 (es)
AU (1) AU670488B2 (es)
CA (1) CA2126228A1 (es)
DE (1) DE69325262T2 (es)
DK (1) DK0626963T3 (es)
ES (1) ES2134926T3 (es)
FI (1) FI943838A0 (es)
GB (1) GB9226855D0 (es)
GR (1) GR3030941T3 (es)
HU (1) HUT67431A (es)
IL (1) IL108087A (es)
MX (1) MX9400206A (es)
MY (1) MY109695A (es)
NZ (1) NZ259330A (es)
PL (1) PL304894A1 (es)
RU (1) RU94040390A (es)
TW (1) TW296383B (es)
WO (1) WO1994014808A1 (es)
ZA (1) ZA939578B (es)

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